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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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近代物理研究所 [83]
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Design and synthesis of CDK9/EZH2 dual-target inhibitors to achieve synergistic antitumor effects
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 294, 页码: 14
作者:
Tian, Lina
;
Xiao, Jian
;
Zeng, Yanping
;
Li, Yangsha
;
Wei, Aihuan
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2025/08/20
CDK9
EZH2
Dual target inhibitor
DLBCL
Heterocycle-fused phenylcyclohexylamines as novel multi-target antagonists of N-methyl-D-aspartate (NMDA) receptor and monoamine transporter for treating depression
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 291, 页码: 20
作者:
Zheng, Fuqiang
;
Hu, Zhengtao
;
Chen, Hai
;
Cheng, Jiaxin
;
Hou, Qiongqiong
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2025/06/23
Heterocycle-fused phenylcyclohexylamines
Multi-target antagonists
NMDAR
Monoamine transporter
Antidepressants
Gravitational wave astronomy with TianQin
期刊论文
OAI收割
REPORTS ON PROGRESS IN PHYSICS, 2025, 卷号: 88, 期号: 5
作者:
Li, En-Kun
;
Liu, Shuai
;
Torres-Orjuela, Alejandro
;
Chen, Xian
;
Inayoshi, Kohei
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2025/05/26
gravitational wave
astronomy
TianQin
Design and Development of a Novel Oral 4′-Fluorouridine Double Prodrug VV261 against SFTSV
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 9, 页码: 9811-9826
作者:
Cheng, Yong
;
Zheng, Wei
;
Dong, Xinru
;
Sun, Tengxiao
;
Xu, Mengwei
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2025/06/23
Design, Synthesis, and Biological Evaluation of Pyrrolo[1,2-
a
]quinoxalin-4(5
H
)-one Derivatives as Potent and Orally Available Noncovalent Bruton's Tyrosine Kinase (BTK) Inhibitors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 8, 页码: 8841-8860
作者:
Tian, Chaoquan
;
Du, Husheng
;
Sha, Wenjie
;
Wu, Lingkang
;
Yu, Zhixiao
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2025/05/27
Broadband γ-Ray Spectrum of Supernova Remnant Cassiopeia A
期刊论文
OAI收割
ASTROPHYSICAL JOURNAL LETTERS, 2025, 卷号: 982, 期号: 1
作者:
Cao, Zhen
;
Aharonian, F.
;
Bai, Y. X.
;
Bao, Y. W.
;
Bastieri, D.
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2025/05/05
Constraining the Cosmic-Ray Energy Based on Observations of Nearby Galaxy Clusters by LHAASO
期刊论文
OAI收割
ASTROPHYSICAL JOURNAL LETTERS, 2025, 卷号: 982, 期号: 1
作者:
Cao, Zhen
;
Aharonian, F.
;
Bai, Y. X.
;
Bao, Y. W.
;
Bastieri, D.
  |  
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2025/05/05
Electrophysiological Abnormalities and Pharmacological Corrections of Pathogenic Missense Variants in KCNQ3
期刊论文
OAI收割
NEUROSCIENCE BULLETIN, 2025, 页码: 11
作者:
Wu, Xiaorong
;
Gong, Jili
;
Qiu, Li
;
Yang, Guimei
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2025/05/27
KCNQ3
Self-limited familial neonatal epilepsy
Neurodevelopmental disorder
Pynegabine
Amitriptyline
Electrophysiology
Terrestrial ecosystem response to Early Cretaceous global environmental change: A calibrated, high-resolution Aptian record from Northeast China
期刊论文
OAI收割
EARTH AND PLANETARY SCIENCE LETTERS, 2025, 卷号: 653, 页码: 13
作者:
  |  
收藏
  |  
浏览/下载:46/0
  |  
提交时间:2025/04/03
Early Cretaceous
Aptian
CA-ID-TIMS geochronology
Astrochronology
Carbon isotope stratigraphy
Mercury evidence for volcanism driving environmental changes during the protracted Late Ordovician mass extinction and early Silurian recovery
期刊论文
OAI收割
CHEMICAL GEOLOGY, 2025, 卷号: 674, 页码: 11
作者:
Li, Yanfang
;
Tian, Hui
;
Zhang, Tongwei
;
Shen, Baojian
;
Shao, Deyong
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2025/04/01
Volcanic activity
Mercury isotope
Ordovician-Silurian transition
Hirnantian glaciation
Mass extinctions
Black shale