中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [4]
地球环境研究所 [2]
采集方式
OAI收割 [6]
内容类型
期刊论文 [6]
发表日期
2024 [2]
2022 [1]
2021 [1]
2018 [2]
学科主题
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Design and development of a series of 4-(piperazin-1-yl)pyrimidines as irreversible menin inhibitors
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 280, 页码: 20
作者:
Luo, Menglan
;
Ye, Yunfei
;
Tang, Lu
;
Kan, Weijuan
;
Chen, Lin
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/11/26
Menin
Covalent inhibitor
Antitumor
Degradation
Discovery of Novel 2-Aminopyridine-Based and 2-Aminopyrimidine-Based Derivatives as Potent CDK/HDAC Dual Inhibitors for the Treatment of Refractory Solid Tumors and Hematological Malignancies
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 17, 页码: 15220-15245
作者:
Saidahmatov, Abdusaid
;
Li, Jianan
;
Xu, Shihao
;
Hu, Xiaobei
;
Gao, Xiangqian
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2024/10/21
Structure-Activity Relationship Study of Indolin-5-yl-cyclopropanamine Derivatives as Selective Lysine Specific Demethylase 1 (LSD1) Inhibitors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 5, 页码: 4335-4349
作者:
Li, Chunpu
;
Su, Mingbo
;
Zhu, Wei
;
Kan, Weijuan
;
Ge, Tianpeng
  |  
收藏
  |  
浏览/下载:46/0
  |  
提交时间:2022/06/15
Identification of pyrogallol as a warhead in design of covalent inhibitors for the SARS-CoV-2 3CL protease
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2021, 卷号: 12, 期号: 1, 页码: 12
作者:
Su, Haixia
;
Yao, Sheng
;
Zhao, Wenfeng
;
Zhang, Yumin
;
Liu, Jia
  |  
收藏
  |  
浏览/下载:64/0
  |  
提交时间:2021/08/17
Carbon isotopic composition of branched tetraether membrane lipids in a loess-paleosol sequence and its geochemical significance
期刊论文
OAI收割
Palaeogeography, Palaeoclimatology, Palaeoecology, 2018, 卷号: 504, 页码: 150-155
作者:
Sheng, WJ (Sheng, Weijuan)[ 1 ]
;
Liu, WG (Liu, Weiguo)[ 1,2 ]
;
Lu, HX (Lu, Hongxuan)[ 1 ]
  |  
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2018/11/21
GDGTs
Paleovegetation
Microbiological degradation
Heterotrophism
Total organic carbon
Carbon isotopic composition of branched tetraether membrane lipids in a loess-paleosol sequence and its geochemical significance
期刊论文
OAI收割
Palaeogeography, Palaeoclimatology, Palaeoecology, 2018, 卷号: 504, 页码: 150-155
作者:
Lu, HX (Lu, Hongxuan)[ 1 ]
;
Liu, WG (Liu, Weiguo)[ 1,2 ]
;
Sheng, WJ (Sheng, Weijuan)[ 1 ]
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2018/11/20
Gdgts
Paleovegetation
Microbiological Degradation
Heterotrophism
Total Organic Carbon