中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海硅酸盐研究所 [36]
地质与地球物理研究... [13]
上海药物研究所 [11]
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期刊论文 [81]
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Single Amine or Guanidine Modification on Norvancomycin and Vancomycin to Overcome Multidrug-Resistance through Augmented Lipid II Binding and Increased Membrane Activity
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 22, 页码: 20639-20663
作者:
Bian, Xiaolei
;
Chen, Zhifu
;
Li, Fang
;
Xie, Yuanyuan
;
Li, Yi
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收藏
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浏览/下载:5/0
  |  
提交时间:2024/12/11
Discovery of Alkyl Conjugated Diene Diacids as Novel ACLY Inhibitors
期刊论文
OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2024, 卷号: 44, 期号: 11, 页码: 3476-3489
作者:
Cheng, Tingting
;
Song, Gaolei
;
Cheng, Long
;
Wang, Fan
;
Sun, Xinyu
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收藏
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浏览/下载:6/0
  |  
提交时间:2025/02/28
metabolic diseases
ATP-citrate lyase (ACLY)
lipogenesis
ACLY inhibitors
dienyldicarboxylic acid
Simultaneous determination of BGT-002 and its acyl glucuronide metabolite ZM326E-M2 in human plasma by liquid chromatography-tandem mass spectrometry and its application to a pharmacokinetic study
期刊论文
OAI收割
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2024, 卷号: 243, 页码: 8
作者:
Zhu, Xueran
;
Cui, Shumin
;
Liu, Xinjing
;
Zhang, Mei
;
Xie, Zhifu
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2024/05/31
ATP-Citrate Lyase
BGT-002
Acyl glucuronide metabolite
Pseudo-MRM
LC-MS/MS
Pharmacokinetics
AMPK phosphorylation of FNIP1 (S220) controls mitochondrial function and muscle fuel utilization during exercise
期刊论文
OAI收割
SCIENCE ADVANCES, 2024, 卷号: 10, 期号: 6, 页码: 15
作者:
Xiao, Liwei
;
Yin, Yujing
;
Sun, Zongchao
;
Liu, Jing
;
Jia, Yuhuan
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收藏
  |  
浏览/下载:19/0
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提交时间:2024/05/31
HIF-1 alpha inhibition in macrophages preserves acute liver failure by reducing IL-1 beta production
期刊论文
OAI收割
FASEB JOURNAL, 2023, 卷号: 37, 期号: 9, 页码: 12
作者:
Kong, Xiangrong
;
Liu, Wei
;
Zhang, Xinwen
;
Zhou, Chendong
;
Sun, Xinyu
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2023/10/17
acute liver failure
cell death
HIF-1 alpha inhibitor
interleukin-1 beta
macrophage
Long-term drying trends since the mid-Holocene in the Qaidam Basin
期刊论文
OAI收割
CATENA, 2023, 卷号: 228, 页码: 14
作者:
Zhang, Ting
;
Wang, Gen
;
Wang, Yongli
;
Wei, Zhifu
;
He, Wei
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收藏
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浏览/下载:23/0
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提交时间:2023/12/29
GDGTs
Climate change
Landscape evolution
Qaidam Basin
Asian summer monsoon
Chemical Weathering Intensity as a Reliable Indicator for Southwest Summer Monsoon Reconstruction: Evidence From Clay Minerals of Qionghai Lake Sediments Since the Last Glacial Maximum
期刊论文
OAI收割
GEOCHEMISTRY GEOPHYSICS GEOSYSTEMS, 2023, 卷号: 24, 期号: 7, 页码: 17
作者:
Yu, Xiaoli
;
Wang, Gen
;
Zhang, Ting
;
Ma, Xueyun
;
Zhang, Xiaomei
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收藏
  |  
浏览/下载:23/0
  |  
提交时间:2024/01/02
clay mineral
chemical weathering intensity
southwest summer monsoon
Last Glacial Maximum
Holocene
Development of the novel ACLY inhibitor 326E as a promising treatment for hypercholesterolemia
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13, 期号: 2, 页码: 739-753
作者:
Xie, Zhifu
;
Zhang, Mei
;
Song, Qian
;
Cheng, Long
;
Zhang, Xinwen
  |  
收藏
  |  
浏览/下载:20/0
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提交时间:2024/03/27
Hypercholesterolemia
Atherosclerosis
Liver
ATP-Citrate lyase (ACLY)
Lipogenesis
Cholesterol efflux
ACLY inhibitor
Application of Pb Isotopes and REY Patterns in Tracing Heavy Metals in Farmland Soils from the Upper-Middle Area of Yangtze River
期刊论文
OAI收割
International Journal of Environmental Research and Public, 2023, 卷号: 20, 期号: 2
作者:
Yongqiang Ning
;
Bizheng Yang
;
Shaochen Yang
;
Jiaxin Ye
;
Junjie Li
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收藏
  |  
浏览/下载:10/0
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提交时间:2024/06/18
Long-term drying trend during 51.8-37.5 Ma in the Nangqian Basin, central-eastern Qinghai-Tibet Plateau
期刊论文
OAI收割
FRONTIERS IN EARTH SCIENCE, 2022, 卷号: 10, 页码: 17
作者:
Li, Shangkun
;
Ma, Xueyun
;
Jiang, Shaohua
;
Wang, Gen
;
Zhang, Ting
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2023/04/03
biomarkers
paleoclimate
paleovegetation
Nangqian Basin
Qinghai-Tibet Plateau