中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
广州生物医药与健康研... [8]
上海药物研究所 [2]
采集方式
OAI收割 [10]
内容类型
期刊论文 [10]
发表日期
2021 [1]
2015 [7]
2014 [2]
学科主题
Pharmacolo... [6]
Chemistry [4]
Biochemist... [2]
Oncology [2]
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TANK-binding kinase 1 (TBK1): An emerging therapeutic target for drug discovery
期刊论文
OAI收割
DRUG DISCOVERY TODAY, 2021, 卷号: 26, 期号: 10, 页码: 2445-2455
作者:
Xiang, Shuang
;
Song, Shukai
;
Tang, Haotian
;
Smaill, Jeff B.
;
Wang, Aiqun
  |  
收藏
  |  
浏览/下载:48/0
  |  
提交时间:2021/12/01
Antibiotic resistance
Computational biology
Databases
In silico tools
2,4-Diarylamino-pyrimidines as kinase inhibitors co-targeting IGF1R and EGFR(L858R/T790M)
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 19, 页码: 4277-4281
作者:
Chan, Shingpan
;
Han, Kun
;
Qu, Rong
;
Tong, Linjiang
;
Li, Yingjun
  |  
收藏
  |  
浏览/下载:51/0
  |  
提交时间:2019/01/08
EGFR
IGF1R
NSCLC
Dual inhibitor
2,4-Diarylamino-pyrimidines as kinase inhibitors co-targeting IGF1R and EGFR(L858R/T790M)
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 19, 页码: 4277-4281
Chan, Shingpan
;
Han, Kun
;
Qu, Rong
;
Tong, Linjiang
;
Li, Yingjun
;
Zhang, Zhang
;
Cheng, Huimin
;
Lu, Xiaoyun
;
Patterson, Adam
;
Smaill, Jeff
;
Ren, Xiaomei
;
Ding, Jian
;
Xie, Hua
;
Ding, Ke
收藏
  |  
浏览/下载:253/0
  |  
提交时间:2016/12/16
2,4-Diarylamino-pyrimidines as kinase inhibitors co-targeting IGF1R and EGFR(L858R/T790M)
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 19, 页码: 4277-4281
作者:
Smaill, Jeff
;
Lu, Xiaoyun
;
Cheng, Huimin
;
Zhang, Zhang
;
Li, Yingjun
  |  
收藏
  |  
浏览/下载:57/0
  |  
提交时间:2018/12/13
N-(3-Ethynyl-2,4-difluorophenyl)sulfonamide Derivatives as Selective Raf Inhibitors
期刊论文
OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 6, 期号: 5, 页码: 543-547
作者:
Ding, Ke
;
Cheng, Huimin
;
Zhang, Zhang
;
Zhuang, Xiaoxi
;
Li, Yingjun
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2018/12/13
1-Benzyl-4-phenyl-1H-1,2,3-triazoles improve the transcriptional functions of estrogen-related receptor gamma and promote the browning of white adipose
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2015, 卷号: 23, 期号: 13, 页码: 3751-3760
作者:
Yu, Lei
;
Xu, Shilin
;
Mao, Liufeng
;
Ding, Ping
;
Zhuang, Xiaoxi
  |  
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2018/12/13
1-Benzyl-4-phenyl-1H-1,2,3-triazoles improve the transcriptional functions of estrogen-related receptor gamma and promote the browning of white adipose
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2015, 卷号: 23, 期号: 13, 页码: 3751-3760
Xu, Shilin
;
Mao, Liufeng
;
Ding, Ping
;
Zhuang, Xiaoxi
;
Zhou, Yang
;
Yu, Lei
;
Liu, Yingxue
;
Nie, Tao
;
Xu, Tingting
;
Xu, Yong
;
Liu, Jinsong
;
Smaill, Jeff
;
Ren, Xiaomei
;
Wu, Donghai
;
Ding, Ke
收藏
  |  
浏览/下载:49/0
  |  
提交时间:2016/12/16
N-(3-Ethynyl-2,4-difluorophenyl)sulfonamide Derivatives as Selective Raf Inhibitors
期刊论文
OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 6, 期号: 5, 页码: 543-547
Li, Yingjun
;
Cheng, Huimin
;
Zhang, Zhang
;
Zhuang, Xiaoxi
;
Luo, Jinfeng
;
Long, Huoyou
;
Zhou, Yang
;
Xu, Yong
;
Taghipouran, Rana
;
Li, Dan
;
Patterson, Adam
;
Smaill, Jeff
;
Tu, Zhengchao
;
Wu, Donghai
;
Ren, Xiaomei
;
Ding, Ke
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2016/12/16
Bioreductive prodrugs as cancer therapeutics: targeting tumor hypoxia
期刊论文
OAI收割
CHINESE JOURNAL OF CANCER, 2014, 卷号: 33, 期号: 2
作者:
Patterson, Adam V.
;
Guise, Christopher P.
;
Mowday, Alexandra M.
;
Ashoorzadeh, Amir
;
Yuan, Ran
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2018/12/13
Bioreductive prodrugs as cancer therapeutics: targeting tumor hypoxia
期刊论文
OAI收割
CHINESE JOURNAL OF CANCER, 2014, 卷号: 33, 期号: 2
Guise, Christopher P.
;
Mowday, Alexandra M.
;
Ashoorzadeh, Amir
;
Yuan, Ran
;
Lin, Wan-Hua
;
Wu, Dong-Hai
;
Smaill, Jeff B.
;
Patterson, Adam V.
;
Ding, Ke
收藏
  |  
浏览/下载:96/0
  |  
提交时间:2016/12/16