中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共6条,第1-6条 帮助

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Targeted degradation of GOLM1 by CC-885 via CRL4-CRBN E3 ligase inhibits hepatocellular carcinoma progression 期刊论文  OAI收割
CELLULAR SIGNALLING, 2025, 卷号: 130, 页码: 15
作者:  
He, Jingliang;  Guo, Jingli;  Liu, Shunfang;  Li, Hanxue;  Ma, Yuanyuan
  |  收藏  |  浏览/下载:2/0  |  提交时间:2025/04/24
E3 ligase ligand optimization of Clinical PROTACs 期刊论文  OAI收割
FRONTIERS IN CHEMISTRY, 2023, 卷号: 11, 页码: 15
作者:  
Jiang, Hanrui;  Xiong, Huan;  Gu, Shuang-Xi;  Wang, Mingliang
  |  收藏  |  浏览/下载:26/0  |  提交时间:2023/04/10
Design, synthesis, and biological evaluation of Wee1 kinase degraders 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 243, 页码: 21
作者:  
Zhu, Shulei;  Liu, Jieyu;  Xiao, Donghuai;  Wang, Peipei;  Ma, Jingkun
  |  收藏  |  浏览/下载:68/0  |  提交时间:2022/11/11
Design, Synthesis, and Biological Evaluation of HDAC Degraders with CRBN E3 Ligase Ligands 期刊论文  OAI收割
MOLECULES, 2021, 卷号: 26, 期号: 23, 页码: 19
作者:  
Lu, Yingxin;  Sun, Danwen;  Xiao, Donghuai;  Shao, Yingying;  Su, Mingbo
  |  收藏  |  浏览/下载:56/0  |  提交时间:2022/06/15
Discovery of thalidomide-based PROTAC small molecules as the highly efficient SHP2 degraders 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 218, 页码: 14
作者:  
Yang, Xiangbo;  Wang, Zhijia;  Pei, Yuan;  Song, Ning;  Xu, Lei
  |  收藏  |  浏览/下载:43/0  |  提交时间:2021/08/17
The novel cereblon modulator CC-885 inhibits mitophagy via selective degradation of BNIP3L 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 9
作者:  
Hao, Bing-bing;  Li, Xiao-jing;  Jia, Xing-long;  Wang, Yu-xing;  Zhai, Lin-hui
  |  收藏  |  浏览/下载:36/0  |  提交时间:2020/07/01