中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共25条,第1-10条 帮助

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Discovery of Novel 2-Aminopyridine-Based and 2-Aminopyrimidine-Based Derivatives as Potent CDK/HDAC Dual Inhibitors for the Treatment of Refractory Solid Tumors and Hematological Malignancies 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 17, 页码: 15220-15245
作者:  
Saidahmatov, Abdusaid;  Li, Jianan;  Xu, Shihao;  Hu, Xiaobei;  Gao, Xiangqian
  |  收藏  |  浏览/下载:27/0  |  提交时间:2024/10/21
Targeting C/EBP alpha overcomes primary resistance and improves the efficacy of FLT3 inhibitors in acute myeloid leukaemia 期刊论文  OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 18
作者:  
Wang, Hanlin;  Luo, Guanghao;  Hu, Xiaobei;  Xu, Gaoya;  Wang, Tao
  |  收藏  |  浏览/下载:29/0  |  提交时间:2023/10/17
In vitro and in vivo evaluation of the main protease inhibitor FB2001 against SARS-CoV-2 期刊论文  OAI收割
ANTIVIRAL RESEARCH, 2022, 卷号: 208, 页码: 10
作者:  
Shang, Weijuan;  Dai, Wenhao;  Yao, Cheng;  Xu, Ling;  Tao, Xiangming
  |  收藏  |  浏览/下载:32/0  |  提交时间:2023/04/10
Discovery of Novel N-(5-(Pyridin-3-yl)-1H-indazol-3-yl)benzamide Derivatives as Potent Cyclin-Dependent Kinase 7 Inhibitors for the Treatment of Autosomal Dominant Polycystic Kidney Disease 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 19
作者:  
Yang, Bowen;  Zhang, Haoran;  Li, Na;  Gao, Lixin;  Jiang, Hong
  |  收藏  |  浏览/下载:37/0  |  提交时间:2023/04/10
Matrix stiffness exacerbates the proinflammatory responses of vascular smooth muscle cell through the DDR1-DNMT1 mechanotransduction axis 期刊论文  OAI收割
BIOACTIVE MATERIALS, 2022, 卷号: 17, 页码: 406-424
作者:  
Wang, Jin;  Xie, Si-an;  Li, Ning;  Zhang, Tao;  Yao, Weijuan
  |  收藏  |  浏览/下载:55/0  |  提交时间:2022/06/10
A Modified Temperature-Vegetation Dryness Index (MTVDI) for Assessment of Surface Soil Moisture Based on MODIS Data 期刊论文  OAI收割
CHINESE GEOGRAPHICAL SCIENCE, 2022, 卷号: 32, 期号: 4, 页码: 592-605
作者:  
Wang, Hao;  Li, Zongshan;  Zhang, Weijuan;  Ye, Xin;  Liu, Xianfeng
  |  收藏  |  浏览/下载:20/0  |  提交时间:2022/11/07
Structure-Activity Relationship Study of Indolin-5-yl-cyclopropanamine Derivatives as Selective Lysine Specific Demethylase 1 (LSD1) Inhibitors 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 5, 页码: 4335-4349
作者:  
Li, Chunpu;  Su, Mingbo;  Zhu, Wei;  Kan, Weijuan;  Ge, Tianpeng
  |  收藏  |  浏览/下载:52/0  |  提交时间:2022/06/15
Inner nuclear membrane protein TMEM201 promotes breast cancer metastasis by positive regulating TGF beta signaling 期刊论文  OAI收割
ONCOGENE, 2021, 页码: 10
作者:  
Kong, Ya;  Zhang, Yutian;  Wang, Hanlin;  Kan, Weijuan;  Guo, Haoran
  |  收藏  |  浏览/下载:52/0  |  提交时间:2022/01/04
Discovery and Development of a Potent, Selective, and Orally Bioavailable CHK1 Inhibitor Candidate: 5-((4-((3-Amino-3-methylbutyl)amino)-5-(trifluoromethyl)pyrimidin-2-yl)amino)picolinonitrile 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 20, 页码: 15069-15090
作者:  
Jin, Tingting;  Xu, Lei;  Wang, Peipei;  Hu, Xiaobei;  Zhang, Runyuan
  |  收藏  |  浏览/下载:30/0  |  提交时间:2022/01/04
Rational Design and Development of Novel CDK9 Inhibitors for the Treatment of Acute Myeloid Leukemia 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 19, 页码: 14647-14663
作者:  
Han, Xu;  Song, Ning;  Saidahmatov, Abdusaid;  Wang, Peipei;  Wang, Yong
  |  收藏  |  浏览/下载:83/0  |  提交时间:2021/12/16