中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [6]
近代物理研究所 [1]
采集方式
OAI收割 [7]
内容类型
期刊论文 [7]
发表日期
2023 [2]
2022 [1]
2021 [1]
2019 [1]
2016 [1]
2015 [1]
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Discovery of JN122, a Spiroindoline-Containing Molecule that Inhibits MDM2/p53 Protein-Protein Interaction and Exerts Robust In Vivo Antitumor Efficacy
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 24, 页码: 16991-17025
作者:
Cheng, Jing
;
Yan, Ziqin
;
Jiang, Kailong
;
Liu, Chen
;
Xu, Dehua
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2024/02/19
Discovery of toxoflavin,a potent IRE1α inhibitor acting through structure-dependent oxidative inhibition
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2023, 卷号: 44, 期号: 1, 页码: 234
作者:
Liu Changmei
;
Nie Litong
;
Jiang Haini
;
Xu Lei
;
Zhang Kunzhi
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2023/05/22
endoplasmic reticulum stress
toxoflavin
reactive oxygen species
IRE1α
XBP1
Dual inhibition of CHK1/FLT3 enhances cytotoxicity and overcomes adaptive and acquired resistance in FLT3-ITD acute myeloid leukemia
期刊论文
OAI收割
LEUKEMIA, 2022, 页码: 11
作者:
Jiang, Kailong
;
Li, Xuemei
;
Wang, Chang
;
Hu, Xiaobei
;
Wang, Peipei
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2023/04/10
Design, Synthesis, and Biological Evaluation of Orally Bioavailable CHK1 Inhibitors Active against Acute Myeloid Leukemia
期刊论文
OAI收割
CHEMMEDCHEM, 2021, 页码: 12
作者:
Jin, Tingting
;
Wang, Peipei
;
Long, Xiubing
;
Jiang, Kailong
;
Song, Pinrao
  |  
收藏
  |  
浏览/下载:125/0
  |  
提交时间:2021/05/24
CHK1 inhibitor
diaminopyrimidine
DNA damage response
oral bioavailability
Discovery of (R)-5-((5-(1-methyl-1H-pyrazol-4-yl)-4-(methylamino) pyrimidin-2-yl)amino)-3-(piperidin-3-yloxy)picolinonitrile, a novel CHK1 inhibitor for hematologic malignancies
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 173, 页码: 44-62
作者:
Tong, Lexian
;
Song, Pinrao
;
Jiang, Kailong
;
Xu, Lei
;
Jin, Tingting
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2020/07/01
CHK1 kinase inhibitor
Selectivity
Monotherapy
Hematologic malignancies
Alpha Decay of the Neutron-deficient Isotopes 215,216U
期刊论文
OAI收割
原子核物理评论, 2016, 页码: 217-220
作者:
Zhang Zhiyuan
;
Gan Zaiguo
;
Ma Long
;
Yang Huabin
;
Wang Jianguo
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2021/12/13
Disruption of the unfolded protein response (UPR) by lead compound selectively suppresses cancer cell growth
期刊论文
OAI收割
CANCER LETTERS, 2015, 卷号: 360, 期号: 2, 页码: 257-268
作者:
Huang, Hejing
;
Liu, Huanan
;
Liu, Changmei
;
Fan, Lixia
;
Zhang, Xinwen
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2019/01/08
Selective cancer therapy
Unfolded protein response
2DG
UPR disrupter