中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [29]
自动化研究所 [3]
地理科学与资源研究所 [2]
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深圳先进技术研究院 [1]
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期刊论文 [44]
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2025 [2]
2024 [7]
2023 [2]
2022 [4]
2021 [2]
2020 [8]
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Harnessing the Magic Methyl Effect: Discovery of CLPP-2068 as a Novel
Hs
ClpP Activator for the Treatment of Diffuse Large B-Cell Lymphoma
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 4, 页码: 4287-4307
作者:
Sun, Mingyang
;
Chen, Beijing
;
Teng, Dan
;
Zhao, Hongshen
;
Liao, Yilie
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2025/04/01
Auto-RapTAC: A Versatile and Sustainable Platform for the Automated Rapid Synthesis and Evaluation of PROTAC
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 页码: 15
作者:
Chen, Jiexuan
;
Wu, Mingfei
;
Mo, Jun
;
Hong, Ju
;
Wang, Wei
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2025/04/01
Discovery of N-Benzylpiperidinol derivatives as USP7 inhibitors against Hematology
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2024, 卷号: 153, 页码: 13
作者:
Pan, Youlu
;
Chen, Haifeng
;
Fu, Jingfeng
;
Zhang, Jingyu
;
Wang, Peipei
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2024/10/21
Discovery of CLPP-1071 as an Exceptionally Potent and Orally Efficacious Human ClpP Activator with Strong In Vivo Antitumor Activity
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 21
作者:
Chen, Beijing
;
Sun, Mingyang
;
Zhang, Chun
;
Huang, Qi
;
Teng, Dan
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2024/12/25
Discovery of Preclinical Candidate AD1058 as a Highly Potent, Selective, and Brain-Penetrant ATR Inhibitor for the Treatment of Advanced Malignancies
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 15, 页码: 12735-12759
作者:
Liu, Zhi
;
Jiang, Kailong
;
Liu, Yan
;
Li, Junfei
;
Huang, Siqi
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2024/09/26
Design, Synthesis, and Biological Evaluation of 2,4-Diaminopyrimidine Derivatives as Potent CDK7 Inhibitors
期刊论文
OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2024, 页码: 8
作者:
Zhang, Hualin
;
Tu, Yutong
;
Tao, Zhaofan
;
Gao, Lixin
;
Huang, Shengjie
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/08/22
CDK7 inhibitor
2,4-diaminopyrimidine
selectivity
anticancer
Discovery of Orally Bioavailable and Potent CDK9 Inhibitors for Targeting Transcription Regulation in Triple-Negative Breast Cancer
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 12, 页码: 10035-10056
作者:
Wang, Wen-Jing
;
Gao, Lixin
;
Wang, Simei
;
Huang, Wensi
;
Meng, Xin-Yu
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2024/08/20
Moisture source differences between the 2020 and 1998 super Meiyu-flood events in the Yangtze River Valley
期刊论文
OAI收割
WEATHER AND CLIMATE EXTREMES, 2024, 卷号: 43, 页码: 100644
作者:
Zhang, Chi
;
Tang, Qiuhong
;
Zhao, Yang
;
Chen, Deliang
;
Huang, Jinchuan
  |  
收藏
  |  
浏览/下载:40/0
  |  
提交时间:2024/04/08
Meiyu
Precipitation
Moisture source
The Yangtze River valley
WAM2Layers
Quantifying precipitation moisture contributed by different atmospheric circulations across the Tibetan Plateau
期刊论文
OAI收割
JOURNAL OF HYDROLOGY, 2024, 卷号: 628, 页码: 130517
作者:
Zhang, Chi
;
Zhang, Xu
;
Tang, Qiuhong
;
Chen, Deliang
;
Huang, Jinchuan
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2024/01/04
Moisture source
Climate
Circulation systems
Tibetan Plateau
Structure-based identification of new orally bioavailable BRD9-PROTACs for treating acute myelocytic leukemia
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 262, 页码: 18
作者:
Zhang, Jingyu
;
Duan, Haiting
;
Gui, Renzhao
;
Wu, Mingfei
;
Shen, Liteng
  |  
收藏
  |  
浏览/下载:131/0
  |  
提交时间:2023/12/19
Acute myeloid leukemia
Bromodomain-containing protein 9
Proteolysis-targeting chimera
Orally bioavailable
Docking