中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共10条,第1-10条 帮助

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Selective Degradation of TEADs by a PROTAC Molecule Exhibited Robust Anticancer Efficacy In Vitro and In Vivo 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 页码: 25
作者:  
Lu, Yuhang;  Yan, Ziqin;  Sun, Jiaqi;  Wang, Chenxu;  Xu, Lan
  |  收藏  |  浏览/下载:9/0  |  提交时间:2025/04/01
Discovery of a Covalent Inhibitor That Overcame Resistance to Venetoclax in AML Cells Overexpressing BFL-1 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 36
作者:  
Lou, Jianfeng;  Zhou, Qianqian;  Lyu, Xilin;  Cen, Xinyi;  Liu, Chen
  |  收藏  |  浏览/下载:5/0  |  提交时间:2024/08/22
Selective degradation of cellular BRD3 and BRD4-L promoted by PROTAC molecules in six cancer cell lines 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 254, 页码: 17
作者:  
Yan, Ziqin;  Lyu, Xilin;  Lin, Dongze;  Wu, Gaoxing;  Gong, Yang
  |  收藏  |  浏览/下载:44/0  |  提交时间:2023/10/17
A chemical perspective on the modulation of TEAD transcriptional activities: Recent progress, challenges, and opportunities 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 243, 页码: 31
作者:  
Lou, Jianfeng;  Lu, Yuhang;  Cheng, Jing;  Zhou, Feilong;  Yan, Ziqin
  |  收藏  |  浏览/下载:37/0  |  提交时间:2022/12/13
Discovery of a selective and covalent small-molecule inhibitor of BFL-1 protein that induces robust apoptosis in cancer cells 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 236, 页码: 114327
作者:  
Feng, Xuexin;  Yan, Ziqin;  Zhou, Feilong;  Lou, Jianfeng;  Lyu, Xilin
  |  收藏  |  浏览/下载:38/0  |  提交时间:2024/03/21
Structure-Based Discovery of MDM2/4 Dual Inhibitors that Exert Antitumor Activities against MDM4-Overexpressing Cancer Cells 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 8, 页码: 6207-6230
作者:  
Zhang, Shiyan;  Yan, Ziqin;  Li, Yafang;  Gong, Yang;  Lyu, Xilin
  |  收藏  |  浏览/下载:38/0  |  提交时间:2022/08/16
Material properties of phase-separated TFEB condensates regulate the autophagy-lysosome pathway 期刊论文  OAI收割
JOURNAL OF CELL BIOLOGY, 2022, 卷号: 221, 期号: 5, 页码: 27
作者:  
Wang, Zheng;  Chen, Di;  Guan, Dongshi;  Liang, Xiaobo;  Xue, Jianfeng
  |  收藏  |  浏览/下载:37/0  |  提交时间:2022/11/14
Recent Progress and Clinical Development of Inhibitors that Block MDM4/p53 Protein-Protein Interactions 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 15, 页码: 10621-10640
作者:  
Zhang, Shiyan;  Lou, Jianfeng;  Li, Yafang;  Zhou, Feilong;  Yan, Ziqin
  |  收藏  |  浏览/下载:38/0  |  提交时间:2021/11/04
Mapping diffuse emission in lyman UV band 会议论文  OAI收割
Virtual, Online, CA, United states, 2020-12-14
作者:  
Ji, Li
  |  收藏  |  浏览/下载:47/0  |  提交时间:2021/02/05
Heterogeneous mutation pattern in tumor tissue and circulating tumor DNA warrants parallel NGS panel testing 期刊论文  OAI收割
MOLECULAR CANCER, 2018, 卷号: 17, 期号: 1, 页码: 131
作者:  
Guo, Qiaomei;  Wang, Lin;  Hu, Xiaomeng;  Yu, Wenjun;  Lou, Jiatao
  |  收藏  |  浏览/下载:112/0  |  提交时间:2019/04/28