中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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上海药物研究所 [117]
合肥物质科学研究院 [8]
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期刊论文 [144]
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Discovery of a potent and orally bioavailable 3,3-dimethyl-2-oxoindoline STING inhibitor
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2026, 卷号: 301, 页码: 18
作者:
Li, Wenxin
;
Wang, Xiyuan
;
Zang, Shumin
;
Zhou, Rongyao
;
Zhou, Hongfei
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2025/12/04
Discovery of isoindoline-2(1
H
)-carboxamide STING inhibitors as anti-inflammatory agents
期刊论文
OAI收割
MOLECULAR DIVERSITY, 2025, 页码: 13
作者:
Zhou, Xiaoqian
;
Zang, Shumin
;
Yao, Shanyan
;
Zhou, Hongfei
;
Wang, Xiyuan
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2026/01/29
Isoindoline-2(1
H
)-carboxamide
Stimulator of interferon genes
SAR
Inhibitors
Discovery of 3,4-dihydroisoquinoline-2(1H)-carboxamide STING inhibitors as anti-inflammatory agents
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 297, 页码: 20
作者:
Zhou, Xiaoqian
;
Yue, Hangtian
;
Wang, Xiyuan
;
Zang, Shumin
;
Li, Han
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2025/09/09
Stimulator of interferon genes
Inhibitors
Acute kidney injury
3,4-Dihydroisoquinoline-2(1H)-Carboxamide
Predicting the Start of the Growing Season in Boreal Forest Under High and Low Emission Scenarios
期刊论文
OAI收割
EARTHS FUTURE, 2025, 卷号: 13, 期号: 8, 页码: e2024EF005622
作者:
Sun, Zhe
;
Zhao, Jianjun
;
Zhang, Hongyan
;
Wang, Yeqiao
;
Fan, Liangxian
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2025/09/22
Structural Optimization of Next-Generation TRK Inhibitors against Acquired Drug Resistance Mutations for the Treatment of Solid Tumors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 11, 页码: 11484-11501
作者:
Xu, Zichao
;
Liu, Yueling
;
Wang, Peng
;
Peng, Xia
;
Cheng, Jiawei
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2025/08/20
Discovery of Hydrazineyl Amide Derivative of Pseudolaric Acid B for Reprogramming Tumor-Associated Macrophages Against Tumor Growth
期刊论文
OAI收割
MOLECULES, 2025, 卷号: 30, 期号: 10, 页码: 22
作者:
Peng, Xia
;
Yu, Siqi
;
Xu, Lin
;
Wang, Qinghua
;
Yang, Lin
  |  
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2025/07/25
pseudolaric acid B
amide derivatives
tumor-associated macrophages
anti-tumor
repolarization
Discovery of Potent STING Inhibitors Bearing a Difluorobenzodioxol Structural Motif as Potent Anti-Inflammatory Agents
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 8, 页码: 8907-8932
作者:
Shen, Ancheng
;
Wang, Xiyuan
;
Chen, Qingxuan
;
Zhang, Yan
;
Wang, Fang
  |  
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2025/05/27
Discovery of a non-nucleotide stimulator of interferon genes (STING) agonist with systemic antitumor effect
期刊论文
OAI收割
MEDCOMM, 2025, 卷号: 6, 期号: 1, 页码: e70001
作者:
Wang, Xiyuan
;
Zhan, Zhengsheng
;
Wang, Zhen
;
Zhang, Yan
;
Zhao, Kaiyan
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2025/06/04
antitumor
immune memory
innate immunity
STING agonist
Metal-organic framework-based SERS chips enable
in situ
and sensitive detection of dissolved hydrogen sulfide in natural water: Towards a bring-back-chip mode for field analysis
期刊论文
OAI收割
JOURNAL OF HAZARDOUS MATERIALS, 2024, 卷号: 480, 页码: 10
作者:
Si, Meiyu
;
Wang, Yunqing
;
Mei, Rongchao
;
Zhao, Xizhen
;
Yuan, Qi
  |  
收藏
  |  
浏览/下载:55/0
  |  
提交时间:2024/12/06
Hydrogen sulfide
Surface enhanced Raman scattering
Metal-organic framework
in situ sampling
Environmental analysis
Design and synthesis of pyridazin-4-one derivatives as necroptosis inhibitors
期刊论文
OAI收割
ARCHIV DER PHARMAZIE, 2024, 页码: 16
作者:
An, Yuxiang
;
Peng, Xia
;
Wang, Tianchen
;
Liu, Kaiyuan
;
Feng, Dazhi
  |  
收藏
  |  
浏览/下载:53/0
  |  
提交时间:2024/12/25
inhibitor
pharmacokinetic study
pyridazin-4-one
receptor-interacting protein kinase 1
selectivity