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	Discovery of novel 3-hydroxypicolinamides as selective inhibitors of HIV-1 integrase-LEDGF/p75 interaction 期刊论文 OAI收割 European Journal of Medicinal Chemistry, 2017, 卷号: 125, 期号: X, 页码: 1051-1063 作者: Zhang FH; Debnath B; Zheng YT; Neamati N[]; Long YQ[] 收藏 \| 浏览/下载：78/0 \| 提交时间：2016/11/07 3-Hydroxypicolinamide Allosteric inhibitor Dimerization HIV-1 integrase LEDGF/p75
	Design and discovery of flavonoid-based HIV-1 integrase inhibitors targeting both the active site and the interaction with LEDGF/p75 期刊论文 OAI收割 BIOORGANIC & MEDICINAL CHEMISTRY, 2014, 卷号: 22, 期号: 12, 页码: 3146-3158 作者: Li BW; Zhang FH; Serrao E; Chen H; Sanchez TW 收藏 \| 浏览/下载：12/0 \| 提交时间：2014/10/15 Chelation Strand transfer LEDGF/p75 HIV-1 integrase inhibitors Flavonoid
	Repositioning HIV‑1 Integrase Inhibitors for Cancer Therapeutics: 1,6-Naphthyridine-7-carboxamide as a Promising Scaffold with Drug-like Properties 期刊论文 OAI收割 JOURNAL OF MEDICINAL CHEMISTRY, 2012, 卷号: 55, 期号: 22, 页码: 9492-9509 作者: Zeng LF; Wang Y; Kazemi R; Xu SL; Xu ZL 收藏 \| 浏览/下载：20/0 \| 提交时间：2013/04/09
	Efficient synthesis and utilization of phenyl-substituted heteroaromatic carboxylic acids as aryl diketo acid isosteres in the design of novel HIV-1 integrase inhibitors 期刊论文 OAI收割 BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2008, 卷号: 18, 期号: 16, 页码: 4521-4524 作者: Zeng LF; Zhang HS; Wang YH; Sanchez T; Zheng YT 收藏 \| 浏览/下载：24/0 \| 提交时间：2010/08/24 HIV-1 integrase inhibitor bioisostere heteroaromatic carboxylic acid isoxazole isothiazole 1H-pyrazole bioavailability antiviral effect
	Rational design and synthesis of novel dimeric diketoacid-containing inhibitors of HIV-1 integrase: Implication for binding to two metal ions on the active site of integrase 期刊论文 OAI收割 JOURNAL OF MEDICINAL CHEMISTRY, 2004, 卷号: 47, 期号: 10, 页码: 2561-2573 作者: Long, YQ; Jiang, XH; Dayam, R; Sanchez, T; Shoemaker, R \| 收藏 \| 浏览/下载：15/0 \| 提交时间：2019/01/08