中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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上海药物研究所 [242]
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广州生物医药与健康研... [2]
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期刊论文 [248]
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2026 [1]
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Discovery of a potent and orally bioavailable 3,3-dimethyl-2-oxoindoline STING inhibitor
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2026, 卷号: 301, 页码: 18
作者:
Li, Wenxin
;
Wang, Xiyuan
;
Zang, Shumin
;
Zhou, Rongyao
;
Zhou, Hongfei
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Discovery of isoindoline-2(1
H
)-carboxamide STING inhibitors as anti-inflammatory agents
期刊论文
OAI收割
MOLECULAR DIVERSITY, 2025, 页码: 13
作者:
Zhou, Xiaoqian
;
Zang, Shumin
;
Yao, Shanyan
;
Zhou, Hongfei
;
Wang, Xiyuan
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  |  
Discovery of 3,4-dihydroisoquinoline-2(1H)-carboxamide STING inhibitors as anti-inflammatory agents
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 297, 页码: 20
作者:
Zhou, Xiaoqian
;
Yue, Hangtian
;
Wang, Xiyuan
;
Zang, Shumin
;
Li, Han
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Design, synthesis, and biological evaluation of KDM5B degraders against hematologic malignancy cells
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 296, 页码: 17
作者:
Liu, Xiaowen
;
Li, Jiarong
;
Guo, Yihao
;
Xie, Zhicheng
;
Geng, Meiyu
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Discovery of indole derivatives as STING degraders
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 294, 页码: 21
作者:
An, Yuxiang
;
Zhang, Yan
;
Luo, Xin
;
Lan, Yaohan
;
Geng, Meiyu
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Structural Optimization of Next-Generation TRK Inhibitors against Acquired Drug Resistance Mutations for the Treatment of Solid Tumors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 11, 页码: 11484-11501
作者:
Xu, Zichao
;
Liu, Yueling
;
Wang, Peng
;
Peng, Xia
;
Cheng, Jiawei
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Discovery of Hydrazineyl Amide Derivative of Pseudolaric Acid B for Reprogramming Tumor-Associated Macrophages Against Tumor Growth
期刊论文
OAI收割
MOLECULES, 2025, 卷号: 30, 期号: 10, 页码: 22
作者:
Peng, Xia
;
Yu, Siqi
;
Xu, Lin
;
Wang, Qinghua
;
Yang, Lin
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Discovery of Potent STING Inhibitors Bearing a Difluorobenzodioxol Structural Motif as Potent Anti-Inflammatory Agents
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 8, 页码: 8907-8932
作者:
Shen, Ancheng
;
Wang, Xiyuan
;
Chen, Qingxuan
;
Zhang, Yan
;
Wang, Fang
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Quantitation of global histone post-translational modifications reveal anti-inflammatory epigenetic mechanisms of liquiritigenin based on the optimized super-SILAC strategy
期刊论文
OAI收割
FRONTIERS IN CELL AND DEVELOPMENTAL BIOLOGY, 2025, 卷号: 13, 页码: 15
作者:
Liu, Ping
;
Zhang, Jun
;
Zhang, Jingdan
;
Yuan, Yucheng
;
Liu, Zhiqing
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Discovery of a non-nucleotide stimulator of interferon genes (STING) agonist with systemic antitumor effect
期刊论文
OAI收割
MEDCOMM, 2025, 卷号: 6, 期号: 1, 页码: e70001
作者:
Wang, Xiyuan
;
Zhan, Zhengsheng
;
Wang, Zhen
;
Zhang, Yan
;
Zhao, Kaiyan
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