中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共66条,第1-10条 帮助

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A Medicinal Chemistry Perspective on Protein Tyrosine Phosphatase Nonreceptor Type 2 in Tumor Immunology 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 4, 页码: 3995-4021
作者:  
Huang, Qi;  Hu, Linghao;  Chen, Haowen;  Yang, Bingjie;  Sun, Xun
  |  收藏  |  浏览/下载:11/0  |  提交时间:2025/04/01
Harnessing the Magic Methyl Effect: Discovery of CLPP-2068 as a Novel HsClpP Activator for the Treatment of Diffuse Large B-Cell Lymphoma 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 4, 页码: 4287-4307
作者:  
Sun, Mingyang;  Chen, Beijing;  Teng, Dan;  Zhao, Hongshen;  Liao, Yilie
  |  收藏  |  浏览/下载:15/0  |  提交时间:2025/04/01
Discovery of SET domain-binding primary alkylamine-tethered degraders for the simultaneous degradation of NSD2-long and RE-IIBP isoforms 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 283, 页码: 17
作者:  
Hu, Linghao;  Xu, Hesong;  Xu, Ye;  Chen, Haowen;  Jiang, Hanrui
  |  收藏  |  浏览/下载:13/0  |  提交时间:2025/04/01
Discovery of CLPP-1071 as an Exceptionally Potent and Orally Efficacious Human ClpP Activator with Strong In Vivo Antitumor Activity 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 21
作者:  
Chen, Beijing;  Sun, Mingyang;  Zhang, Chun;  Huang, Qi;  Teng, Dan
  |  收藏  |  浏览/下载:16/0  |  提交时间:2024/12/25
Discovery of KW0113 as a First and Effective PROTAC Degrader of DNMT1 Protein 期刊论文  OAI收割
CHEMMEDCHEM, 2024, 页码: 16
作者:  
Wang, Huihui;  Wang, Zhaoliang;  Hu, Linghao;  Yang, Bingjie;  Zong, Liangyi
  |  收藏  |  浏览/下载:13/0  |  提交时间:2024/12/16
Discovery of Preclinical Candidate AD1058 as a Highly Potent, Selective, and Brain-Penetrant ATR Inhibitor for the Treatment of Advanced Malignancies 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 15, 页码: 12735-12759
作者:  
Liu, Zhi;  Jiang, Kailong;  Liu, Yan;  Li, Junfei;  Huang, Siqi
  |  收藏  |  浏览/下载:28/0  |  提交时间:2024/09/26
Discovery of a Covalent Inhibitor Selectively Targeting the Autophosphorylation Site of c-Src Kinase 期刊论文  OAI收割
ACS CHEMICAL BIOLOGY, 2024, 页码: 12
作者:  
Zhang, Huimin;  Xu, Dounan;  Huang, Hongchan;  Jiang, Hao;  Hu, Linghao
  |  收藏  |  浏览/下载:21/0  |  提交时间:2024/05/07
Chromosome-level genome assembly of hadal snailfish reveals mechanisms of deep-sea adaptation in vertebrates 期刊论文  OAI收割
ELIFE, 2023, 卷号: 12, 页码: 51
作者:  
Xu, Wenjie;  Zhu, Chenglong;  Gao, Xueli;  Wu, Baosheng;  Xu, Han
  |  收藏  |  浏览/下载:33/0  |  提交时间:2024/03/11
Discovery of PVD-06 as a Subtype-Selective and Efficient PTPN2 Degrader 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 22, 页码: 15269-15287
作者:  
Hu, Linghao;  Li, Huiyun;  Qin, Junlin;  Yang, Dan;  Liu, Jieming
  |  收藏  |  浏览/下载:45/0  |  提交时间:2024/02/27
Shape-persistent phthalocyanine cages 期刊论文  OAI收割
CELL REPORTS PHYSICAL SCIENCE, 2023, 卷号: 4, 期号: 2, 页码: 101285
作者:  
Hu,Yiming;  Huang,Shaoda;  Wayment,Lacey J.;  Wu,Jingyi;  Xu,Qiucheng
  |  收藏  |  浏览/下载:14/0  |  提交时间:2024/07/22