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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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上海药物研究所 [20]
中国科学院大学 [1]
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OAI收割 [20]
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期刊论文 [21]
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2025 [1]
2023 [2]
2022 [2]
2020 [1]
2019 [4]
2018 [3]
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Discovery of Novel Tridentate Alkenyl Diacid Derivatives as Potent ATP Citrate Lyase Inhibitors for the Treatment of Hepatocellular Carcinoma
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 15, 页码: 15598-15616
作者:
Yang, Yurou
;
Zhai, Jimao
;
Wang, Fan
;
Song, Gaolei
;
Xu, Honghong
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Design, Synthesis, and Pharmacological Evaluation of Isoindoline Analogues as New HPK1 Inhibitors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 23, 页码: 16201-16221
作者:
Xie, Chenghu
;
Liu, Bo
;
Song, Zilan
;
Yang, Ye
;
Dai, Mengdi
  |  
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  |  
Degradation of Cyclin-Dependent Kinase 9/Cyclin T1 by Optimized Microtubule-Associated Protein 1 Light Chain 3 Beta-Recruiting Coumarin Analogs
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 17
作者:
Zeng, Yanping
;
Xiao, Jian
;
Xu, Yuanxin
;
Wei, Fan
;
Tian, Lina
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The HDAC inhibitor GCJ-490A suppresses c-Met expression through IKK? and overcomes gefitinib resistance in non-small cell lung cancer
期刊论文
OAI收割
CANCER BIOLOGY & MEDICINE, 2022, 卷号: 19, 期号: 8, 页码: 1172-1192
作者:
He, Ting
;
Gao, Yinglei
;
Fang, Yanfen
;
Zhang, Yangming
;
Zhang, Shuwei
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F-18-FDG PET as an imaging biomarker for the response to FGFR-targeted therapy of cancer cells via FGFR-initiated mTOR/HK2 axis
期刊论文
OAI收割
THERANOSTICS, 2022, 卷号: 12, 期号: 14, 页码: 6395-6408
作者:
Jiang, Yuchen
;
Zeng, Qinghe
;
Jiang, Qinghui
;
Peng, Xia
;
Gao, Jing
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Design, Synthesis, and Biological Evaluation of HSP90 Inhibitor-SN38 Conjugates for Targeted Drug Accumulation
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 10, 页码: 5421-5441
作者:
Zhu, Shulei
;
Shen, Qianqian
;
Gao, Yinglei
;
Wang, Lei
;
Fang, Yanfen
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Discovery of a series of dimethoxybenzene FGFR inhibitors with 5H-pyrrolo[2,3-b]pyrazine scaffold: structure-activity relationship, crystal structural characterization and and in vivo study
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2019, 卷号: 9, 期号: 2, 页码: 351-368
作者:
Wei, Peng
;
Liu, Bo
;
Wang, Ruifeng
;
Gao, Yinglei
;
Li, Lanlan
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Simultaneous inhibition of PI3K alpha and CDK4/6 synergistically suppresses KRAS-mutated non-small cell lung cancer
期刊论文
OAI收割
CANCER BIOLOGY & MEDICINE, 2019, 卷号: 16, 期号: 1, 页码: 66-+
作者:
Wang, Yuxiang
;
Li, Xian
;
Liu, Xueling
;
Chen, Yi
;
Yang, Chunhao
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Simultaneous inhibition of PI3Kα and CDK4/6 synergistically suppresses KRAS-mutated non-small cell lung cancer
期刊论文
OAI收割
CANCER BIOLOGY & MEDICINE, 2019, 卷号: 16, 期号: 1, 页码: 66-83
作者:
Wang, Yuxiang
;
Li, Xian
;
Liu, Xueling
;
Chen, Yi
;
Yang, Chunhao
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Simultaneous inhibition of PI3Kα and CDK4/6 synergistically suppresses KRAS-mutated non-small cell lung cancer
期刊论文
OAI收割
Cancer Biology and Medicine, 2019, 卷号: 16, 期号: 1, 页码: 66
作者:
Wang Yuxiang
;
Li Xian
;
Liu Xueling
;
Chen Yi
;
Yang Chunhao
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收藏
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