中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
金属研究所 [37]
上海药物研究所 [24]
青海盐湖研究所 [13]
半导体研究所 [4]
合肥物质科学研究院 [4]
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期刊论文 [100]
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2025 [6]
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2022 [8]
2021 [10]
2020 [12]
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Chemistry [2]
材料科学与物理化学 [2]
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yh.qiu@sia... [1]
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Discovery of pyrrolo[2,3-d]pyrimidine derivatives as novel FLT3/ IRAK4 inhibitors
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 296, 页码: 23
作者:
Yuan, Haibin
;
Gao, Yue
;
Wang, Peipei
;
Dong, Xiaowu
;
Li, Jia
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2025/08/20
AML
FLT3/IRAK4 inhibitor
Pyrrolo [2,3-d] pyrimidine
Acquired resistance
Adaptive resistance
Design, synthesis, and evaluation of Menin-targeting compounds for the treatment of acute Myelocytic leukemia (AML)
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 296, 页码: 17
作者:
Mo, Jun
;
Wang, Yuxian
;
Pan, Youlu
;
Xiao, Qitao
;
Zhao, Jinyi
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2025/08/20
Menin
High binding affinity
Anti-proliferation activity
AML
Proteogenomic characterization of non-functional clinically relevant subgroups
期刊论文
OAI收割
CANCER CELL, 2025, 卷号: 43, 期号: 4, 页码: 36
作者:
Ji, Shunrong
;
Cao, Lihua
;
Gao, Jing
;
Du, Yang
;
Ye, Zeng
  |  
收藏
  |  
浏览/下载:57/0
  |  
提交时间:2025/06/23
Development of novel epoxyketone macrocyclic peptidyl proteasome inhibitors through OPA-mediated one-step cyclization of unprotected peptides
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2025, 卷号: 156, 页码: 16
作者:
Zeng, Gongruixue
;
Xu, Gaoya
;
Gao, Lixin
;
Zheng, Xiaoli
;
Chi, Xinglong
  |  
收藏
  |  
浏览/下载:65/0
  |  
提交时间:2025/04/01
Proteasome inhibitors
Macrocycle
Stability
Anti-cancer activities
Discovery of a potential hematologic malignancies therapy: Selective and potent HDAC7 PROTAC degrader targeting non-enzymatic function
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2025, 卷号: 15, 期号: 3, 页码: 1659-1679
作者:
Jin, Yuheng
;
Qi, Xuxin
;
Yu, Xiaoli
;
Cheng, Xirui
;
Chen, Boya
  |  
收藏
  |  
浏览/下载:43/0
  |  
提交时间:2025/06/23
HDAC7
PROTAC
Selectivity
Hematologic malignancies
Non-enzymatic function
Auto-RapTAC: A Versatile and Sustainable Platform for the Automated Rapid Synthesis and Evaluation of PROTAC
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 页码: 15
作者:
Chen, Jiexuan
;
Wu, Mingfei
;
Mo, Jun
;
Hong, Ju
;
Wang, Wei
  |  
收藏
  |  
浏览/下载:65/0
  |  
提交时间:2025/04/01
Exploration of novel 20S proteasome activators featuring anthraquinone structures and their application in hypoxic cardiomyocyte protection
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2024, 卷号: 115, 页码: 10
作者:
Yu, Qian
;
Gao, Lixin
;
Xu, Linhao
;
Han, Yubing
;
Cao, Yu
  |  
收藏
  |  
浏览/下载:74/0
  |  
提交时间:2024/12/11
Dynamic fatigue damage behaviors and mechanisms of overhead transmission Al wires at elevated temperatures
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF FATIGUE, 2024, 卷号: 188, 页码: 12
作者:
Wang, Shuo
;
Hou, Jiapeng
;
Li, Chenghui
;
Gong, Baishan
;
Liu, Hanzhong
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2025/04/27
Overhead Al wires
Elevated temperature
Dynamic fatigue
Damage mechanism
Fatigue strength prediction
Dynamic fatigue damage behaviors and mechanisms of overhead transmission Al wires at elevated temperatures
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF FATIGUE, 2024, 卷号: 188, 页码: 12
作者:
Wang, Shuo
;
Hou, Jiapeng
;
Li, Chenghui
;
Gong, Baishan
;
Liu, Hanzhong
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2025/04/27
Overhead Al wires
Elevated temperature
Dynamic fatigue
Damage mechanism
Fatigue strength prediction
Dynamic fatigue damage behaviors and mechanisms of overhead transmission Al wires at elevated temperatures
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF FATIGUE, 2024, 卷号: 188, 页码: 12
作者:
Wang, Shuo
;
Hou, Jiapeng
;
Li, Chenghui
;
Gong, Baishan
;
Liu, Hanzhong
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2025/04/27
Overhead Al wires
Elevated temperature
Dynamic fatigue
Damage mechanism
Fatigue strength prediction