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Chinese Academy of Sciences Institutional Repositories Grid
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昆明植物研究所 [77]
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Discovery of a potent PROTAC degrader for RNA demethylase FTO as antileukemic therapy
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2024, 卷号: 14, 期号: 12, 页码: 5382-5392
作者:
Liu, Lu
;
Qiu, Yuanlai
;
Suo, Yuying
;
Tong, Siyao
;
Wang, Yiqing
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2025/04/01
N 6-Methyladenosine
FTO
PROTAC
RNA epigenetics
Antileukemia
19
F qNMR based pharmacokinetics, metabolism and mass balance studies of SARS-CoV-2-3CL protease inhibitor simnotrelvir (SIM0417) in humans
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2024, 页码: 11
作者:
Wang, Ze-yu
;
Ren, Yong-mei
;
Hu, Shu-wei
;
Zhang, Nai-xia
;
Dong, Meng-xiao
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/11/05
COVID-19
simnotrelvir
F-19 qNMR
pharmacokinetics
metabolism
mass balance.
Devonian sea surface temperature and paleoecology changes constrained by in situ oxygen isotopes of fish fossils
期刊论文
OAI收割
PALAEOGEOGRAPHY PALAEOCLIMATOLOGY PALAEOECOLOGY, 2024, 卷号: 639, 页码: 12
作者:
Lu, Chang
;
Cui, Xin-Dong
;
Chen, Jun
;
Cui, Ze-Xian
;
Zhu, Min
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2024/06/05
Paleotemperature
Paleoecology
SIMS
Oxygen isotope
Devonian
Fish enamel
Devonian sea surface temperature and paleoecology changes constrained by in situ oxygen isotopes of fish fossils
期刊论文
OAI收割
PALAEOGEOGRAPHY PALAEOCLIMATOLOGY PALAEOECOLOGY, 2024, 卷号: 639, 页码: 12
作者:
Lu, Chang
;
Cui, Xin-Dong
;
Chen, Jun
;
Cui, Ze-Xian
;
Zhu, Min
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2024/09/12
Paleotemperature
Paleoecology
SIMS
Oxygen isotope
Devonian
Fish enamel
Structure-Activity Relationships of 2-(Arylthio)benzoic Acid FTO Inhibitors
期刊论文
OAI收割
ISRAEL JOURNAL OF CHEMISTRY, 2024, 页码: 13
作者:
Yan, Chao
;
Zhang, Qian
;
Xiao, Pan
;
Xie, Xinyun
;
Li, Ming
  |  
收藏
  |  
浏览/下载:66/0
  |  
提交时间:2024/03/25
RNA modification
m(6)A
FTO
anticancer
Chemical Inhibitors Targeting the Oncogenic m
6
A Modifying Proteins
期刊论文
OAI收割
ACCOUNTS OF CHEMICAL RESEARCH, 2023, 卷号: 56, 期号: 21, 页码: 3010-3022
作者:
Huang, Yue
;
Xia, Wenyang
;
Dong, Ze
;
Yang, Cai-Guang
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2023/12/11
Trapped and Leaking Energetic Particles in Injection Flux Tubes of Saturn's Magnetosphere
期刊论文
OAI收割
GEOPHYSICAL RESEARCH LETTERS, 2023, 卷号: 50, 期号: 19, 页码: 10
作者:
Yin, Ze-Fan
;
Sun, Yi-Xin
;
Zhou, Xu-Zhi
;
Pan, Dong-Xiao
;
Yao, Zhong-Hua
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2023/12/29
interchange injection
flux tube
energetic particles
Saturn's magnetosphere
magnetic gradient drift
particle trapping
Design, synthesis, and biological evaluation of novel spirocyclic compounds as potential anti-glioblastoma agents
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 258, 页码: 22
作者:
Zhu, Heping
;
Song, Xiaomin
;
Pan, Yihui
;
Li, Ming
;
Chen, Liang
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收藏
  |  
浏览/下载:31/0
  |  
提交时间:2023/10/17
Glioblastoma
Spirocyclic compounds
Drug design
Antiproliferation
Rational Design of RNA Demethylase FTO Inhibitors with Enhanced Antileukemia Drug-Like Properties
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 22
作者:
Xiao, Pan
;
Duan, Zongliang
;
Liu, Zeyu
;
Chen, Liang
;
Zhang, Deyan
  |  
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2023/10/17
A Virtual Ultrasonography Simulator for Skill Training Using Magnetic-Inertial Probe Tracking
期刊论文
OAI收割
IEEE-ASME TRANSACTIONS ON MECHATRONICS, 2023, 页码: 10
作者:
Wang, Heng
;
Dong, Shuda
;
Yang, Qi
;
Han, Jiancheng
;
He, Ze'an
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2023/11/17