中国科学院机构知识库网格
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Development and Validation of an ADA-Tolerant Assay for Quantification of an Exatecan-Based ADC in Monkey Plasma
期刊论文
OAI收割
MOLECULES, 2024, 卷号: 29, 期号: 3, 页码: 14
作者:
Tao, Yimin
;
Lu, Wei
;
Gao, Jinli
;
Yang, Shuangshuang
;
Ruan, Chaoyi
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2024/03/13
antibody-drug conjugate (ADC)
bioanalysis
anti-drug antibody (ADA)
ligand binding assay (LBA)
ADA-tolerant assay
Inhibiting Endothelial Cell-Mediated T Lymphocyte Apoptosis with Integrin-Targeting Peptide-Drug Conjugate Filaments for Chemoimmunotherapy of Triple-Negative Breast Cancer
期刊论文
OAI收割
ADVANCED MATERIALS, 2023, 页码: 12
作者:
Cai, Ying
;
Zhu, Binyu
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2024/01/16
Fas ligand
immunotherapy
peptide-drug conjugate
triple-negative breast cancer
tumor-associated endothelial cells
Molecular recognition of niacin and lipid-lowering drugs by the human hydroxycarboxylic acid receptor 2
期刊论文
OAI收割
CELL REPORTS, 2023, 卷号: 42, 期号: 11, 页码: 19
作者:
Zhu, Shengnan
;
Yuan, Qingning
;
Li, Xinzhu
;
He, Xinheng
;
Shen, Shiyi
  |  
收藏
  |  
浏览/下载:192/0
  |  
提交时间:2024/01/16
different ligands
recognition
ligand selectivity
receptor
Discovery of Potent and Selective CB2 Agonists Utilizing a Function-Based Computational Screening Protocol
期刊论文
OAI收割
ACS CHEMICAL NEUROSCIENCE, 2023, 卷号: 14, 期号: 21, 页码: 3941-3958
作者:
Ge, Haixia
;
Ji, Beihong
;
Fang, Jiahui
;
Wang, Jiayang
;
Li, Jing
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2023/12/11
function-based ligand design
receptor-ligandbinding profile
CB1/CB2
structure-activityrelationship
D3CARP: a comprehensive platform with multiple-conformation based docking, ligand similarity search and deep learning approaches for target prediction and virtual screening
期刊论文
OAI收割
COMPUTERS IN BIOLOGY AND MEDICINE, 2023, 卷号: 164, 页码: 8
作者:
Shi, Yulong
;
Zhang, Xinben
;
Yang, Yanqing
;
Cai, Tingting
;
Peng, Cheng
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2023/10/17
Target prediction
Virtual screening
Molecular docking
Ligand similarity search
Deep learning
Structural insights into the interaction of three Y- shaped ligands with PI3Kα
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2023, 卷号: 120, 期号: 34, 页码: 9
作者:
Zhou, Qingtong
;
Liu, Xiao
;
Neri, Dario
;
Li, Wenxin
;
Favalli, Nicholas
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2023/12/08
phosphoinositide 3-kinase
drug target
ligand
binding pocket
chemical scaffold
Surface modification of Fe5C2 by binding silica-based ligand: A theoretical explanation of enhanced C2 oxygenate selectivity
期刊论文
OAI收割
MOLECULAR CATALYSIS, 2023, 卷号: 547, 页码: 113333
作者:
Yin, Junqing
;
Wang, Shuyuan
;
Xu, Dan
;
You, Yong
;
Liu, Xingchen
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2023/09/05
Surface modification
Iron carbide
Support -like ligand
Catalytic selectivity
Fischer-Tropsch Synthesis
Receptor-Ligand Binding: Effect of Mechanical Factors
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2023, 卷号: 24, 期号: 10, 页码: 9062
作者:
Du, Ruotian
;
Li L(李龙)
;
Ji, Jing
;
Fan, Yubo
;
Li L(李龙)
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2023/06/15
receptor-ligand binding
tension
shear stress
stretch
compression
substrate stiffness
biomechanics
mechanotransduction
Two dimensional measurements of receptor ligand interactions
期刊论文
OAI收割
FRONTIERS IN MOLECULAR BIOSCIENCES, 2023, 卷号: 10, 页码: 1154074
作者:
Zheng SJ(郑松杰)
;
Zou M(邹敏)
;
Shao YF(邵颖峰)
;
Wu, Huaping
;
Wu, Helong
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2023/04/20
receptor ligand interaction
binding kinetics
kinetic on rate
kinetic off rate
binding affinity
two dimensional measuring methods
Modulating Catalytic Activity and Stability of Atomically Precise Gold Nanoclusters as Peroxidase Mimics via Ligand Engineering
期刊论文
OAI收割
ACS NANO, 2023, 页码: 10
作者:
Shan, Huiting
;
Shi, Jiafu
;
Chen, Tiankai
;
Cao, Yitao
;
Yao, Qiaofeng
  |  
收藏
  |  
浏览/下载:0/0
  |  
提交时间:2023/05/19
gold nanoclusters
ligand engineering
peroxidase mimic catalysis
catalytic activity
stability