中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共276条,第1-10条 帮助

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Construction of PROTAC Library via Liquid-Phase Synthesis Enabled by a Hydrophobic Tag 期刊论文  OAI收割
ORGANIC LETTERS, 2026, 卷号: 28, 期号: 8, 页码: 2747-2752
作者:  
Zhou, Yifeng;  He, Wei;  Zhou, Zehui;  Wu, Min;  Wu, Qianping
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Discovery of novel selective PRMT5-MTA inhibitors through structure-based virtual screening 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2026, 卷号: 168, 页码: 17
作者:  
Ma, Ning;  Chen, Yang;  Liang, Yiru;  Chen, Xiaoxu;  Song, Fengnan
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Furo[2,3-f]quinazolin-7(6H)-one Derivatives as Potent, Selective, and Orally Bioavailable MAT2A Inhibitors for MTAP-Deficient Cancer Therapy 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 22, 页码: 24213-24231
作者:  
Shi, Zihan;  Lin, Kexin;  Lin, Lijie;  Chen, Zhiyi;  Xie, Zhiyin
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A pan-KRAS inhibitor and its derived degrader elicit multifaceted anti-tumor efficacy in KRAS-driven cancers 期刊论文  OAI收割
CANCER CELL, 2025, 卷号: 43, 期号: 10, 页码: 32
作者:  
Feng, Juanjuan;  Xiao, Xuanzheng;  Xia, Xinting;  Min, Jian;  Tang, Weiying
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Methotrexate exerts antitumor immune activity and improves the clinical efficacy of immunotherapy in patients with solid tumors 期刊论文  OAI收割
SCIENCE TRANSLATIONAL MEDICINE, 2025, 卷号: 17, 期号: 801, 页码: 18
作者:  
Yang, Ruirui;  Wang, Bei;  Su, Zhaoming;  Song, Ying;  Zhang, Yingying
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Design, synthesis, and activity evaluation of indole derivatives as potential stabilizers for p53 Y220C 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2025, 卷号: 121, 页码: 9
作者:  
Li, Linquan;  Gu, Xi;  Meng, Jingyi;  Wen, Yiming;  Yi, Jing
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Discovery and Identification of a Novel PORCN Inhibitor via Structure-Based Virtual Screening 期刊论文  OAI收割
ACS CHEMICAL BIOLOGY, 2025, 卷号: 20, 期号: 6, 页码: 1319-1332
作者:  
Yang, Xinyu;  Li, Yanbei;  Zhou, Jingyi;  Zhou, Yuanyang;  Lin, Kexin
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Discovery of 3-(Fluoro-imidazolyl)pyridazine Derivatives as Potent STING Agonists with Antitumor Activity 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 10, 页码: 9864-9885
作者:  
Hou, Hui;  Zhou, Jingyi;  Sui, Qibang;  Zhang, Changfa;  Su, Zhaoming
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Recent advances in targeted degradation in the RAS pathway 期刊论文  OAI收割
FUTURE MEDICINAL CHEMISTRY, 2025, 卷号: 17, 期号: 6, 页码: 693-708
作者:  
Ge, Zhiming;  Fan, Zisheng;  He, Wei;  Zhou, Guizhen;  Zhou, Yidi
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Targeting the histone reader ZMYND8 inhibits antiandrogen-induced neuroendocrine tumor transdifferentiation of prostate cancer 期刊论文  OAI收割
NATURE CANCER, 2025, 页码: 37
作者:  
Wang, Hanling;  Zhang, Sulin;  Pan, Qiang;  Guo, Jiacheng;  Li, Ni
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