中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [7]
南海海洋研究所 [1]
采集方式
OAI收割 [8]
内容类型
期刊论文 [8]
发表日期
2024 [1]
2022 [2]
2020 [1]
2018 [1]
2015 [1]
2013 [1]
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学科主题
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Simultaneous determination of unecritinib (TQ-B3101) and its active metabolite crizotinib in rat plasma by LC-MS/MS:An application to pharmacokinetic studies
期刊论文
OAI收割
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2024, 卷号: 246, 页码: 9
作者:
Wang, Hong
;
Chen, Huixian
;
Cui, Xinran
;
Zhang, Yuchen
;
Zhou, Jialan
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2024/07/12
Unecritinib (TQ-B3101)
Crizotinib
Carboxylesterases
LC-MS/MS
Hydrolytic metabolism
Quantification of the major circulating metabolite of BS1801, an ebselen analog, in human plasma
期刊论文
OAI收割
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2022, 卷号: 212, 页码: 10
作者:
Tian, Qianqian
;
Jiang, Jinfang
;
Yin, Hanwei
;
Ma, Jiao
;
Deng, Guozhen
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2022/06/15
BS1801
Ebselen
Circulating metabolite
Human plasma
LC-MS/MS
Investigating the Metabolic Mechanisms of Butaselen, An Ebselen Analog
期刊论文
OAI收割
CURRENT DRUG METABOLISM, 2022, 卷号: 23, 期号: 11, 页码: 928-939
作者:
Tian, Qianqian
;
Jiang, Jinfang
;
Yin, Hanwei
;
Zhang, Yifan
;
Li, Yilin
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2023/04/10
Butaselen
ebselen
covalent binding
Se-methylation
cytosol
TPMT
A marine fungus-derived nitrobenzoyl sesquiterpenoid suppresses receptor activator of NF-kappa B ligand-induced osteoclastogenesis and inflammatory bone destruction
期刊论文
OAI收割
BRITISH JOURNAL OF PHARMACOLOGY, 2020, 卷号: 177, 期号: 18, 页码: 4242, 4260
作者:
Tan, Yanhui
;
Deng, Wende
;
Zhang, Yueyang
;
Ke, Minhong
;
Zou, Binhua
  |  
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2020/09/22
DC-STAMP
NF-kappa B
NFATc1
nitrobenzoyl sesquiterpenoids
osteoclast
osteolysis
Differences in the In Vivo and In Vitro Metabolism of Imrecoxib in Humans: Formation of the Rate-Limiting Aldehyde Intermediate
期刊论文
OAI收割
DRUG METABOLISM AND DISPOSITION, 2018, 卷号: 46, 期号: 9, 页码: 1320-1328
作者:
Hou, Xiangyu
;
Zhou, Jialan
;
Yu, Songda
;
Zhou, Lei
;
Zhang, Yifan
  |  
收藏
  |  
浏览/下载:77/0
  |  
提交时间:2019/01/08
Metabolism of MRX-I, a Novel Antibacterial Oxazolidinone, in Humans: The Oxidative Ring Opening of 2,3-Dihydropyridin-4-One Catalyzed by Non-P450 Enzymes
期刊论文
OAI收割
DRUG METABOLISM AND DISPOSITION, 2015, 卷号: 43, 期号: 5, 页码: 646-659
作者:
Meng, Jian
;
Zhong, Dafang
;
Li, Liang
;
Yuan, Zhengyu
;
Yuan, Hong
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2019/01/08
Metabolism and bioactivation of famitinib, a novel inhibitor of receptor tyrosine kinase, in cancer patients
期刊论文
OAI收割
BRITISH JOURNAL OF PHARMACOLOGY, 2013, 卷号: 168, 期号: 7, 页码: 1687-1706
作者:
Xie, Cen
;
Zhou, Jialan
;
Guo, Zitao
;
Diao, Xingxing
;
Gao, Zhiwei
  |  
收藏
  |  
浏览/下载:60/0
  |  
提交时间:2019/01/08
famitinib
metabolism
bioactivation
quinone-imine
hepatotoxicity
In Vitro Studies on the Oxidative Metabolism of 20(S)-Ginsenoside Rh2 in Human, Monkey, Dog, Rat, and Mouse Liver Microsomes, and Human Liver S9
期刊论文
OAI收割
DRUG METABOLISM AND DISPOSITION, 2012, 卷号: 40, 期号: 10, 页码: 2041-2053
作者:
Li, Liang
;
Chen, Xiaoyan
;
Zhou, Jialan
;
Zhong, Dafang
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2019/01/08