中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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高能物理研究所 [145]
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Design, synthesis, and evaluation of Menin-targeting compounds for the treatment of acute Myelocytic leukemia (AML)
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 296, 页码: 17
作者:
Mo, Jun
;
Wang, Yuxian
;
Pan, Youlu
;
Xiao, Qitao
;
Zhao, Jinyi
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2025/08/20
Menin
High binding affinity
Anti-proliferation activity
AML
The Overview and Trial Observations of AIMS
期刊论文
OAI收割
RESEARCH IN ASTRONOMY AND ASTROPHYSICS, 2025, 卷号: 25, 期号: 7
作者:
Deng, Yuanyong
;
Wang, Dongguang
;
Hua, Jianwen
;
Xu, Songbo
;
Liang, Ming
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2025/07/14
Sun: infrared
methods: observational
instrumentation: spectrographs
Ordovician-Devonian granites and Li-Be-bearing pegmatites in the Altyn Tagh Orogen, NW China
期刊论文
OAI收割
GEOLOGICAL SOCIETY OF AMERICA BULLETIN, 2025, 页码: 21
作者:
Jing, Yan
;
Zhang, Chuan-lin
;
Wang, Chen
;
Ge, Wen-chun
;
Song, Zhi-hao
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2025/07/11
Organic amendments promote soil phosphorus related functional genes and microbial phosphorus cycling
期刊论文
OAI收割
GEODERMA, 2025, 卷号: 456, 页码: 117247
作者:
Wu, Wenchao
;
Zhang, Yangjian
;
Turner, Benjamin L.
;
He, Yunlong
;
Chen, Xiaodong
  |  
收藏
  |  
浏览/下载:40/0
  |  
提交时间:2025/04/21
Fertilization regimes
Soil microbes
Soil phosphatase
Functional genes
Phosphorus cycling
Global synthesis
Development of novel epoxyketone macrocyclic peptidyl proteasome inhibitors through OPA-mediated one-step cyclization of unprotected peptides
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2025, 卷号: 156, 页码: 16
作者:
Zeng, Gongruixue
;
Xu, Gaoya
;
Gao, Lixin
;
Zheng, Xiaoli
;
Chi, Xinglong
  |  
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2025/04/01
Proteasome inhibitors
Macrocycle
Stability
Anti-cancer activities
Discovery of a potential hematologic malignancies therapy: Selective and potent HDAC7 PROTAC degrader targeting non-enzymatic function
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2025, 卷号: 15, 期号: 3, 页码: 1659-1679
作者:
Jin, Yuheng
;
Qi, Xuxin
;
Yu, Xiaoli
;
Cheng, Xirui
;
Chen, Boya
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2025/06/23
HDAC7
PROTAC
Selectivity
Hematologic malignancies
Non-enzymatic function
Rubiadin Mediates the Upregulation of Hepatic Hepcidin and Alleviates Iron Overload via BMP6/SMAD1/5/9-Signaling Pathway
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2025, 卷号: 26, 期号: 3, 页码: 14
作者:
Xie, Xueting
;
Chang, Linyue
;
Zhu, Xinyue
;
Gong, Fengbei
;
Che, Linlin
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2025/04/01
rubiadin
hepcidin
iron metabolism
iron overload
BMP6/SMAD1/5/9-signaling pathway
Auto-RapTAC: A Versatile and Sustainable Platform for the Automated Rapid Synthesis and Evaluation of PROTAC
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 页码: 15
作者:
Chen, Jiexuan
;
Wu, Mingfei
;
Mo, Jun
;
Hong, Ju
;
Wang, Wei
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2025/04/01
Discovery of N-Benzylpiperidinol derivatives as USP7 inhibitors against Hematology
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2024, 卷号: 153, 页码: 13
作者:
Pan, Youlu
;
Chen, Haifeng
;
Fu, Jingfeng
;
Zhang, Jingyu
;
Wang, Peipei
  |  
收藏
  |  
浏览/下载:40/0
  |  
提交时间:2024/10/21
Environmental changes and human impacts over the past 1200 years: Evidence from high-resolution pollen records from peat in the Yunnan-Guizhou Plateau, Southwest China
期刊论文
OAI收割
PALAEOGEOGRAPHY PALAEOCLIMATOLOGY PALAEOECOLOGY, 2024, 卷号: 655, 页码: 14
作者:
Li, Shuming
;
Wei, Lisi
;
Zhao, Wenwei
;
Ren, Weihe
;
Gu, Qinran
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2024/12/30
Pollen
Human impact
Vegetation dynamics
Climate change
Southwest China
Southwest China