中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共248条,第1-10条 帮助

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Discovery of novel selective PRMT5-MTA inhibitors through structure-based virtual screening 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2026, 卷号: 168, 页码: 17
作者:  
Ma, Ning;  Chen, Yang;  Liang, Yiru;  Chen, Xiaoxu;  Song, Fengnan
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Furo[2,3-f]quinazolin-7(6H)-one Derivatives as Potent, Selective, and Orally Bioavailable MAT2A Inhibitors for MTAP-Deficient Cancer Therapy 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 22, 页码: 24213-24231
作者:  
Shi, Zihan;  Lin, Kexin;  Lin, Lijie;  Chen, Zhiyi;  Xie, Zhiyin
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Discovery of 3-(Fluoro-imidazolyl)pyridazine Derivatives as Potent STING Agonists with Antitumor Activity 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 10, 页码: 9864-9885
作者:  
Hou, Hui;  Zhou, Jingyi;  Sui, Qibang;  Zhang, Changfa;  Su, Zhaoming
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Targeting the histone reader ZMYND8 inhibits antiandrogen-induced neuroendocrine tumor transdifferentiation of prostate cancer 期刊论文  OAI收割
NATURE CANCER, 2025, 页码: 37
作者:  
Wang, Hanling;  Zhang, Sulin;  Pan, Qiang;  Guo, Jiacheng;  Li, Ni
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Discovery of novel covalent stabilizers for p53 Y220C using structure-based drug discovery methods 期刊论文  OAI收割
MOLECULAR DIVERSITY, 2025, 页码: 14
作者:  
Wen, Yiming
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SurfDock is a surface-informed diffusion generative model for reliable and accurate protein-ligand complex prediction 期刊论文  OAI收割
NATURE METHODS, 2024, 页码: 24
作者:  
Cao, Duanhua;  Chen, Mingan;  Zhang, Runze;  Wang, Zhaokun;  Huang, Manlin
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Identifying compound-protein interactions with knowledge graph embedding of perturbation transcriptomics 期刊论文  OAI收割
CELL GENOMICS, 2024, 卷号: 4, 期号: 10, 页码: 100655
作者:  
Ni, Shengkun;  Kong, Xiangtai;  Zhang, Yingying;  Chen, Zhengyang;  Wang, Zhaokun
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Targeting STING oligomerization with licochalcone D ameliorates STING-driven inflammatory diseases 期刊论文  OAI收割
SCIENCE CHINA-LIFE SCIENCES, 2024, 页码: 14
作者:  
Zhang, Yinghui;  Liu, Yadan;  Jiang, Bing;  Chen, Lifan;  Hu, Jie
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Generic protein-ligand interaction scoring by integrating physical prior knowledge and data augmentation modelling 期刊论文  OAI收割
NATURE MACHINE INTELLIGENCE, 2024, 页码: 21
作者:  
Cao, Duanhua;  Chen, Geng;  Jiang, Jiaxin;  Yu, Jie;  Zhang, Runze
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KinomeMETA: a web platform for kinome-wide polypharmacology profiling with meta-learning 期刊论文  OAI收割
NUCLEIC ACIDS RESEARCH, 2024, 页码: 9
作者:  
Li, Zhaojun;  Qu, Ning;  Zhou, Jingyi;  Sun, Jingjing;  Ren, Qun
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