中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [5]
计算技术研究所 [1]
采集方式
OAI收割 [6]
内容类型
期刊论文 [6]
发表日期
2023 [1]
2022 [1]
2021 [1]
2019 [1]
2018 [1]
2009 [1]
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YCH1899, a Highly Effective Phthalazin-1(2H)-one Derivative That Overcomes Resistance to Prior PARP Inhibitors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 20
作者:
Sun, Yuting
;
Yang, Hui
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2023/10/17
Design, synthesis and pharmacological evaluation of new PARP1 inhibitors by merging pharmacophores of olaparib and the natural product alantolactone
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 240, 页码: 114574
作者:
Kayumov, Muzaffar
;
Jia, Li
;
Pardaev, Azizbek
;
Song, Shan-Shan
;
Mirzaakhmedov, Sharafitdin
  |  
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2024/03/21
PARP1
Olaparib
Alantolactone
Syntheticlethality
BRCA1/2mutant
Development of Potent NEDD8-Activating Enzyme Inhibitors Bearing a Pyrimidotriazole Scaffold
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 9, 页码: 6161-6178
作者:
Xiong, Chaodong
;
Zhou, Lina
;
Tan, Jing
;
Song, Shanshan
;
Bao, Xubin
  |  
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2021/08/17
Preclinical characterization of SHR6390, a novel CDK 4/6 inhibitor, invitro and in human tumor xenograft models
期刊论文
OAI收割
CANCER SCIENCE, 2019, 卷号: 110, 期号: 4, 页码: 1420-1430
作者:
Long, Fei
;
He, Ye
;
Fu, Haoyu
;
Li, Yun
;
Bao, Xubin
  |  
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2020/07/01
breast cancer
CDK 4/6
drug resistance
palbociclib
SHR6390
Combined inhibition of PI3K delta and FLT3 signaling exerts synergistic antitumor activity and overcomes acquired drug resistance in FLT3-activated acute myeloid leukemia
期刊论文
OAI收割
CANCER LETTERS, 2018, 卷号: 420, 页码: 49-59
作者:
He, Ye
;
Sun, Liping
;
Xu, Yongping
;
Fu, Li
;
Li, Yun
  |  
收藏
  |  
浏览/下载:50/0
  |  
提交时间:2019/01/08
Acute myeloid leukemia
FLT3
PI3K delta
CAL101
Synergistic effect
An efficient design for fast memory registration in RDMA
期刊论文
OAI收割
JOURNAL OF NETWORK AND COMPUTER APPLICATIONS, 2009, 卷号: 32, 期号: 3, 页码: 642-651
作者:
Ou, Li
;
He, Xubin
;
Han, Jizhong
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2019/12/16
RDMA
Memory registration
Cache
Performance evaluation