中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [6]
化学研究所 [5]
自动化研究所 [4]
过程工程研究所 [3]
生态环境研究中心 [1]
烟台海岸带研究所 [1]
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OAI收割 [20]
内容类型
期刊论文 [19]
会议论文 [1]
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2023 [4]
2022 [3]
2021 [5]
2020 [1]
2019 [2]
2018 [1]
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学科主题
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Design, synthesis and biological evaluation of chalcone derivatives as potent and orally active hCYP3A4 inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2023, 卷号: 95, 页码: 9
作者:
Lu, Shiwei
;
Zhang, Feng
;
Gong, Jiahao
;
Huang, Jian
;
Zhu, Guanghao
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2023/12/08
Cytochrome P450 3A4 (CYP3A4)
Inhibitors
Isoquinoline chalcones
Orally active
Discovery of seven-membered ring berberine analogues as highly potent and specific hCES2A inhibitors
期刊论文
OAI收割
CHEMICO-BIOLOGICAL INTERACTIONS, 2023, 卷号: 378, 页码: 11
作者:
Yang, Yun
;
Xiong, Yuan
;
Zhu, Guanghao
;
Sun, Mengru
;
Zou, Kun
  |  
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2023/10/17
Human carboxylesterase 2 (hCES2A)
Berberine analogues
Structure -activity relationships (SAR)
Inhibition kinetics
Selectivity
Aero-Engine Remaining Useful Life Estimation Based on CAE-TCN Neural Networks
期刊论文
OAI收割
APPLIED SCIENCES-BASEL, 2023, 卷号: 13, 期号: 1, 页码: 15
作者:
Ren, Guanghao
;
Wang, Yun
;
Shi, Zhenyun
;
Zhang, Guigang
;
Jin, Feng
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2023/02/22
remaining useful life estimation
aero-engine
convolutional autoencoder
temporal convolutional network
Discovery and mechanism of action of Thonzonium bromide from an FDA-approved drug library with potent and broad-spectrum inhibitory activity against main proteases of human coronaviruses
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2023, 卷号: 130, 页码: 11
作者:
Wang, Ruyu
;
Zhai, Guanglei
;
Zhu, Guanghao
;
Wang, Mengge
;
Gong, Xiaoyi
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2023/04/10
SARS-CoV-23CLpro
Thonzonium bromide
Mechanism of action
Broad-spectrum inhibitor
Chemo- and Site-Selective Lysine Modification of Peptides and Proteins under Native Conditions Using the Water-Soluble Zolinium
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 14
作者:
Sun, Haiguo
;
Xi, Mengyu
;
Jin, Qiang
;
Zhu, Zhengdan
;
Zhang, Yani
  |  
收藏
  |  
浏览/下载:44/0
  |  
提交时间:2022/09/30
Discovery of a Potent and Selective Degrader for USP7
期刊论文
OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2022, 卷号: 61, 期号: 33, 页码: e202204395
作者:
Pei, Yuan
;
Fu, Jingfeng
;
Shi, Yunkai
;
Zhang, Mengmeng
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2024/03/21
Apoptotic Pathway
Mutant p53
p53 Mutant Cancer Cells
PROTAC
USP7 Degrader
Two‑stage hybrid network for segmentation of COVID‑19 pneumonia lesions in CT images: a multicenter study
期刊论文
OAI收割
Medical & Biological Engineering & Computing, 2022, 页码: 2721-2736
作者:
Yaxin Shang
;
Zechen Wei
;
Hui Hui
;
Xiaohu Li
;
Liang Li
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/06/28
Image-to-Images Translation for Multiple Virtual Histological Staining of Unlabeled Human Carotid Atherosclerotic Tissue
期刊论文
OAI收割
MOLECULAR IMAGING AND BIOLOGY, 2021, 页码: 11
作者:
Zhang, Guanghao
;
Ning, Bin
;
Hui, Hui
;
Yu, Tengfei
;
Yang, Xin
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2021/12/28
Multiple virtual histological staining
Pix2pix network
Human carotid atheroma
Blind evaluation
Bright-field microscopic imaging
Fast Fault Diagnosis System Based on Data Mining AR Algorithm
会议论文
OAI收割
Nanjing, China, 2021-10
作者:
Yu Yahan
;
Du Juan
;
Ren Guanghao
;
Tan Yao
;
Wang Jian
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2023/06/02
The loss of RNA N-6-adenosine methyltransferase Mettl14 in tumor-associated macrophages promotes CD8(+) T cell dysfunction and tumor growth
期刊论文
OAI收割
CANCER CELL, 2021, 卷号: 39, 期号: 7, 页码: 945-+
作者:
Dong, Lihui
;
Chen, Chuanyuan
;
Zhang, Yawei
;
Guo, Peijin
;
Wang, Zhenghang
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2021/12/22