中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共21条,第1-10条 帮助

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Novel Aryl Sulfonium Modification on Vancomycin to Tackle MRSA and VRE In Vitro and In Vivo through Dual Enhanced Cell-Wall and Membrane Inhibition 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 8, 页码: 8310-8329
作者:  
Xie, Yuanyuan;  Wang, Xiaowen;  Chang, Taopeng;  Chen, Zhifu;  Luo, Youhong
  |  收藏  |  浏览/下载:2/0  |  提交时间:2025/06/23
A Rationally Designed Sulfonium Lipoglycopeptide with Micelles Self-Assembly to Combat Multidrug Resistance via Dual Enhanced Cell Wall-Membrane Inhibition and T7SS Proteins Downregulation 期刊论文  OAI收割
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2025, 卷号: 147, 期号: 15, 页码: 12587-12603
作者:  
Xie, Yuanyuan;  Wang, Xiaowen;  Li, Fang;  Chen, Zhifu;  Li, Qun
  |  收藏  |  浏览/下载:1/0  |  提交时间:2025/05/27
Single Amine or Guanidine Modification on Norvancomycin and Vancomycin to Overcome Multidrug-Resistance through Augmented Lipid II Binding and Increased Membrane Activity 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 22, 页码: 20639-20663
作者:  
Bian, Xiaolei;  Chen, Zhifu;  Li, Fang;  Xie, Yuanyuan;  Li, Yi
  |  收藏  |  浏览/下载:10/0  |  提交时间:2024/12/11
A Vancomycin-Templated DNA-Encoded Library for Combating Drug-Resistant Bacteria 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 5, 页码: 3778-3794
作者:  
Guan, Dongliang;  Liu, Jiaxiang;  Chen, Feifei;  Li, Jian;  Wang, Xiaowen
  |  收藏  |  浏览/下载:19/0  |  提交时间:2024/05/07
A facile and selective derivatization approach on kynurenine-NH2 in daptomycin, leading to the discovery of hexakynomycin to combat multidrug-resistant Gram-positive pathogens especially daptomycin-resistant bacteria 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 259, 页码: 14
作者:  
Guan, Dongliang;  Li, Jian;  Chen, Feifei;  Li, Jiaqi;  Bian, Xiaolei
  |  收藏  |  浏览/下载:20/0  |  提交时间:2023/10/17
Carbohydrate Strengthens the Immunotherapeutic Effect of Small-Molecule PD-L1 Inhibitors 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 11, 页码: 7179-7204
作者:  
Dong, Qian;  Tong, Mengya;  Yu, Xiaolu;  Wang, Lei;  Ao, Jiwei
  |  收藏  |  浏览/下载:42/0  |  提交时间:2023/10/17
Single Modification at the N-Terminus of Norvancomycin to Combat Drug-Resistant Gram-Positive Bacteria 期刊论文  OAI收割
CHEMMEDCHEM, 2023, 卷号: 18, 期号: 9
作者:  
Guan, Dongliang;  Chen, Feifei;  Shi, Wei;  Lan, Lefu;  Huang, Wei
  |  收藏  |  浏览/下载:15/0  |  提交时间:2024/03/27
Potentiation of Vancomycin: Creating Cooperative Membrane Lysis through a "Derivatization-for-Sensitization" Approach 期刊论文  OAI收割
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2022, 卷号: 144, 期号: 23, 页码: 10622-10639
作者:  
Lei, E.;  Tao, Huanyu;  Jiao, Shang;  Yang, Anming;  Zhou, Yu
  |  收藏  |  浏览/下载:50/0  |  提交时间:2022/08/16
Impurity Identification and Scale-Up of a Novel Glycopeptide Antibiotic 期刊论文  OAI收割
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2021, 卷号: 25, 期号: 11, 页码: 2390-2402
作者:  
Jiao, Shang;  Guan, Dongliang;  Xu, Lili;  Liu, Bo;  Shi, Weiwei
  |  收藏  |  浏览/下载:40/0  |  提交时间:2022/01/18
Total and Semisyntheses of Polymyxin Analogues with 2-Thr or 10-Thr Modifications to Decipher the Structure-Activity Relationship and Improve the Antibacterial Activity 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 9, 页码: 5746-5765
作者:  
Li, Jian;  Guan, Dongliang;  Chen, Feifei;  Shi, Weiwei;  Lan, Lefu
  |  收藏  |  浏览/下载:24/0  |  提交时间:2021/08/17