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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [40]
化学研究所 [15]
地质与地球物理研究所 [9]
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期刊论文 [113]
会议论文 [2]
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Limnology [1]
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共115条,第1-10条
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Discovery of Novel Class of METTL3 Inhibitors with a Pyridin-2(1
H
)-one Moiety
期刊论文
OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2025, 卷号: 16, 期号: 11, 页码: 2257-2263
作者:
Zhang, Weihang
;
Huang, Yuting
;
Yang, Hong
;
Wan, Haiyan
;
Lei, Xinsheng
  |  
收藏
  |  
Pretargeted Mitochondrial Delivery of Organoarsenicals for Cancer Immunotherapy
期刊论文
OAI收割
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2025, 卷号: 147, 期号: 42, 页码: 38534-38548
作者:
Wang, Run
;
Tian, Yuyang
;
Lu, Xuliang
;
Fang, Leyi
;
Miao, Yinxing
  |  
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  |  
Discovery of Potent and Selective FABP4/5 Inhibitors with an Isoquinolone Scaffold as Potential Therapeutics for Inflammation-Related Diseases
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 19, 页码: 20207-20227
作者:
He, Yulong
;
Li, Shunyi
;
Chen, Yuqi
;
Xu, Yiyang
;
Wang, Yujie
  |  
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  |  
Bacteriochlorophyll reveals estuarine hypoxia and anoxygenic photosynthetic carbon fixation
期刊论文
OAI收割
LIMNOLOGY AND OCEANOGRAPHY, 2025, 页码: 13
作者:
Kan, Jiawei
;
Duan, Liqin
;
Song, Jinming
;
Yin, Meiling
;
Li, Xuegang
  |  
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  |  
Discovery of novel TLR2 antagonists as anti-inflammatory agents
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2025, 卷号: 164, 页码: 15
作者:
Tang, Xuehang
;
Qi, Luyao
;
Li, Yingxia
;
Tang, Wei
;
Zhang, Wei
  |  
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  |  
Discovery of CZL-046 with an (
S
)-3-Fluoropyrrolidin-2-one Scaffold as a p300 Bromodomain Inhibitor for the Treatment of Multiple Myeloma
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 20, 页码: 18606-18628
作者:
Chen, Zonglong
;
Yang, Hong
;
Zhang, Yan
;
Lyu, Xiaodong
;
Shi, Qiongyu
  |  
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  |  
Development of ketalized unsaturated saccharides as multifunctional cysteine-targeting covalent warheads
期刊论文
OAI收割
COMMUNICATIONS CHEMISTRY, 2024, 卷号: 7, 期号: 1, 页码: 10
作者:
Dong, Sanfeng
;
Huang, Hui
;
Li, Jintian
;
Li, Xiaomei
;
Bunu, Samuel Jacob
  |  
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  |  
Vertical variations of bacteriohopanepolyols near the Changjiang Estuary waters: Implications for marine hypoxia and bacterial activities
期刊论文
OAI收割
CHEMICAL GEOLOGY, 2024, 卷号: 651, 页码: 14
作者:
Yin, Meiling
;
Duan, Liqin
;
Song, Jinming
;
Kan, Jiawei
;
Yuan, Huamao
  |  
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  |  
Discovery of Novel PROTAC Degraders of p300/CBP as Potential Therapeutics for Hepatocellular Carcinoma
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 4, 页码: 2466-2486
作者:
Chang, Qi
;
Li, Jiayi
;
Deng, Yue
;
Zhou, Ruilin
;
Wang, Bingwei
  |  
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  |  
Design and synthesis of cantharidin derivative DCZ5418 as a TRIP13 inhibitor with anti-multiple myeloma activity
in
vitro
and
in
vivo
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2024, 卷号: 98, 页码: 7
作者:
Dong, Sanfeng
;
Hu, Ke
;
Shi, Yulong
;
Wang, Guanli
;
Yu, Dandan
  |  
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  |