中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共252条,第1-10条 帮助

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Discovery of a potent and orally bioavailable 3,3-dimethyl-2-oxoindoline STING inhibitor 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2026, 卷号: 301, 页码: 18
作者:  
Li, Wenxin;  Wang, Xiyuan;  Zang, Shumin;  Zhou, Rongyao;  Zhou, Hongfei
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Discovery of isoindoline-2(1H)-carboxamide STING inhibitors as anti-inflammatory agents 期刊论文  OAI收割
MOLECULAR DIVERSITY, 2025, 页码: 13
作者:  
Zhou, Xiaoqian;  Zang, Shumin;  Yao, Shanyan;  Zhou, Hongfei;  Wang, Xiyuan
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Discovery of 3,4-dihydroisoquinoline-2(1H)-carboxamide STING inhibitors as anti-inflammatory agents 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 297, 页码: 20
作者:  
Zhou, Xiaoqian;  Yue, Hangtian;  Wang, Xiyuan;  Zang, Shumin;  Li, Han
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Design, synthesis, and biological evaluation of KDM5B degraders against hematologic malignancy cells 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 296, 页码: 17
作者:  
Liu, Xiaowen;  Li, Jiarong;  Guo, Yihao;  Xie, Zhicheng;  Geng, Meiyu
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Discovery of indole derivatives as STING degraders 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 294, 页码: 21
作者:  
An, Yuxiang;  Zhang, Yan;  Luo, Xin;  Lan, Yaohan;  Geng, Meiyu
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Structural Optimization of Next-Generation TRK Inhibitors against Acquired Drug Resistance Mutations for the Treatment of Solid Tumors 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 11, 页码: 11484-11501
作者:  
Xu, Zichao;  Liu, Yueling;  Wang, Peng;  Peng, Xia;  Cheng, Jiawei
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Discovery of Hydrazineyl Amide Derivative of Pseudolaric Acid B for Reprogramming Tumor-Associated Macrophages Against Tumor Growth 期刊论文  OAI收割
MOLECULES, 2025, 卷号: 30, 期号: 10, 页码: 22
作者:  
Peng, Xia;  Yu, Siqi;  Xu, Lin;  Wang, Qinghua;  Yang, Lin
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Discovery of Potent STING Inhibitors Bearing a Difluorobenzodioxol Structural Motif as Potent Anti-Inflammatory Agents 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 8, 页码: 8907-8932
作者:  
Shen, Ancheng;  Wang, Xiyuan;  Chen, Qingxuan;  Zhang, Yan;  Wang, Fang
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Quantitation of global histone post-translational modifications reveal anti-inflammatory epigenetic mechanisms of liquiritigenin based on the optimized super-SILAC strategy 期刊论文  OAI收割
FRONTIERS IN CELL AND DEVELOPMENTAL BIOLOGY, 2025, 卷号: 13, 页码: 15
作者:  
Liu, Ping;  Zhang, Jun;  Zhang, Jingdan;  Yuan, Yucheng;  Liu, Zhiqing
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Discovery of a non-nucleotide stimulator of interferon genes (STING) agonist with systemic antitumor effect 期刊论文  OAI收割
MEDCOMM, 2025, 卷号: 6, 期号: 1, 页码: e70001
作者:  
Wang, Xiyuan;  Zhan, Zhengsheng;  Wang, Zhen;  Zhang, Yan;  Zhao, Kaiyan
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