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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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福建物质结构研究所 [20]
上海药物研究所 [12]
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期刊论文 [60]
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Copper pyrazole addition regulates soil mineral nitrogen turnover by mediating microbial traits
期刊论文
OAI收割
FRONTIERS IN MICROBIOLOGY, 2024, 卷号: 15
作者:
Wang, Yuming
;
Zhong, Wenling
;
Zhang, Xiwen
;
Cao, Minghui
;
Ni, Zheng
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2024/11/20
nitrification inhibitors
copper pyrazole
soil mineral nitrogen
microbial community
nitrogen-cycling genes
fDiscovery of pyrazole-thiophene derivatives as highly Potent, orally active Akt inhibitors
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 180, 页码: 72-85
作者:
Zhan, Wenhu
;
Che, Jinxin
;
Xu, Lei
;
Wu, Yizhe
;
Hu, Xiaobei
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2020/07/01
Pyrazole-thiophene derivatives
Akt inhibitor
Antitumor
Discovery of 1,3-diphenyl-1H-pyrazole derivatives containing rhodanine-3-alkanoic acid groups as potential PTP1B inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 卷号: 29, 期号: 10, 页码: 1187-1193
作者:
Sun, Liangpeng
;
Wang, Peipei
;
Xu, Lili
;
Gao, Lixin
;
Li, Jia
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2020/07/01
PTP1B inhibitor
1,3-Diphenyl-1H-pyrazole
Rhodanine-3-alkanoic acid
A novel series of 4-methyl substituted pyrazole derivatives as potent glucagon receptor antagonists: Design, synthesis and evaluation of biological activities
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 期号: 8, 页码: 1896-1908
作者:
Shu, Shuangjie
;
Dai, Antao
;
Wang, Jiang
;
Wang, Bin
;
Feng, Yang
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2019/01/08
Pyrazole derivatives
Glucagon receptor antagonist
Docking study
Binding pocket
Metal organic frameworks (MOFs) for magnetic solid-phase extraction of pyrazole/pyrrole pesticides in environmental water samples followed by HPLC-DAD determination
期刊论文
OAI收割
TALANTA, 2016, 卷号: 161, 页码: 686-692
作者:
Ma, Jiping
;
Yao, Zhidan
;
Hou, Liwei
;
Lu, Wenhui
;
Yang, Qipeng
收藏
  |  
浏览/下载:54/0
  |  
提交时间:2016/12/19
Metal-organic frameworks (MOFs)
Magnetic solid-phase extraction
Pyrazole
Pyrrole
Water samples
Design, synthesis, structure-activity relationships, and docking studies of pyrazole-containing derivatives as a novel series of potent glucagon receptor antagonists
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 12, 页码: 2852-2863
作者:
Shu, Shuangjie
;
Cai, Xiaoqing
;
Li, Jia
;
Feng, Yang
;
Dai, Antao
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2019/01/08
Glucagon receptor
Antagonist
Molecular docking
Pyrazole
Type 2 diabetes mellitus
Structural optimization and biological evaluation of 1,5-disubstituted pyrazole-3-carboxamines as potent inhibitors of human 5-lipoxygenase
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2016, 卷号: 6, 期号: 1, 页码: 32-45
作者:
Zhou, Yu
;
Liu, Jun
;
Zheng, Mingyue
;
Zheng, Shuli
;
Jiang, Chunyi
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收藏
  |  
浏览/下载:29/0
  |  
提交时间:2019/01/08
5-Lipoxygenase
5-LOX inhibitors
Pyrazole derivatives
Leukotrienes-related diseases
In vivo
Benzo-fuse heterocyle
Ischemic incults
Brain inflammation
structuraloptimizationandbiologicalevaluationofl5disubstitutedpyrazole3carboxaminesaspotentinhibitorsofhuman5lipoxygenase
期刊论文
OAI收割
actapharmaceuticasinicab, 2016, 卷号: 6, 期号: 1, 页码: 32
作者:
Zhou Yu
;
Liu Jun
;
Zheng Mingyue
;
Zheng Shuli
;
Jiang Chunyi
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2020/07/01
5-Lipoxygenase
5-LOX inhibitors
Pyrazole derivatives
Leukotrienes-related diseases
In vivo
Benzo-fused heterocycle
Ischemic incults
Brain inflammation
Structural optimization and biological evaluation of l,5-disubstituted pyrazole-3-carboxamines as potent inhibitors of human 5-lipoxygenase
期刊论文
OAI收割
Acta Pharmaceutica Sinica B, 2016, 卷号: 6, 期号: 1, 页码: 32
作者:
Zhou Yu
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2020/12/24
5-Lipoxygenase
5-LOX inhibitors
Pyrazole derivatives
Leukotrienes-related diseases
In vivo
Benzo-fused heterocycle
Ischemic incults
Brain inflammation
Structure-Activity Relationship of Diacylhydrazine Derivatives Fluoride-Containing Pyrazolyl Moiety
期刊论文
OAI收割
ASIAN JOURNAL OF CHEMISTRY, 2013, 卷号: 25, 期号: 15, 页码: 8600-8602
作者:
Bi, Hui-Min
;
Xie, Peng-Tao
;
Li, Shu-Xian
;
Li, Yong-Li
;
Dong, Chun-Hua
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2019/04/09
Fluoride Pyrazole
Diacylhydrazine
Biological Activity
Structure-activity Relationship