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Construction of PROTAC Library via Liquid-Phase Synthesis Enabled by a Hydrophobic Tag
期刊论文
OAI收割
ORGANIC LETTERS, 2026, 卷号: 28, 期号: 8, 页码: 2747-2752
作者:
Zhou, Yifeng
;
He, Wei
;
Zhou, Zehui
;
Wu, Min
;
Wu, Qianping
  |  
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Discovery of novel selective PRMT5-MTA inhibitors through structure-based virtual screening
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2026, 卷号: 168, 页码: 17
作者:
Ma, Ning
;
Chen, Yang
;
Liang, Yiru
;
Chen, Xiaoxu
;
Song, Fengnan
  |  
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  |  
Furo[2,3-
f
]quinazolin-7(6
H
)-one Derivatives as Potent, Selective, and Orally Bioavailable MAT2A Inhibitors for MTAP-Deficient Cancer Therapy
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 22, 页码: 24213-24231
作者:
Shi, Zihan
;
Lin, Kexin
;
Lin, Lijie
;
Chen, Zhiyi
;
Xie, Zhiyin
  |  
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  |  
A pan-KRAS inhibitor and its derived degrader elicit multifaceted anti-tumor efficacy in
KRAS
-driven cancers
期刊论文
OAI收割
CANCER CELL, 2025, 卷号: 43, 期号: 10, 页码: 32
作者:
Feng, Juanjuan
;
Xiao, Xuanzheng
;
Xia, Xinting
;
Min, Jian
;
Tang, Weiying
  |  
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  |  
Methotrexate exerts antitumor immune activity and improves the clinical efficacy of immunotherapy in patients with solid tumors
期刊论文
OAI收割
SCIENCE TRANSLATIONAL MEDICINE, 2025, 卷号: 17, 期号: 801, 页码: 18
作者:
Yang, Ruirui
;
Wang, Bei
;
Su, Zhaoming
;
Song, Ying
;
Zhang, Yingying
  |  
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  |  
Design, synthesis, and activity evaluation of indole derivatives as potential stabilizers for p53 Y220C
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2025, 卷号: 121, 页码: 9
作者:
Li, Linquan
;
Gu, Xi
;
Meng, Jingyi
;
Wen, Yiming
;
Yi, Jing
  |  
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  |  
Discovery and Identification of a Novel PORCN Inhibitor via Structure-Based Virtual Screening
期刊论文
OAI收割
ACS CHEMICAL BIOLOGY, 2025, 卷号: 20, 期号: 6, 页码: 1319-1332
作者:
Yang, Xinyu
;
Li, Yanbei
;
Zhou, Jingyi
;
Zhou, Yuanyang
;
Lin, Kexin
  |  
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  |  
Discovery of 3-(Fluoro-imidazolyl)pyridazine Derivatives as Potent STING Agonists with Antitumor Activity
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 10, 页码: 9864-9885
作者:
Hou, Hui
;
Zhou, Jingyi
;
Sui, Qibang
;
Zhang, Changfa
;
Su, Zhaoming
  |  
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  |  
Recent advances in targeted degradation in the RAS pathway
期刊论文
OAI收割
FUTURE MEDICINAL CHEMISTRY, 2025, 卷号: 17, 期号: 6, 页码: 693-708
作者:
Ge, Zhiming
;
Fan, Zisheng
;
He, Wei
;
Zhou, Guizhen
;
Zhou, Yidi
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Targeting the histone reader ZMYND8 inhibits antiandrogen-induced neuroendocrine tumor transdifferentiation of prostate cancer
期刊论文
OAI收割
NATURE CANCER, 2025, 页码: 37
作者:
Wang, Hanling
;
Zhang, Sulin
;
Pan, Qiang
;
Guo, Jiacheng
;
Li, Ni
  |  
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