中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共2417条,第1-10条 帮助

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Conformational restriction enables discovering a series of chroman derivatives as potent and selective NaV1.8 inhibitors with improved pharmacokinetic properties 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 293, 页码: 24
作者:  
Li, Na;  Wang, Linlin;  Hu, Xinyuan;  Xu, Haiyan;  Yang, Bowen
  |  收藏  |  浏览/下载:1/0  |  提交时间:2025/08/20
Immunosuppressive nitrogen-containing triterpenoid saponins from Mussaenda erosa and the therapeutic efficacy of heinsiagenin A in a murine lupus erythematosus model 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2025, 卷号: 163, 页码: 11
作者:  
Xu, Yidan;  Xiang, Mai;  Chang, Yuan;  Chen, Zhenhua;  Zhang, Rujun
  |  收藏  |  浏览/下载:1/0  |  提交时间:2025/08/20
EP240801a/XRF 240801B: An X-Ray Flash Detected by the Einstein Probe and the Implications of Its Multiband Afterglow 期刊论文  OAI收割
ASTROPHYSICAL JOURNAL LETTERS, 2025, 卷号: 988, 期号: 1
作者:  
Jiang, Shuai-Qing;  Xu, Dong;  Hoof, Agnes P. C. van;  Lei, Wei-Hua;  Liu, Yuan
  |  收藏  |  浏览/下载:21/0  |  提交时间:2025/07/28
Study of ultra-high-energy gamma-ray source 1LHAASO J0056+6346u and its possible origins 期刊论文  OAI收割
SCIENCE CHINA-PHYSICS MECHANICS & ASTRONOMY, 2025, 卷号: 68, 期号: 7
作者:  
Cao, Zhen;  Aharonian, F.;  Axikegu;  Bai, Y. X.;  Bao, Y. W.
  |  收藏  |  浏览/下载:33/0  |  提交时间:2025/06/10
Green synthesis of 2-trifluoromethylquinoline skeletons via organocatalytic N-[(α-trifluoromethyl)vinyl]isatins CN bond activation 期刊论文  OAI收割
CHINESE CHEMICAL LETTERS, 2025, 卷号: 36, 期号: 7, 页码: 10
作者:  
Ji, Cong-Bin;  Xie, Ding-Xiong;  Chen, Mei;  Lan, Ye-Ying;  Zhang, Bao-Hua
  |  收藏  |  浏览/下载:17/0  |  提交时间:2025/07/25
NMRExtractor: leveraging large language models to construct an experimental NMR database from open-source scientific publications 期刊论文  OAI收割
CHEMICAL SCIENCE, 2025, 卷号: 16, 期号: 25, 页码: 11548-11558
作者:  
Wang, Qinggong;  Zhang, Wei;  Chen, Mingan;  Li, Xutong;  Xiong, Zhaoping
  |  收藏  |  浏览/下载:1/0  |  提交时间:2025/08/20
Rapid Discovery of Celastrol Derivatives as Potent and Selective PRDX1 Inhibitors via Microplate-Based Parallel Compound Library and In Situ Screening 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 13, 页码: 13609-13627
作者:  
Chen, Shuang;  Wang, Zhenyu;  Gao, Jia;  Wang, Yanlin;  Liang, Jiayin
  |  收藏  |  浏览/下载:5/0  |  提交时间:2025/08/20
Contrastive learning-based drug screening model for GluN1/GluN3A inhibitors 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2025, 页码: 13
作者:  
Li, Kun;  Zeng, Yue;  Xiong, Yi-da;  Wu, Hao-chen;  Fang, Sui
  |  收藏  |  浏览/下载:3/0  |  提交时间:2025/08/20
De novo design of protein condensation inhibitors by targeting an allosteric site of cGAS 期刊论文  OAI收割
NATURE COMMUNICATIONS, 2025, 卷号: 16, 期号: 1, 页码: 20
作者:  
Zhao, Wenfeng;  Chen, Guofeng;  He, Jian;  Shen, Xiaofang;  Xiong, Muya
  |  收藏  |  浏览/下载:5/0  |  提交时间:2025/08/20
Microstructure, seepage regimes and stress-strain analysis of bedded rock salt interface 期刊论文  OAI收割
JOURNAL OF ENERGY STORAGE, 2025, 卷号: 120, 页码: 13
作者:  
Chen, Xiangsheng;  Li, Yinping;  Shi, Xilin
  |  收藏  |  浏览/下载:11/0  |  提交时间:2025/06/27