中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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上海药物研究所 [88]
西北高原生物研究所 [18]
中国科学院大学 [4]
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期刊论文 [109]
会议论文 [1]
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2020 [5]
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Discovery of a potent and orally bioavailable 3,3-dimethyl-2-oxoindoline STING inhibitor
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2026, 卷号: 301, 页码: 18
作者:
Li, Wenxin
;
Wang, Xiyuan
;
Zang, Shumin
;
Zhou, Rongyao
;
Zhou, Hongfei
  |  
收藏
  |  
Discovery of isoindoline-2(1
H
)-carboxamide STING inhibitors as anti-inflammatory agents
期刊论文
OAI收割
MOLECULAR DIVERSITY, 2025, 页码: 13
作者:
Zhou, Xiaoqian
;
Zang, Shumin
;
Yao, Shanyan
;
Zhou, Hongfei
;
Wang, Xiyuan
  |  
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  |  
Discovery of 3,4-dihydroisoquinoline-2(1H)-carboxamide STING inhibitors as anti-inflammatory agents
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 297, 页码: 20
作者:
Zhou, Xiaoqian
;
Yue, Hangtian
;
Wang, Xiyuan
;
Zang, Shumin
;
Li, Han
  |  
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  |  
Discovery of indole derivatives as STING degraders
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 294, 页码: 21
作者:
An, Yuxiang
  |  
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  |  
Dual targeting of VEGFR2 and CSF1R with SYHA1813 confers novel strategy for treating both BRAF wild-type and mutant melanoma
期刊论文
OAI收割
CANCER CELL INTERNATIONAL, 2025, 卷号: 25, 期号: 1, 页码: 12
作者:
Shi, Wenhao
;
Tang, Haotian
;
Tong, Linjiang
;
Song, Peiran
;
Huang, Yuqing
  |  
收藏
  |  
Discovery of a non-nucleotide stimulator of interferon genes (STING) agonist with systemic antitumor effect
期刊论文
OAI收割
MEDCOMM, 2025, 卷号: 6, 期号: 1, 页码: e70001
作者:
Wang, Xiyuan
;
Zhan, Zhengsheng
;
Wang, Zhen
;
Zhang, Yan
;
Zhao, Kaiyan
  |  
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  |  
Synthesis and evaluation of hybrid molecules as RIPK1 and HDACs dual inhibitors
期刊论文
OAI收割
JOURNAL OF MOLECULAR STRUCTURE, 2024, 卷号: 1318, 页码: 13
作者:
Tang, Mingze
;
Zhou, Xuan
;
Shen, Qianqian
;
Fang, Chen
;
Peng, Xia
  |  
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  |  
Design and synthesis of pyridazin-4-one derivatives as necroptosis inhibitors
期刊论文
OAI收割
ARCHIV DER PHARMAZIE, 2024, 页码: 16
作者:
An, Yuxiang
;
Peng, Xia
;
Wang, Tianchen
;
Liu, Kaiyuan
;
Feng, Dazhi
  |  
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  |  
Design, synthesis, and structure-activity relationship studies of 6,7-dihydro-5
H
-pyrrolo[1,2-
b
][1,2,4]triazole derivatives as necroptosis inhibitors
期刊论文
OAI收割
RSC MEDICINAL CHEMISTRY, 2024, 卷号: 15, 期号: 7, 页码: 2514-2526
作者:
Jin, Zechen
;
Dai, Yang
;
Ji, Yinchun
;
Peng, Xia
;
Duan, Wenhu
  |  
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  |  
Discovery and optimization of 3-(indolin-5-yloxy)pyridin-2-amine derivatives as potent necroptosis inhibitors
期刊论文
OAI收割
ARCHIV DER PHARMAZIE, 2024, 页码: 21
作者:
Lan, Yaohan
;
Ji, Yinchun
;
Peng, Xia
  |  
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