机构

• 上海药物研究所 [9]
• 合肥物质科学研究院 [7]
• 金属研究所 [5]
• 力学研究所 [1]
• 物理研究所 [1]
• 武汉物理与数学研究所 [1]
• 更多

采集方式

• OAI收割 [25]
• iSwitch采集 [1]

内容类型

• 期刊论文 [26]

发表日期

• 2025 [2]
• 2024 [5]
• 2023 [1]
• 2022 [2]
• 2021 [4]
• 2020 [2]
• 更多

学科主题

筛选

浏览/检索结果: 共26条，第1-10条 帮助 条数/页： 5101520253035404550556065707580859095100 排序方式： 请选择题名升序题名降序提交时间升序提交时间降序作者升序作者降序发表日期升序发表日期降序 Development of novel epoxyketone macrocyclic peptidyl proteasome inhibitors through OPA-mediated one-step cyclization of unprotected peptides 期刊论文  OAI收割 BIOORGANIC CHEMISTRY, 2025, 卷号: 156, 页码: 16 作者:  Zeng, Gongruixue;  Xu, Gaoya;  Gao, Lixin;  Zheng, Xiaoli;  Chi, Xinglong   |  收藏  |  浏览/下载：9/0  |  提交时间：2025/04/01 Proteasome inhibitors  Macrocycle  Stability  Anti-cancer activities   Auto-RapTAC: A Versatile and Sustainable Platform for the Automated Rapid Synthesis and Evaluation of PROTAC 期刊论文  OAI收割 JOURNAL OF MEDICINAL CHEMISTRY, 2025, 页码: 15 作者:  Chen, Jiexuan;  Wu, Mingfei;  Mo, Jun;  Hong, Ju;  Wang, Wei   |  收藏  |  浏览/下载：13/0  |  提交时间：2025/04/01 Exploration of novel 20S proteasome activators featuring anthraquinone structures and their application in hypoxic cardiomyocyte protection 期刊论文  OAI收割 BIOORGANIC & MEDICINAL CHEMISTRY, 2024, 卷号: 115, 页码: 10 作者:  Yu, Qian;  Gao, Lixin;  Xu, Linhao;  Han, Yubing;  Cao, Yu   |  收藏  |  浏览/下载：11/0  |  提交时间：2024/12/11 Single-cell sequencing reveals the heterogeneity of pancreatic neuroendocrine tumors under genomic instability and histological grading 期刊论文  OAI收割 ISCIENCE, 2024, 卷号: 27, 期号: 9, 页码: 18 作者:  Ye, Zeng;  Zhou, Yan;  Hu, Yuheng;  Li, Qiang;  Xu, Zijin   |  收藏  |  浏览/下载：11/0  |  提交时间：2024/11/05 tumor cells  CNV neutral tumor cells  neuroendocrine cells  profile   Discovery of a Highly Potent and Selective BRD9 PROTAC Degrader Based on E3 Binder Investigation for the Treatment of Hematological Tumors 期刊论文  OAI收割 JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 28 作者:  Duan, Haiting;  Zhang, Jingyu;  Gui, Renzhao;  Lu, Yang;  Pang, Ao   |  收藏  |  浏览/下载：7/0  |  提交时间：2024/08/20 Discovery of potent small molecule ubiquitin-specific protease 10 inhibitors with anti-hepatocellular carcinoma activity through regulating YAP expression 期刊论文  OAI收割 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 272, 页码: 21 作者:  Lu, Yang;  Gao, Jian;  Wang, Peipei;  Chen, Haifeng;  He, Xinjun   |  收藏  |  浏览/下载：6/0  |  提交时间：2024/07/12 Hepatocellular carcinoma  Ubiquitin-specific protease 10  Deubiquitination  Selectivity   Extinction of microgravity partially premixed flame aboard the Chinese Space Station 期刊论文  OAI收割 PROCEEDINGS OF THE COMBUSTION INSTITUTE, 2024, 卷号: 40, 期号: 1-4, 页码: 7 作者:  Wen, Yuzhe;  Li, Longfei;  Li, Xingxian;  Luo, Lei;  Chen, Tao   |  收藏  |  浏览/下载：5/0  |  提交时间：2024/08/23 Partially premixed flame  Non-premixed flame  Radiation  Microgravity  Extinction   Structure-based identification of new orally bioavailable BRD9-PROTACs for treating acute myelocytic leukemia 期刊论文  OAI收割 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 262, 页码: 18 作者:  Zhang, Jingyu;  Duan, Haiting;  Gui, Renzhao;  Wu, Mingfei;  Shen, Liteng   |  收藏  |  浏览/下载：132/0  |  提交时间：2023/12/19 Acute myeloid leukemia  Bromodomain-containing protein 9  Proteolysis-targeting chimera  Orally bioavailable  Docking   Design, synthesis and biological evaluation of sulfonamides inhibitors of XPO1 displaying activity against multiple myeloma cells 期刊论文  OAI收割 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 235 作者:  Qu, Bingxue;  Xu, Yongjin;  Lu, Yang;  Zhuang, Weihao;  Jin, Xinxin   |  收藏  |  浏览/下载：43/0  |  提交时间：2022/12/23 XPO1  Multiple myeloma  MM.1S  N-phenylsulfonamide  Oral administration   High efficacy of PD-1 inhibitor after initial failure of PD-L1 inhibitor in Relapsed/Refractory classical Hodgkin Lymphoma 期刊论文  OAI收割 BMC CANCER, 2022, 卷号: 22 作者:  Chen, Xi;  Kong, Haiying;  Luo, Linxiang;  Han, Shuiyun;  Lei, Tao   |  收藏  |  浏览/下载：65/0  |  提交时间：2022/02/14 Hodgkin lymphoma  PD-1 inhibitor  PD-L1 inhibitor  PD-L2  Molecular phenotype  Tumor microenvironment