中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共207条,第1-10条 帮助

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Residue-Selective Inhibitors Discovery via Covalent DNA-Encoded Chemical Libraries with Diverse Warheads 期刊论文  OAI收割
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2025, 卷号: 147, 期号: 18, 页码: 15469-15481
作者:  
Wu, Xinyuan;  Pan, Jiayi;  Fan, Rufeng;  Zhang, Yiwei;  Wang, Chao
  |  收藏  |  浏览/下载:3/0  |  提交时间:2025/06/23
Design and synthesis of pyridazin-4-one derivatives as necroptosis inhibitors 期刊论文  OAI收割
ARCHIV DER PHARMAZIE, 2024, 页码: 16
作者:  
An, Yuxiang;  Peng, Xia;  Wang, Tianchen;  Liu, Kaiyuan;  Feng, Dazhi
  |  收藏  |  浏览/下载:16/0  |  提交时间:2024/12/25
Transcriptomic decoding of regional cortical vulnerability to major depressive disorder 期刊论文  OAI收割
COMMUNICATIONS BIOLOGY, 2024, 卷号: 7, 期号: 1, 页码: 12
作者:  
Zhu, Jiajia;  Chen, Xiao;  Lu, Bin;  Li, Xue-Ying;  Wang, Zi-Han
  |  收藏  |  浏览/下载:22/0  |  提交时间:2024/09/10
Remodeling tumor-associated macrophage for anti-cancer effects by rational design of irreversible inhibition of mitogen-activated protein kinase-activated protein kinase 2 期刊论文  OAI收割
MEDCOMM, 2024, 卷号: 5, 期号: 7, 页码: e634
作者:  
Wang, Danyi;  Sun, Deqiao;  Wang, Xiaoyan;  Peng, Xia;  Ji, Yinchun
  |  收藏  |  浏览/下载:1/0  |  提交时间:2025/06/04
Discovery, Optimization, and Evaluation of Novel Pyridin-2(1H)-one Analogues as Potent TRK Inhibitors for Cancer Treatment 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 2, 页码: 1168-1183
作者:  
Xu, Zichao;  Peng, Xia;  Zhang, Renjie;  Ji, Yinchun;  You, Mengke
  |  收藏  |  浏览/下载:34/0  |  提交时间:2024/02/27
Structure-based drug discovery of novel fused- pyrazolone carboxamide derivatives as potent and selective AXL inhibitors 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13, 期号: 12, 页码: 4918-4933
作者:  
Fang, Feifei;  Dai, Yang;  Wang, Hao;  Ji, Yinchun;  Liang, Xuewu
  |  收藏  |  浏览/下载:28/0  |  提交时间:2024/01/26
SYK-mediated epithelial cell state is associated with response to c-Met inhibitors in c-Met-overexpressing lung cancer 期刊论文  OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2023, 卷号: 8, 期号: 1, 页码: 13
作者:  
Zhou, Ji;  Zhang, Xu-Chao;  Xue, Shan;  Dai, Mengdi;  Wang, Yueliang
  |  收藏  |  浏览/下载:29/0  |  提交时间:2023/10/17
Laeviganoids A-T, ent-Clerodane-Type Diterpenoids from Croton laevigatus 期刊论文  OAI收割
JOURNAL OF NATURAL PRODUCTS, 2023, 页码: 15
作者:  
Wang, Cheng-Lei;  Dai, Yang;  Zhu, Qiong;  Peng, Xia;  Liu, Quan-Fang
  |  收藏  |  浏览/下载:17/0  |  提交时间:2023/10/17
Structural Optimization of Fibroblast Growth Factor Receptor Inhibitors for Treating Solid Tumors 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 5, 页码: 3226-3249
作者:  
Li, Chunpu;  Dai, Yang;  Kong, Xiangtai;  Wang, Bao;  Peng, Xia
  |  收藏  |  浏览/下载:19/0  |  提交时间:2024/03/27
Discovery of 3-Aminopyrazole Derivatives as New Potent and Orally Bioavailable AXL Inhibitors 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 22, 页码: 15374-15390
作者:  
Chan, Shingpan;  Zhang, Yunong;  Wang, Jie;  Yu, Qiuchun;  Peng, Xia
  |  收藏  |  浏览/下载:49/0  |  提交时间:2023/04/10