中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [19]
采集方式
OAI收割 [19]
内容类型
期刊论文 [19]
发表日期
2025 [7]
2024 [5]
2023 [2]
2020 [1]
2019 [1]
2018 [1]
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The enedioic acid analog 326E alleviates metabolic dysfunction-associated steatohepatitis via dual targeting at ACLY and PPARα
期刊论文
OAI收割
CELL METABOLISM, 2025, 卷号: 37, 期号: 11, 页码: 2149-2166
作者:
Xie, Zhifu
;
Cheng, Long
;
Hu, Yue
;
Song, Gaolei
;
Wang, Fan
  |  
收藏
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Discovery of Novel Tridentate Alkenyl Diacid Derivatives as Potent ATP Citrate Lyase Inhibitors for the Treatment of Hepatocellular Carcinoma
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 15, 页码: 15598-15616
作者:
Yang, Yurou
  |  
收藏
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Dietary timing enhances exercise by modulating fat-muscle crosstalk via adipocyte AMPKa2 signaling
期刊论文
OAI收割
CELL METABOLISM, 2025, 卷号: 37, 期号: 6, 页码: 24
作者:
Chen, Jianghui
;
Xiang, Jing
;
Zhou, Meiyu
;
Huang, Rongfeng
;
Zhang, Jianxin
  |  
收藏
  |  
Novel Aryl Sulfonium Modification on Vancomycin to Tackle MRSA and VRE In Vitro and In Vivo through Dual Enhanced Cell-Wall and Membrane Inhibition
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 8, 页码: 8310-8329
作者:
Xie, Yuanyuan
;
Wang, Xiaowen
;
Chang, Taopeng
;
Chen, Zhifu
;
Luo, Youhong
  |  
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A Rationally Designed Sulfonium Lipoglycopeptide with Micelles Self-Assembly to Combat Multidrug Resistance via Dual Enhanced Cell Wall-Membrane Inhibition and T7SS Proteins Downregulation
期刊论文
OAI收割
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2025, 卷号: 147, 期号: 15, 页码: 12587-12603
作者:
Xie, Yuanyuan
;
Wang, Xiaowen
;
Li, Fang
;
Chen, Zhifu
;
Li, Qun
  |  
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  |  
A natural small molecule isoginkgetin alleviates hypercholesterolemia and atherosclerosis by targeting ACLY
期刊论文
OAI收割
THERANOSTICS, 2025, 卷号: 15, 期号: 10, 页码: 4325-4344
作者:
Zhang, Zhidan
;
Chen, Meijie
;
Xu, Yitong
;
Wang, Zhihua
;
Liu, Zhenghong
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  |  
A Phase I Study to Evaluate the Safety, Tolerability, Pharmacokinetics of BGT-002, a Novel ATP-Citrate Lyase Inhibitor, in Healthy Chinese Subjects
期刊论文
OAI收割
DRUG DESIGN DEVELOPMENT AND THERAPY, 2025, 卷号: 19, 页码: 1783-1794
作者:
Liu, Yun
;
Yu, Chengyin
;
Zhang, Yifan
;
Xie, Zhifu
;
Wang, Yating
  |  
收藏
  |  
Single Amine or Guanidine Modification on Norvancomycin and Vancomycin to Overcome Multidrug-Resistance through Augmented Lipid II Binding and Increased Membrane Activity
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 22, 页码: 20639-20663
作者:
Bian, Xiaolei
;
Chen, Zhifu
;
Li, Fang
;
Xie, Yuanyuan
;
Li, Yi
  |  
收藏
  |  
Discovery of Alkyl Conjugated Diene Diacids as Novel ACLY Inhibitors
期刊论文
OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2024, 卷号: 44, 期号: 11, 页码: 3476-3489
作者:
Cheng, Tingting
;
Song, Gaolei
;
Cheng, Long
;
Wang, Fan
;
Sun, Xinyu
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Potential therapeutic strategies for MASH: from preclinical to clinical development
期刊论文
OAI收割
LIFE METABOLISM, 2024, 卷号: 3, 期号: 5, 页码: loae029
作者:
Xie, Zhifu
;
Li, Yufeng
;
Cheng, Long
;
Huang, Yidan
;
Rao, Wanglin
  |  
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