中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
首页
机构
成果
学者
登录
注册
登陆
×
验证码:
换一张
忘记密码?
记住我
×
校外用户登录
CAS IR Grid
机构
上海药物研究所 [138]
金属研究所 [28]
广州能源研究所 [16]
西北高原生物研究所 [9]
国家授时中心 [6]
烟台海岸带研究所 [5]
更多
采集方式
OAI收割 [242]
iSwitch采集 [3]
内容类型
期刊论文 [241]
会议论文 [3]
CNKI期刊论文 [1]
发表日期
2025 [14]
2024 [37]
2023 [27]
2022 [28]
2021 [25]
2020 [20]
更多
学科主题
Biochemist... [2]
Biology [1]
Biophysics [1]
Chemistry,... [1]
Chemistry,... [1]
Chemistry,... [1]
更多
筛选
浏览/检索结果:
共245条,第1-10条
帮助
条数/页:
5
10
15
20
25
30
35
40
45
50
55
60
65
70
75
80
85
90
95
100
排序方式:
请选择
题名升序
题名降序
提交时间升序
提交时间降序
作者升序
作者降序
发表日期升序
发表日期降序
Discovery and Identification of a Novel PORCN Inhibitor via Structure-Based Virtual Screening
期刊论文
OAI收割
ACS CHEMICAL BIOLOGY, 2025, 卷号: 20, 期号: 6, 页码: 1319-1332
作者:
Yang, Xinyu
;
Li, Yanbei
;
Zhou, Jingyi
;
Zhou, Yuanyang
;
Lin, Kexin
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2025/07/25
Palladium-Catalyzed Enantioselective Arylative Dearomatization of Naphthols and Phenols for Constructing Quinazoline-Containing Spirocycles
期刊论文
OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2025, 页码: 9
作者:
Zhang, Chiyue
;
Xu, Gaoya
;
Zhao, Wenlu
;
Li, Xutong
;
Zheng, Mingyue
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2025/07/25
Antiproliferative activity
Catalytic asymmetric dearomatization
Palladium
Quinazoline-containing spirocycles
Three-dimensionality
Discovery of 3-(Fluoro-imidazolyl)pyridazine Derivatives as Potent STING Agonists with Antitumor Activity
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 10, 页码: 9864-9885
作者:
Hou, Hui
;
Zhou, Jingyi
;
Sui, Qibang
;
Zhang, Changfa
;
Su, Zhaoming
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2025/07/25
Microbiota-shaped neutrophil senescence regulates sexual dimorphism in bladder cancer
期刊论文
OAI收割
NATURE IMMUNOLOGY, 2025, 卷号: 26, 期号: 5, 页码: 46
作者:
Zhu, Qingchen
;
Zhang, Guiheng
;
Cao, Ming
;
Huang, Huan
;
He, Dan
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2025/06/23
Bridging chemistry and artificial intelligence by a reaction description language
期刊论文
OAI收割
NATURE MACHINE INTELLIGENCE, 2025, 卷号: 7, 期号: 5, 页码: 16
作者:
Xiong, Jiacheng
;
Zhang, Wei
;
Wang, Yinquan
;
Huang, Jiatao
;
Shi, Yuqi
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2025/07/25
Residue-Selective Inhibitors Discovery via Covalent DNA-Encoded Chemical Libraries with Diverse Warheads
期刊论文
OAI收割
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2025, 卷号: 147, 期号: 18, 页码: 15469-15481
作者:
Wu, Xinyuan
;
Pan, Jiayi
;
Fan, Rufeng
;
Zhang, Yiwei
;
Wang, Chao
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2025/06/23
Proteome-Wide Data Guides the Discovery of Lysine-Targeting Covalent Inhibitors Using DNA-Encoded Chemical Libraries
期刊论文
OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2025, 页码: 14
作者:
Wu, Xinyuan
;
Li, Shunyao
;
Liang, Ting
;
Yu, Qing
;
Zhang, Yiwei
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2025/06/23
Activity-based protein profiling data
Covalent DNA-encoded chemical library
Covalent ligand selection
Lysine-targeting covalent inhibitors
Recent advances in targeted degradation in the RAS pathway
期刊论文
OAI收割
FUTURE MEDICINAL CHEMISTRY, 2025, 卷号: 17, 期号: 6, 页码: 693-708
作者:
Ge, Zhiming
;
Fan, Zisheng
;
He, Wei
;
Zhou, Guizhen
;
Zhou, Yidi
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2025/04/24
RAS
cancer
mutation
degrader
PROTAC
Targeting the histone reader ZMYND8 inhibits antiandrogen-induced neuroendocrine tumor transdifferentiation of prostate cancer
期刊论文
OAI收割
NATURE CANCER, 2025, 页码: 37
作者:
Wang, Hanling
;
Zhang, Sulin
;
Pan, Qiang
;
Guo, Jiacheng
;
Li, Ni
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2025/05/27
Discovery of novel covalent stabilizers for p53 Y220C using structure-based drug discovery methods
期刊论文
OAI收割
MOLECULAR DIVERSITY, 2025, 页码: 14
作者:
Wen, Yiming
;
Xu, Peijia
;
Chen, Yijie
;
Meng, Jingyi
;
Zheng, Mingyue
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2025/04/01
p53 Y220C
Covalent stabilizer
Virtual screening
Molecular dynamics
DNA binding
Structure-activity relationship
Cancer therapy