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Chinese Academy of Sciences Institutional Repositories Grid
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高能物理研究所 [167]
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期刊论文 [248]
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2026 [1]
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Physics [1]
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Discovery of novel selective PRMT5-MTA inhibitors through structure-based virtual screening
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2026, 卷号: 168, 页码: 17
作者:
Ma, Ning
;
Chen, Yang
;
Liang, Yiru
;
Chen, Xiaoxu
;
Song, Fengnan
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Furo[2,3-
f
]quinazolin-7(6
H
)-one Derivatives as Potent, Selective, and Orally Bioavailable MAT2A Inhibitors for MTAP-Deficient Cancer Therapy
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 22, 页码: 24213-24231
作者:
Shi, Zihan
;
Lin, Kexin
;
Lin, Lijie
;
Chen, Zhiyi
;
Xie, Zhiyin
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Discovery of 3-(Fluoro-imidazolyl)pyridazine Derivatives as Potent STING Agonists with Antitumor Activity
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 10, 页码: 9864-9885
作者:
Hou, Hui
;
Zhou, Jingyi
;
Sui, Qibang
;
Zhang, Changfa
;
Su, Zhaoming
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Targeting the histone reader ZMYND8 inhibits antiandrogen-induced neuroendocrine tumor transdifferentiation of prostate cancer
期刊论文
OAI收割
NATURE CANCER, 2025, 页码: 37
作者:
Wang, Hanling
;
Zhang, Sulin
;
Pan, Qiang
;
Guo, Jiacheng
;
Li, Ni
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Discovery of novel covalent stabilizers for p53 Y220C using structure-based drug discovery methods
期刊论文
OAI收割
MOLECULAR DIVERSITY, 2025, 页码: 14
作者:
Wen, Yiming
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SurfDock is a surface-informed diffusion generative model for reliable and accurate protein-ligand complex prediction
期刊论文
OAI收割
NATURE METHODS, 2024, 页码: 24
作者:
Cao, Duanhua
;
Chen, Mingan
;
Zhang, Runze
;
Wang, Zhaokun
;
Huang, Manlin
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Identifying compound-protein interactions with knowledge graph embedding of perturbation transcriptomics
期刊论文
OAI收割
CELL GENOMICS, 2024, 卷号: 4, 期号: 10, 页码: 100655
作者:
Ni, Shengkun
;
Kong, Xiangtai
;
Zhang, Yingying
;
Chen, Zhengyang
;
Wang, Zhaokun
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Targeting STING oligomerization with licochalcone D ameliorates STING-driven inflammatory diseases
期刊论文
OAI收割
SCIENCE CHINA-LIFE SCIENCES, 2024, 页码: 14
作者:
Zhang, Yinghui
;
Liu, Yadan
;
Jiang, Bing
;
Chen, Lifan
;
Hu, Jie
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Generic protein-ligand interaction scoring by integrating physical prior knowledge and data augmentation modelling
期刊论文
OAI收割
NATURE MACHINE INTELLIGENCE, 2024, 页码: 21
作者:
Cao, Duanhua
;
Chen, Geng
;
Jiang, Jiaxin
;
Yu, Jie
;
Zhang, Runze
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KinomeMETA: a web platform for kinome-wide polypharmacology profiling with meta-learning
期刊论文
OAI收割
NUCLEIC ACIDS RESEARCH, 2024, 页码: 9
作者:
Li, Zhaojun
;
Qu, Ning
;
Zhou, Jingyi
;
Sun, Jingjing
;
Ren, Qun
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