中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [5]
采集方式
OAI收割 [5]
内容类型
期刊论文 [5]
发表日期
2023 [1]
2021 [1]
2019 [1]
2018 [1]
2015 [1]
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Discovery of 4-oxo-4,5-dihydropyrazolo[1,5-a]quinoxaline-7-carboxamide derivatives as PI3K alpha inhibitors via virtual screening and docking-based structure optimization
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2023, 卷号: 86, 页码: 15
作者:
Gu, Dongyan
;
Zhang, Mengmeng
;
Cai, Lvtao
;
Wang, Chang
;
Zhou, Yu -Bo
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2023/10/17
PI3K alpha inhibitors
Virtual screening
Structure optimization
Discovery of 2-(5-(quinolin-6-yl)-1,3,4-oxadiazol-2-yl)acetamide derivatives as novel PI3K alpha inhibitors via docking-based virtual screening
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 29, 页码: 9
作者:
Gu, Dongyan
;
Cheng, Gang
;
Zhang, Mengmeng
;
Zhou, Yu-Bo
;
Li, Jia
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2021/05/24
PI3K alpha inhibitors
Virtual screening
2-(5-(quinolin-6-yl)-1,3,4 oxadiazol-2-yl)acetamide
Molecular dynamics
Design, synthesis, and biological evaluation of thieno[3,2-d]pyrimidine derivatives as potential simplified phosphatidylinositol 3-kinase alpha inhibitors
期刊论文
OAI收割
CHEMICAL BIOLOGY & DRUG DESIGN, 2019, 卷号: 94, 期号: 6, 页码: 2013-2022
作者:
Yang, Xiuyan
;
Deng, Meng
;
Zhang, Xi
;
Wang, Yi
;
Song, Kun
  |  
收藏
  |  
浏览/下载:42/0
  |  
提交时间:2020/07/01
PI3K alpha inhibitors
proliferation inhibition
thieno[3
2-d]pyrimidine derivatives
High-throughput screening campaigns against a PI3K alpha isoform bearing the H1047R mutation identified potential inhibitors with novel scaffolds
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 11, 页码: 1816-1822
作者:
Wang, Jia
;
Gong, Grace Qun
;
Zhou, Yan
;
Lee, Woo-Jeong
;
Buchanan, Christina Maree
  |  
收藏
  |  
浏览/下载:95/0
  |  
提交时间:2019/01/08
high throughput screening
PI3 kinase
PI3K alpha H1047R
inhibitors
molecular modeling
designsynthesisandbiologicalevaluationofacylhydrazonederivativesaspi3kinhibitors
期刊论文
OAI收割
chinesechemicalletters, 2015, 卷号: 26, 期号: 1, 页码: 118
作者:
Gao Guorui
;
Liu Jiali
;
Mei Desheng
;
Ding Jian
;
Meng Linghua
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2020/07/01
PI3-KINASE P110-ALPHA INHIBITORS
3-KINASE
PATHWAY
PI3K
Inhibitor
Aclhydrazone