中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
机构
采集方式
内容类型
发表日期
学科主题
筛选

浏览/检索结果: 共42条,第1-10条 帮助

条数/页: 排序方式:
Discovery and Identification of a Novel PORCN Inhibitor via Structure-Based Virtual Screening 期刊论文  OAI收割
ACS CHEMICAL BIOLOGY, 2025, 卷号: 20, 期号: 6, 页码: 1319-1332
作者:  
Yang, Xinyu;  Li, Yanbei;  Zhou, Jingyi;  Zhou, Yuanyang;  Lin, Kexin
  |  收藏  |  浏览/下载:10/0  |  提交时间:2025/07/25
Discovery of 3-(Fluoro-imidazolyl)pyridazine Derivatives as Potent STING Agonists with Antitumor Activity 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 10, 页码: 9864-9885
作者:  
Hou, Hui;  Zhou, Jingyi;  Sui, Qibang;  Zhang, Changfa;  Su, Zhaoming
  |  收藏  |  浏览/下载:11/0  |  提交时间:2025/07/25
P2DFlow: A Protein Ensemble Generative Model with SE(3) Flow Matching 期刊论文  OAI收割
JOURNAL OF CHEMICAL THEORY AND COMPUTATION, 2025, 卷号: 21, 期号: 6, 页码: 3288-3296
作者:  
Jin, Yaowei;  Huang, Qi;  Song, Ziyang;  Zheng, Mingyue;  Teng, Dan
  |  收藏  |  浏览/下载:11/0  |  提交时间:2025/04/24
Discovery of novel covalent stabilizers for p53 Y220C using structure-based drug discovery methods 期刊论文  OAI收割
MOLECULAR DIVERSITY, 2025, 页码: 14
作者:  
Wen, Yiming;  Xu, Peijia;  Chen, Yijie;  Meng, Jingyi;  Zheng, Mingyue
  |  收藏  |  浏览/下载:36/0  |  提交时间:2025/04/01
Harnessing the Magic Methyl Effect: Discovery of CLPP-2068 as a Novel HsClpP Activator for the Treatment of Diffuse Large B-Cell Lymphoma 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 4, 页码: 4287-4307
作者:  
Sun, Mingyang;  Chen, Beijing;  Teng, Dan;  Zhao, Hongshen;  Liao, Yilie
  |  收藏  |  浏览/下载:34/0  |  提交时间:2025/04/01
Design, synthesis, and structure-activity relationship studies of triazolo-pyrimidine derivatives as WRN inhibitors for the treatment of MSI tumors 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 282, 页码: 21
作者:  
Sui, Qibang;  Zhou, Yuanyang;  Li, Manjia;  Wang, Dan;  Cui, Rongrong
  |  收藏  |  浏览/下载:21/0  |  提交时间:2024/12/25
Discovery of CLPP-1071 as an Exceptionally Potent and Orally Efficacious Human ClpP Activator with Strong In Vivo Antitumor Activity 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 21
作者:  
Chen, Beijing;  Sun, Mingyang;  Zhang, Chun;  Huang, Qi
  |  收藏  |  浏览/下载:35/0  |  提交时间:2024/12/25
Targeting STING oligomerization with licochalcone D ameliorates STING-driven inflammatory diseases 期刊论文  OAI收割
SCIENCE CHINA-LIFE SCIENCES, 2024, 页码: 14
作者:  
  |  收藏  |  浏览/下载:35/0  |  提交时间:2024/10/21
Population structure and breed identification of Chinese indigenous sheep breeds using whole genome SNPs and InDels 期刊论文  OAI收割
GENETICS SELECTION EVOLUTION, 2024, 卷号: 56, 期号: 1
作者:  
Zhao, Chang-heng;  Wang, Dan;  Yang, Cheng;  Chen, Yan;  Teng, Jun
  |  收藏  |  浏览/下载:28/0  |  提交时间:2024/11/27
Magnetic and transport properties in antiferromagnetic antiperovskite Eu3SnO 期刊论文  OAI收割
PHYSICAL REVIEW MATERIALS, 2023, 卷号: 7, 期号: 7, 页码: 7
作者:  
Li, Mingze;  Han, Dan;  Wang, Zhenhua;  Li, Bing;  Yang, Teng
  |  收藏  |  浏览/下载:45/0  |  提交时间:2024/01/08