中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [8]
昆明植物研究所 [1]
采集方式
OAI收割 [9]
内容类型
期刊论文 [9]
发表日期
2021 [1]
2012 [2]
2010 [2]
2009 [3]
2008 [1]
学科主题
Pharmacolo... [3]
Chemistry [2]
Biochemist... [1]
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Bitter Melon and Diabetes Mellitus
期刊论文
OAI收割
FOOD REVIEWS INTERNATIONAL, 2021
作者:
Gao,Ya
;
Li,Xian
;
Huang,Yanjie
;
Chen,Jianchao
;
Qiu,Minghua
  |  
收藏
  |  
浏览/下载:47/0
  |  
提交时间:2022/04/02
Bitter melon
diabetes mellitus
crude extracts
phyto-metabolites
hypoglycemic mechanism
MOMORDICA-CHARANTIA L.
11-BETA-HYDROXYSTEROID DEHYDROGENASE TYPE-1
ALPHA-GLUCOSIDASE INHIBITION
INSULIN-RESISTANCE
ANTIDIABETIC ACTIVITIES
GUT MICROBIOTA
STRUCTURAL-CHARACTERIZATION
PHENOLIC-COMPOUNDS
OXIDATIVE STRESS
PROTEIN-KINASE
Discovery of 2-Alkyl-1-arylsulfonylprolinamides as 11 beta-Hydroxysteroid Dehydrogenase Type 1 Inhibitors
期刊论文
OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2012, 卷号: 3, 期号: 10, 页码: 793-798
作者:
Yu, Jianxin
;
Liu, Haiyan
;
Xia, Guangxin
;
Liu, Lin
;
Xu, Zhenmin
  |  
收藏
  |  
浏览/下载:152/0
  |  
提交时间:2019/01/08
metabolic syndrome
enzyme inhibitor
11 beta-hydroxysteroid dehydrogenase type 1
sulfonamide
2-alkylproline
prolinamide
Emodin, an 11 beta-hydroxysteroid dehydrogenase type 1 inhibitor, regulates adipocyte function in vitro and exerts anti-diabetic effect in ob/ob mice
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2012, 卷号: 33, 期号: 9, 页码: 1195-1203
作者:
Wang, Yue-jing
;
Huang, Su-ling
;
Feng, Ying
;
Ning, Meng-meng
;
Leng, Ying
  |  
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2019/01/08
emodin
11 beta-hydroxysteroid dehydrogenase type 1
adipocyte
glucocorticoid
type 2 diabetes
ob/ob mice
Emodin, a natural product, selectively inhibits 11 beta-hydroxysteroid dehydrogenase type 1 and ameliorates metabolic disorder in diet-induced obese mice
期刊论文
OAI收割
BRITISH JOURNAL OF PHARMACOLOGY, 2010, 卷号: 161, 期号: 1, 页码: 113-126
作者:
Feng, Ying
;
Huang, Su-Ling
;
Dou, Wei
;
Zhang, Song
;
Chen, Jun-Hua
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2019/01/08
emodin
11 beta-hydroxysteroid dehydrogenase type 1
diet-induced obese mice
insulin resistance
metabolic syndrome
type 2 diabetes
Derivatives of (phenylsulfonamido-methyl)nicotine and (phenylsulfonamido-methyl)thiazole as novel 11 beta-hydroxysteroid dehydrogenase type 1 inhibitors: synthesis and biological activities in vitro
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2009, 卷号: 30, 期号: 9, 页码: 1344-1350
作者:
Zhang, Xu
;
Zhou, Yang
;
Shen, Yu
;
Du, Li-li
;
Chen, Jun-hua
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2019/01/08
11 beta-hydroxysteroid dehydrogenase type 1
inhibitors
molecular modeling