中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [7]
广州生物医药与健康研... [2]
采集方式
OAI收割 [9]
内容类型
期刊论文 [9]
发表日期
2024 [6]
2023 [1]
2007 [2]
学科主题
Chemistry [1]
Pharmacolo... [1]
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浏览/检索结果:
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Application of Electro-Activated Dissociation Fragmentation Technique to Identifying Glucuronidation and Oxidative Metabolism Sites of Vepdegestrant by Liquid Chromatography-High Resolution Mass Spectrometry
期刊论文
OAI收割
DRUG METABOLISM AND DISPOSITION, 2024, 卷号: 52, 期号: 7, 页码: 634-643
作者:
He, Yifei
;
Hou, Pengyi
;
Long, Zhimin
;
Zheng, Yuandong
;
Tang, Chongzhuang
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2024/11/26
IDENTIFYING ACCURATE METABOLISM SITES OF VEPDEGESTRANT USING NOVEL ELECTRON-ACTIVATED DISSOCIATION HIGHRESOLUTION MASS SPECTROMETRY
期刊论文
OAI收割
DRUG METABOLISM AND PHARMACOKINETICS, 2024, 卷号: 55, 页码: 1
作者:
He, Yifei
;
Hou, Pengyi
;
Long, Zhimin
;
Zheng, Yuadong
;
Tang, Chongzhuang
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2024/10/21
AN OVERVIEW OF CDE TECHNICAL GUIDELINE FOR NONCLINICAL STUDY OF ADCS: IMPORTANCE AND STRATEGY OF STUDYING RELEASE OF PAYLOAD-CONTAINING COMPONENTS FROM ADC AND THEIR FURTHER METABOLISM
期刊论文
OAI收割
DRUG METABOLISM AND PHARMACOKINETICS, 2024, 卷号: 55, 页码: 1
作者:
Tang, Chongzhuang
;
Li, Zhiqiang
;
He, Yifei
;
Li, Linwei
;
Diao, Xingxing
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/10/21
Cytochrome P450 2B6 and UDP-Glucuronosyltransferase Enzyme-Mediated Clearance of Ciprofol (HSK3486) in Humans: The Role of Hepatic and Extrahepatic MetabolismS
期刊论文
OAI收割
DRUG METABOLISM AND DISPOSITION, 2024, 卷号: 52, 期号: 2, 页码: 106-117
作者:
Zhou, Yufan
;
Dong, Hongjiao
;
Fan, Jiang
;
Zhu, Mingshe
;
Liu, Lu
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收藏
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浏览/下载:22/0
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提交时间:2024/05/31
Metabolism investigation of the peptide-drug conjugate LN005 in rats using UHPLC-HRMS
期刊论文
OAI收割
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2024, 卷号: 238, 页码: 11
作者:
Wang, Weiqiang
;
Chen, Chong
;
Luo, Jing
;
Tang, Chongzhuang
;
Zheng, Yuandong
  |  
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2024/01/16
LN005
Metabolism
Peptide -drug conjugates
UHPLC-HRMS
Doxorubicin
Metabolite characterisation of the peptide-drug conjugate LN005 in liver S9s by UHPLC-Orbitrap-HRMS
期刊论文
OAI收割
XENOBIOTICA, 2024, 页码: 9
作者:
Yuan, Yali
;
Wang, Weiqiang
;
Luo, Jing
;
Tang, Chongzhuang
;
Zheng, Yuandong
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收藏
  |  
浏览/下载:20/0
  |  
提交时间:2024/02/19
peptide-drug conjugate
PDC
LN005
metabolite identification
liver S9s
Conference report for the 10th China Bioanalysis Forum annual meeting
期刊论文
OAI收割
BIOANALYSIS, 2023, 页码: 4
作者:
Dong, Kelly
;
Zhu, Mingshe
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收藏
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浏览/下载:18/0
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提交时间:2023/12/19
China Bioanalysis Forum
CBF
ICH M10
DMPK and Bioanalysis for New Modalities
Development and full validation of six inhibition assays for five major cytochrome P450 enzymes in human liver microsomes using an automated 96-well microplate incubation format and LC-MS/MS analysis
期刊论文
OAI收割
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2007, 卷号: 44, 期号: 1, 页码: 211-223
作者:
Dai, Renke
;
Yao, Ming
;
Zhu, Mingshe
;
Sinz, Michael W.
;
Zhang, Hongjian
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收藏
  |  
浏览/下载:16/0
  |  
提交时间:2018/12/13
Development and full validation of six inhibition assays for five major cytochrome P450 enzymes in human liver microsomes using an automated 96-well microplate incubation format and LC-MS/MS analysis
期刊论文
OAI收割
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2007, 卷号: 44, 期号: 1, 页码: 211-223
Yao, Ming
;
Zhu, Mingshe
;
Sinz, Michael W.
;
Zhang, Hongjian
;
Humphreys, W. Griffith
;
Rodrigues, A. David
;
Dai, Renke
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2016/12/16