中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [51]
西安光学精密机械研究... [4]
上海营养与健康研究所 [3]
古脊椎动物与古人类研... [3]
生物物理研究所 [2]
海洋研究所 [2]
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OAI收割 [69]
内容类型
期刊论文 [68]
会议论文 [1]
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2026 [2]
2025 [4]
2024 [6]
2023 [5]
2022 [4]
2021 [6]
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Immunology [2]
Biochemist... [1]
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材料科学与物理化学 [1]
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Soil organic carbon fractions and stability shifts in response to plant mixed-growth in coastal wetlands of southeastern China
期刊论文
OAI收割
CATENA, 2026, 卷号: 263, 页码: 14
作者:
Ren, Xiaoying
;
Xu, Jiayi
;
Wang, Weiqi
;
Yin, Rongbin
;
Li, Yuan
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2026/01/19
Southeastern China
Organic carbon fractions
Carbon pool stability
Plant mixing
Coastal wetland soils
Novel thieno[2,3-b]pyridine derivatives protect islet through DRAK2 kinase inhibition
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2026, 卷号: 301, 页码: 18
作者:
Lian, Kaiyue
;
Li, Ruihan
;
Lu, Yuting
;
Song, Gaolei
;
Zhang, Xinwen
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2025/12/04
DRAK2
Inhibitor
Thieno[2
b ]pyridine
Diabetes
The enedioic acid analog 326E alleviates metabolic dysfunction-associated steatohepatitis via dual targeting at ACLY and PPARα
期刊论文
OAI收割
CELL METABOLISM, 2025, 卷号: 37, 期号: 11, 页码: 2149-2166
作者:
Xie, Zhifu
;
Cheng, Long
;
Hu, Yue
;
Song, Gaolei
;
Wang, Fan
  |  
收藏
  |  
浏览/下载:0/0
  |  
提交时间:2026/01/28
Mechanism of hydroxamic acid group metabolism to carboxylic acid: Oxidation versus hydrolysis
期刊论文
OAI收割
DRUG METABOLISM AND DISPOSITION, 2025, 卷号: 53, 期号: 10, 页码: 11
作者:
Huang, Xiyue
;
Zhou, Lei
;
Chen, Huixian
;
Sun, Xiaowei
;
Cao, Mengyi
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2025/12/04
Hydroxamic acid group
Bisthianostat
HDAC inhibitor
Cytochrome P450 enzymes
Oxidative cleavage
Discovery of Novel Tridentate Alkenyl Diacid Derivatives as Potent ATP Citrate Lyase Inhibitors for the Treatment of Hepatocellular Carcinoma
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 15, 页码: 15598-15616
作者:
Yang, Yurou
;
Zhai, Jimao
;
Wang, Fan
;
Song, Gaolei
;
Xu, Honghong
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2025/09/09
A Phase I Study to Evaluate the Safety, Tolerability, Pharmacokinetics of BGT-002, a Novel ATP-Citrate Lyase Inhibitor, in Healthy Chinese Subjects
期刊论文
OAI收割
DRUG DESIGN DEVELOPMENT AND THERAPY, 2025, 卷号: 19, 页码: 1783-1794
作者:
Liu, Yun
;
Yu, Chengyin
;
Zhang, Yifan
;
Xie, Zhifu
;
Wang, Yating
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2025/04/24
safety
tolerability
pharmacokinetics
pharmacodynamics
BGT-002
novel ACLY inhibitor
Discovery of Alkyl Conjugated Diene Diacids as Novel ACLY Inhibitors
期刊论文
OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2024, 卷号: 44, 期号: 11, 页码: 3476-3489
作者:
Cheng, Tingting
;
Song, Gaolei
;
Cheng, Long
;
Wang, Fan
;
Sun, Xinyu
  |  
收藏
  |  
浏览/下载:60/0
  |  
提交时间:2025/02/28
metabolic diseases
ATP-citrate lyase (ACLY)
lipogenesis
ACLY inhibitors
dienyldicarboxylic acid
A brain-to-gut signal controls intestinal fat absorption
期刊论文
OAI收割
NATURE, 2024, 页码: 27
作者:
Lyu, Qianqian
;
Xue, Wenzhi
;
Liu, Ruixin
;
Ma, Qinyun
;
Kasaragod, Vikram Babu
  |  
收藏
  |  
浏览/下载:89/0
  |  
提交时间:2024/11/26
Discovery of GPR84 Fluorogenic Probes Based on a Novel Antagonist for GPR84 Bioimaging
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 16
作者:
Xiao, Yufeng
;
Chen, Jing
;
Li, Shaoxian
;
Zhang, Qing
;
Liu, Yin
  |  
收藏
  |  
浏览/下载:56/0
  |  
提交时间:2024/08/22
The trunk replaces the longer mandible as the main feeding organ in elephant evolution
期刊论文
OAI收割
ELIFE, 2024, 卷号: 12, 期号: 1, 页码: 22
作者:
Li, Chunxiao
;
Deng, Tao
;
Wang, Yang
;
Sun, Fajun
;
Wolff, Burt
  |  
收藏
  |  
浏览/下载:57/0
  |  
提交时间:2025/01/03
Miocene
elephant
trunk
mandible
stable isotope
finite element analysis
None