中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
首页
机构
成果
学者
登录
注册
登陆
×
验证码:
换一张
忘记密码?
记住我
×
校外用户登录
CAS IR Grid
机构
广州生物医药与健康研... [9]
金属研究所 [2]
上海药物研究所 [1]
大连化学物理研究所 [1]
南京地理与湖泊研究所 [1]
采集方式
OAI收割 [14]
内容类型
期刊论文 [14]
发表日期
2022 [1]
2021 [2]
2018 [1]
2016 [5]
2013 [5]
学科主题
Pharmacolo... [4]
Science & ... [2]
筛选
浏览/检索结果:
共14条,第1-10条
帮助
条数/页:
5
10
15
20
25
30
35
40
45
50
55
60
65
70
75
80
85
90
95
100
排序方式:
请选择
题名升序
题名降序
提交时间升序
提交时间降序
作者升序
作者降序
发表日期升序
发表日期降序
Changes of the physicochemical properties of extracellular polymeric substances (EPS) from Microcystis aeruginosa in response to microplastics
期刊论文
OAI收割
ENVIRONMENTAL POLLUTION, 2022, 卷号: 315
作者:
Ye, Tianran
;
Yang, Ao
;
Wang, Yulai
;
Song, Na
;
Wang, Ping
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2023/12/19
A new designed method for evaluating the repairability of a newly developed 5Cr5MoV cold working die steel
期刊论文
OAI收割
AIP ADVANCES, 2021, 卷号: 11, 期号: 3, 页码: 8
作者:
Liang, Yan
;
Wang, Qiang
;
Song, Yulai
;
Liu, Yaohui
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2021/10/15
A new designed method for evaluating the repairability of a newly developed 5Cr5MoV cold working die steel
期刊论文
OAI收割
AIP ADVANCES, 2021, 卷号: 11, 期号: 3, 页码: 8
作者:
Liang, Yan
;
Wang, Qiang
;
Song, Yulai
;
Liu, Yaohui
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2021/10/15
Y08060: A Selective BET Inhibitor for Treatment of Prostate Cancer
期刊论文
OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2018, 卷号: 9, 期号: 3, 页码: 262-267
作者:
Xiang, Quping
;
Zhang, Yan
;
Li, Jiaguo
;
Xue, Xiaoqian
;
Wang, Chao
  |  
收藏
  |  
浏览/下载:47/0
  |  
提交时间:2019/06/20
Bromodomain
Brd4
Prostate Cancer
Epigenetics
Discovery of Benzo[cd]indol-2(1H)-ones as Potent and Specific BET Bromodomain Inhibitors: Structure-Based Virtual Screening, Optimization, and Biological Evaluation
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 4, 页码: 1565-1579
作者:
Tu, Zhengchao
;
Zhou, Yulai
;
Ding, Ke
;
Xu, Yong
;
Xue, Xiaoqian
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2018/12/13
Identification of N-phenyl-2-(N-phenylphenylsulfonamido) acetamides as new ROR gamma inverse agonists: Virtual screening, structure-based optimization, and biological evaluation
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 116, 页码: 13-26
作者:
Xue, Xiaoqian
;
Song, Yu
;
Qian, Chao-Nan
;
Yan, Weiqun
;
Xing, Yanli
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2018/12/13
Discovery of Benzo[cd]indol-2(1H)-ones as Potent and Specific BET Bromodomain Inhibitors: Structure-Based Virtual Screening, Optimization, and Biological Evaluation
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 4, 页码: 1565-1579
Xue, Xiaoqian
;
Zhang, Yan
;
Liu, Zhaoxuan
;
Song, Ming
;
Xing, Yanli
;
Xiang, Qiuping
;
Wang, Zhen
;
Tu, Zhengchao
;
Zhou, Yulai
;
Ding, Ke
;
Xu, Yong
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2016/12/16
Identification of N-phenyl-2-(N-phenylphenylsulfonamido) acetamides as new ROR gamma inverse agonists: Virtual screening, structure-based optimization, and biological evaluation
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 116, 页码: 13-26
Song, Yu
;
Xue, Xiaoqian
;
Wu, Xishan
;
Wang, Rui
;
Xing, Yanli
;
Yan, Weiqun
;
Zhou, Yulai
;
Qian, Chao-Nan
;
Zhang, Yan
;
Xu, Yong
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2016/12/16
Discovery and structural optimization of 4-(4-(benzyloxy) phenyl)-3,4-dihydropyrimidin-2(1H)-ones as RORc inverse agonists
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2016, 卷号: 37, 期号: 11, 页码: 1516
作者:
Wu Xishan
;
Wang Rui
;
Xing Yanli
;
Xue Xiaoqian
;
Zhang Yan
  |  
收藏
  |  
浏览/下载:94/0
  |  
提交时间:2020/12/24
GAMMA-T
ORPHAN RECEPTORS
CELL-DIFFERENTIATION
LIGAND
IDENTIFICATION
MODULATORS
DERIVATIVES
PROTEIN
INHIBITORS
DOCKING
nuclear receptor
RORc
inverse agonist
SAR
structure-based optimization
autoimmune disease
Enhanced Production of Recombinant Secretory Proteins in Pichia pastoris by Optimizing Kex2 P1' site
期刊论文
OAI收割
PLOS ONE, 2013, 卷号: 8, 期号: 9
作者:
Zhou, Yulai
;
Wang, Yu
;
Xu, Aimin
;
Li, Shiwu
;
Liu, Pentao
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2018/12/13