中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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Pharmacokinetics, mass balance, and metabolism of [
14
C]PLB1004, a selective and irreversible EGFR-TKI in humans
期刊论文
OAI收割
CANCER CHEMOTHERAPY AND PHARMACOLOGY, 2025, 卷号: 95, 期号: 1, 页码: 14
作者:
Liu, Donghui
;
Li, Qian
;
Yan, Shu
;
Zhang, Xinyue
;
Li, Weiqiang
  |  
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2025/04/01
PLB1004
[C-14]PLB1004
Radioactivity
Mass balance
EGFR-TKI
Pharmacokinetics, mass balance, and metabolism of [
14
C]FCN-437c, a selective and potent CDK4/6 inhibitor in humans
期刊论文
OAI收割
CANCER CHEMOTHERAPY AND PHARMACOLOGY, 2025, 卷号: 95, 期号: 1, 页码: 12
作者:
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2025/07/25
FCN-437c
CDK4/6 inhibitor
Mass balance
Radiopharmacokinetics
Drug metabolism
Torque work of origin-destination flows: Quantifying urban place centrality from a physical perspective
期刊论文
OAI收割
COMPUTERS ENVIRONMENT AND URBAN SYSTEMS, 2025, 卷号: 121, 页码: 102311
作者:
Yan, Xiaorui
;
Pei, Tao
;
Song, Ci
;
Fang, Zidong
;
Liu, Xiaohan
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2025/07/18
Place centrality
Origin-destination flows
Torque work
Multiscale analysis
Intra-day dynamic
Urban science
Discovery of novel imidazo[2,1-b][1,3,4]thiadiazole analogs as fluorescent SHP2 inhibitors
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2025, 卷号: 163, 页码: 10
作者:
Zhang, Chun
;
Yan, Xue
;
Gao, Li-Xin
;
Cao, Zi-Tong
;
Cao, Qing
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2025/08/20
Imidazo[2,1-b][1,3,4]thiadiazole
Inhibitory activities
Fluorescence imaging
Zebrafish
SHP2
Study of ultra-high-energy gamma-ray source 1LHAASO J0056+6346u and its possible origins
期刊论文
OAI收割
SCIENCE CHINA-PHYSICS MECHANICS & ASTRONOMY, 2025, 卷号: 68, 期号: 7
作者:
Cao, Zhen
;
Aharonian, F.
;
Axikegu
;
Bai, Y. X.
;
Bao, Y. W.
  |  
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2025/06/10
gamma rays
cosmic rays
supernova remnant
young massive cluster
pulsar
Metabolomic and evolutionary integration unveils medicinal potential in six
Corydalis
species
期刊论文
OAI收割
MOLECULAR HORTICULTURE, 2025, 卷号: 5, 期号: 1, 页码: 14
作者:
Gao, Yun
;
Zhou, Xiangyu
;
Yan, Mengxiao
;
Wang, Zhengwei
;
Zhong, Xin
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2025/08/20
Corydalis
genus
Benzylisoquinoline alkaloids (BIAs)
Evolutionary analysis
Metabolomics
Medicinal resources
Incorporation of Mometasone Furoate into a Cyclodextrin Metal-Organic Framework to Optimize Nasal Administration
期刊论文
OAI收割
PHARMACEUTICS, 2025, 卷号: 17, 期号: 6, 页码: 17
作者:
Li, Jie
;
Guo, Yuhua
;
Liu, Yan
;
Gao, Qingfang
;
Wang, Siwen
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2025/08/20
mometasone furoate
cyclodextrin metal-organic framework
nasal powder spray
three-dimensional biomimetic model of the human nasal cavity
Contrastive learning-based drug screening model for GluN1/GluN3A inhibitors
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2025, 页码: 13
作者:
Li, Kun
;
Zeng, Yue
;
Xiong, Yi-da
;
Wu, Hao-chen
;
Fang, Sui
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2025/08/20
drug-target affinity prediction
virtual screening
contrastive learning
graph neural network
N
-methyl-
D
-aspartate (NMDA) receptors
GluN3A subunit.
Gravitational wave astronomy with TianQin
期刊论文
OAI收割
REPORTS ON PROGRESS IN PHYSICS, 2025, 卷号: 88, 期号: 5
作者:
Li, En-Kun
;
Liu, Shuai
;
Torres-Orjuela, Alejandro
;
Chen, Xian
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2025/05/26
gravitational wave
astronomy
TianQin
Diverse Secondary Metabolites From the
Ligia exotica-
Derived Fungus
Diaporthe melitensis
HZ-1
期刊论文
OAI收割
CHEMISTRY & BIODIVERSITY, 2025, 页码: 7
作者:
Zhu, Ming-Xin
;
Hao, Yi
;
Yan, Bing-Yuan
;
Jin, Yang
;
Gao, Zhen
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2025/06/23
antibacterial activities
Diaporthe melitensis
Ligia exotica
marine natural products