中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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上海药物研究所 [219]
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期刊论文 [1239]
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Tumor-targeted PROTAC prodrug nanoplatform enables precise protein degradation and combination cancer therapy
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2024, 页码: 12
作者:
Zou, Zhi-feng
;
Yang, Lei
;
Nie, Hui-jun
;
Gao, Jing
;
Lei, Shu-min
  |  
收藏
  |  
浏览/下载:0/0
  |  
提交时间:2024/05/22
proteolysis-targeting chimeras
tumor-targeted delivery
precise protein degradation
combination therapy
triple-negative breast cancer
Excessive fatty acids activate PRMT5/MDM2/Drosha pathway to regulate miRNA biogenesis and lipid metabolism
期刊论文
OAI收割
LIVER INTERNATIONAL, 2024, 页码: 17
作者:
Hou, Aijun
;
Xu, Xiaoding
;
Zhang, Yu
;
He, Hongxiu
;
Feng, Yihan
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2024/05/07
Drosha degradation
lipid metabolism
miRNA biogenesis
NAFLD
PRMT5
Discovery of a Covalent Inhibitor Selectively Targeting the Autophosphorylation Site of c-Src Kinase
期刊论文
OAI收割
ACS CHEMICAL BIOLOGY, 2024, 页码: 12
作者:
Zhang, Huimin
;
Xu, Dounan
;
Huang, Hongchan
;
Jiang, Hao
;
Hu, Linghao
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2024/05/07
Ent-labdane-type diterpene glycosides obtained from
Rubus
chingii
Hu and their inhibitory effects on PDE5A activity
期刊论文
OAI收割
FITOTERAPIA, 2024, 卷号: 173, 页码: 14
作者:
Yu, Jun-dong
;
Wang, Jing-Yi
;
Liu, Jia-yuan
;
Xu, Ye-chun
;
Zhang, Xue
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2024/02/27
diterpene glycosides
Rubus Chingii Hu
PDE5A inhibitory activity
ent-labdane
Country-specific net-zero strategies of the pulp and paper industry
期刊论文
OAI收割
NATURE, 2024, 卷号: 626, 期号: 7998, 页码: 24
作者:
Dai, Min
;
Sun, Mingxing
;
Chen, Bin
;
Shi, Lei
;
Jin, Mingzhou
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2024/04/01
Characteristics of Paleontological Communities in Surface Sediments of the Southern South China Sea and Their Paleoclimatic and Paleoenvironmental Significance
期刊论文
OAI收割
JOURNAL OF EARTH SCIENCE, 2024, 卷号: 35, 期号: 1, 页码: 144-154
作者:
Zhao, Jing
;
Zhang, Li
;
Wang, Xiaoyan
;
Ge, Jinglian
;
Xu, Min
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2024/05/15
southern South China Sea
sediments
foraminifera
diatom
pollen
The carbon budget of China: 1980-2021
期刊论文
OAI收割
SCIENCE BULLETIN, 2024, 卷号: 69, 期号: 1, 页码: 114-124
作者:
Xia, Xiaosheng
;
Ren, Peiyang
;
Wang, Xuhui
;
Liu, Dan
;
Chen, Xiuzhi
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2024/04/01
CO2 emission
Land carbon sink
China
Carbon neutrality
Carbon budget
Reorganization of intrinsic functional connectivity in early-stage Parkinson's disease patients with probable REM sleep behavior disorder
期刊论文
OAI收割
NPJ PARKINSONS DISEASE, 2024, 卷号: 10, 期号: 1, 页码: 11
作者:
Dan, Xiao-Juan
;
Wang, Yu-Wei
;
Sun, Jun-Yan
;
Gao, Lin-Lin
;
Chen, Xiao
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/01/31
Discovery of hematopoietic progenitor kinase 1 inhibitors using machine learning-based screening and free energy perturbation
期刊论文
OAI收割
JOURNAL OF BIOMOLECULAR STRUCTURE & DYNAMICS, 2024, 页码: 13
作者:
Feng, Dazhi
;
Liu, Bo
;
Chen, Zhiwei
;
Xu, Jinyi
;
Geng, Meiyu
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2024/02/27
HPK1 inhibitor
machine learning
virtual screening
free energy perturbation
structural modification
Heat sensitive E-helix cut ferritin nanocages for facile and high-efficiency loading of doxorubicin
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2023, 卷号: 253
作者:
Xia, Haining
;
Xu, Huangtao
;
Wang, Jiarong
;
Wang, Changhao
;
Chen, Ruiguo
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2023/11/17
Ferritin nanocages
Drug loading
Structural modification
Thermal response
Ion-assisted