中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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高能物理研究所 [386]
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Design and synthesis of CDK9/EZH2 dual-target inhibitors to achieve synergistic antitumor effects
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 294, 页码: 14
作者:
Tian, Lina
;
Xiao, Jian
;
Zeng, Yanping
;
Li, Yangsha
;
Wei, Aihuan
  |  
收藏
  |  
浏览/下载:0/0
  |  
提交时间:2025/08/20
CDK9
EZH2
Dual target inhibitor
DLBCL
Discovery of novel Ebola entry inhibitors with 1,2,3,4-tetrahydroisoquinoline-3-carboxamide based on (3S,4aS,8aS)-2-(3-amino-2-hydroxypropyl) decahydroisoquinoline-3-carboxamide scaffold
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2025, 卷号: 123, 页码: 4
作者:
Lin, Junzhen
;
Xiao, Fuling
;
Han, Sheng
;
Hu, Youhong
;
Zuo, Jianping
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2025/06/23
Ebola virus entry inhibitor
Tetrahydroisoquinoline
Conceptualization and assessment of groundwater-seawater interactions on bedrock islands
期刊论文
OAI收割
JOURNAL OF HYDROLOGY, 2025, 卷号: 655, 页码: 132886
作者:
Gong, Rong
;
Han, Dongmei
;
Xiao, Yi
;
Song, Xianfang
;
Wang, Wei
  |  
收藏
  |  
浏览/下载:45/0
  |  
提交时间:2025/04/21
Groundwater-seawater interactions
Bedrock islands
Nitrate-nitrogen
Chloride
Groundwater management
Study of ultra-high-energy gamma-ray source 1LHAASO J0056+6346u and its possible origins
期刊论文
OAI收割
SCIENCE CHINA-PHYSICS MECHANICS & ASTRONOMY, 2025, 卷号: 68, 期号: 7
作者:
Cao, Zhen
;
Aharonian, F.
;
Axikegu
;
Bai, Y. X.
;
Bao, Y. W.
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2025/06/10
gamma rays
cosmic rays
supernova remnant
young massive cluster
pulsar
A BODIPY-tagged trivalent glycocluster for receptor-targeting fluorescence imaging of live cells
期刊论文
OAI收割
CHEMICAL SCIENCE, 2025, 卷号: 16, 期号: 25, 页码: 11481-11486
作者:
Guo, Chen
;
Si, Fang-Yu
;
Wang, Chen-Han
;
Wang, Ning
;
Hu, Xi-Le
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2025/07/25
Advancing active compound discovery for novel drug targets: insights from AI-driven approaches
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2025, 页码: 12
作者:
Wang, Xing-you
;
Chen, Yang
;
Li, Yu-fan
;
Wei, Chao-yang
;
Liu, Meng-ya
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2025/08/20
AI-driven drug discovery
novel drug targets
molecular design
ligand exploration
phenotypic drug discovery
undruggable targets
Nitrogen sensitivity of soil microorganism community in alpine desert steppe is not always higher than that in alpine steppe
期刊论文
OAI收割
GLOBAL ECOLOGY AND CONSERVATION, 2025, 卷号: 59, 页码: e03459
作者:
Wang, Zhishu
;
Xiao, Jianyu
;
Han, Fusong
;
Huang, Shaolin
;
Yu, Chengqun
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2025/04/21
Steppe types
Nitrogen addition gradients
Nitrogen sensitivity
Soil microbial community
Tibetan Plateau
Recent Advancement in Fluorescent Probes for Peroxynitrite (ONOO
-
)
期刊论文
OAI收割
SENSORS, 2025, 卷号: 25, 期号: 10, 页码: 41
作者:
Han, Hai-Hao
;
Ge, Pan-Xin
;
Li, Wen-Jia
;
Hu, Xi-Le
;
He, Xiao-Peng
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2025/07/25
peroxynitrite (ONOO-)
fluorescent probes
bioimaging
in vivo
disease diagnosis and treatment
Structure-activity relationship analysis of meta-substituted N-cyclopropylmethyl-nornepenthones with mixed KOR/MOR activities
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 289, 页码: 15
作者:
Tang, Siyuan
;
Hu, Shuyang
;
Feng, Lijing
;
Kong, Linghui
;
Gui, Jiangwen
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2025/05/27
N-Cyclopropylmethyl-nornepenthones
Structure-activity relationship
MOR antagonist
KOR agonist
Substance use disorder
Exploring Origin-Dependent Susceptibility of Smooth Muscle Cells to Aortic Diseases Through Intersectional Genetics
期刊论文
OAI收割
CIRCULATION, 2025, 卷号: 151, 期号: 17, 页码: 1248-1267
作者:
Han, Ximeng
;
Li, Yi
;
Wang, Enci
;
Zhu, Huan
;
Huang, Xiuzhen
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2025/06/23
aortic diseases
developmental origin
lineage tracing
smooth muscle cell
TGF-beta