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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
广州能源研究所 [22]
上海药物研究所 [11]
金属研究所 [7]
海洋研究所 [2]
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期刊论文 [53]
CNKI期刊论文 [1]
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2025 [1]
2024 [6]
2023 [2]
2022 [3]
2021 [15]
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学科主题
Biochemist... [1]
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浏览/检索结果:
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Harnessing the Magic Methyl Effect: Discovery of CLPP-2068 as a Novel
Hs
ClpP Activator for the Treatment of Diffuse Large B-Cell Lymphoma
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 4, 页码: 4287-4307
作者:
Sun, Mingyang
;
Chen, Beijing
;
Teng, Dan
;
Zhao, Hongshen
;
Liao, Yilie
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2025/04/01
Discovery of CLPP-1071 as an Exceptionally Potent and Orally Efficacious Human ClpP Activator with Strong In Vivo Antitumor Activity
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 21
作者:
Chen, Beijing
;
Sun, Mingyang
;
Zhang, Chun
;
Huang, Qi
;
Teng, Dan
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2024/12/25
An updated patent review of SOS1 inhibitors (2022-present)
期刊论文
OAI收割
EXPERT OPINION ON THERAPEUTIC PATENTS, 2024, 页码: 15
作者:
Zhou, Guizhen
;
Zhou, Chuan
;
Ma, Xinyi
;
Xu, Jiahang
;
Zhou, Zehui
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2024/12/11
SOS1
KRAS
cancer
inhibitor
drug discovery
Amelioration of nonalcoholic fatty liver disease by inhibiting the deubiquitylating enzyme RPN11
期刊论文
OAI收割
CELL METABOLISM, 2024, 卷号: 36, 期号: 10, 页码: 25
作者:
Zhou, Bing
;
Luo, Yunchen
;
Bi, Hanqi
;
Zhang, Ni
;
Ma, Mingyue
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/11/26
Targeting STING oligomerization with licochalcone D ameliorates STING-driven inflammatory diseases
期刊论文
OAI收割
SCIENCE CHINA-LIFE SCIENCES, 2024, 页码: 14
作者:
Zhang, Yinghui
;
Liu, Yadan
;
Jiang, Bing
;
Chen, Lifan
;
Hu, Jie
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2024/10/21
cGAS-STING signaling
STING inhibitor
TransformerCPI model
Licochalcone D
inflammatory diseases
Design, synthesis, and bioevaluation of SOS1 PROTACs derived from pyrido [2,3-
d
]pyrimidin-7-one-based SOS1 inhibitor
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2024, 卷号: 107, 页码: 9
作者:
Wang, Kun
;
Zhou, Zehui
;
Ma, Xinyi
;
Xu, Jiahang
;
Xu, Wangyang
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2024/07/12
SOS1
KRAS mutation
PROTAC
Anti-cancer activity
Structure-based design of pan-coronavirus inhibitors targeting host cathepsin L and calpain-1
期刊论文
OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2024, 卷号: 9, 期号: 1, 页码: 14
作者:
Xie, Xiong
;
Lan, Qiaoshuai
;
Zhao, Jinyi
;
Zhang, Sulin
;
Liu, Lu
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2024/05/07
Precise measurement method of carrier motion state in microgravity environment
期刊论文
OAI收割
MEASUREMENT, 2023, 卷号: 222, 页码: 17
作者:
Liu, Mingyue
;
Zhu, Huizhong
;
Xu, Xinchao
;
Ma, Youqing
;
Zhang, Shuo
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2023/11/28
Multi-camera calibration
Stereo vision
Extraction of homonymous points
Random Sample Consensus (RANSAC)
Carrier motion state
Sequence-based drug design as a concept in computational drug design
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 21
作者:
Chen, Lifan
;
Fan, Zisheng
;
Chang, Jie
;
Yang, Ruirui
;
Hou, Hui
  |  
收藏
  |  
浏览/下载:44/0
  |  
提交时间:2023/10/17
Low-oxygen rare earth steels
期刊论文
OAI收割
NATURE MATERIALS, 2022, 页码: 9
作者:
Li, Dianzhong
;
Wang, Pei
;
Chen, Xing-Qiu
;
Fu, Paixian
;
Luan, Yikun
  |  
收藏
  |  
浏览/下载:54/0
  |  
提交时间:2022/10/08