中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
长春应用化学研究所 [4]
上海药物研究所 [3]
昆明植物研究所 [1]
采集方式
OAI收割 [8]
内容类型
期刊论文 [8]
发表日期
2018 [1]
2016 [1]
2015 [2]
2013 [1]
2008 [1]
2007 [2]
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Design, synthesis and biological evaluation of C(4) substituted monobactams as antibacterial agents against multidrug-resistant Gram-negative bacteria
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 151, 页码: 98-109
作者:
Kou, Qunhuan
;
Wang, Ting
;
Zou, Feng
;
Zhang, Shuhua
;
Chen, Qian
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2019/01/08
Monobactam
C(4) substituents
Pyridone
MDR Gram-negative bacteria
Antibacterial activity
Discovery of 1,3-Diaryl-pyridones as Potent VEGFR-2 Inhibitors: Design, Synthesis, and Biological Evaluation
期刊论文
OAI收割
CHEMICAL BIOLOGY & DRUG DESIGN, 2016, 卷号: 87, 期号: 5, 页码: 694-703
作者:
Yan, Wei
;
Huang, Zhaoru
;
Wang, Zhengyu
;
Cao, Sufen
;
Tong, Linjiang
  |  
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2019/01/08
1
3-Diaryl-pyridone
angiogenesis
anticancer agent
Chan-Lam coupling
VEGFR-2 inhibitors
Three new anti-HBV active constituents from the traditional Chinese herb of Yin-Chen (Artemisia scoparia)
期刊论文
OAI收割
JOURNAL OF ETHNOPHARMACOLOGY, 2015, 卷号: 176, 页码: 109-117
作者:
Geng, Chang-An
;
Huang, Xiao-Yan
;
Chen, Xing-Long
;
Ma, Yun-Bao
;
Rong, Guang-Qing
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2016/02/01
Artemisia scoparia (Yin-Chen)
4-pyridone glycoside
Polyacetylenes
Anti-HBV activity
LCMS
Discovery of potent 1H-imidazo[4,5-b]pyridine-based c-Met kinase inhibitors via mechanism-directed structural optimization
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 3, 页码: 708-716
作者:
An, Xiao-De
;
Liu, Hongyan
;
Xu, Zhong-Liang
;
Jin, Yi
;
Peng, Xia
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2019/01/08
c-Met tyrosine kinase
Small molecule inhibitor
Imidazonaphthyridinone
Imidazopyridine
Binding mode
Pyridone-3-carboxamide
Cyclopropane-1,1-dicarboxamide
Hydrogen Bond-Assisted 6 pi-Azaelectrocyclization of Penta-2,4-dienamides: Synthesis of Dihydropyridin-2(3H)-ones
期刊论文
OAI收割
journal of organic chemistry, 2013, 卷号: 78, 期号: 7, 页码: 3323-3328
Liu X
;
Zhang N
;
Yang JM
;
Liang YJ
;
Zhang R
;
Dong DW
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2014/04/16
ELECTROCYCLIC RING-CLOSURE
DIELS-ALDER REACTIONS
ENANTIOSELECTIVE SYNTHESIS
CLOSING METATHESIS
HIGHLY EFFICIENT
BRASSARDS DIENE
DELTA-LACTAMS
2-PYRIDONE
CYCLIZATION
AMINES
A Facile and Efficient Synthesis of Polyfunctionalized Pyridin-2(1H)-ones from β-Oxo Amides under Vilsmeier Conditions
期刊论文
OAI收割
Organic letters, 2008, 卷号: 10, 期号: 2, 页码: 345-348
Xiang DX
;
Wang KW
;
Liang YJ
;
Zhou GY
;
Dong DW*
收藏
  |  
浏览/下载:186/53
  |  
提交时间:2010/04/14
ONE-POT SYNTHESIS
HAACK REACTION
KETENE DITHIOACETALS
PYRIDINE RINGS
CYCLOADDITION
2-PYRIDONE
REAGENTS
CONSTRUCTION
CYCLIZATION
ANNULATION
Vilsmeier-Haack reactions of 2-arylamino-3-acetyl-5,6-dihydro-4H-pyrans toward the synthesis of highly substituted pyridin-2(1H)-ones
期刊论文
OAI收割
journal of organic chemistry, 2007, 卷号: 72, 期号: 22, 页码: 8593-8596
Xiang DX
;
Yang Y
;
Zhang R
;
Liang YJ
;
Pan W
;
Huang J
;
Dong DW
收藏
  |  
浏览/下载:184/30
  |  
提交时间:2010/07/13
CROSS-COUPLING REACTIONS
ONE-POT SYNTHESIS
CARBONYL-COMPOUNDS
PYRIDINE RINGS
STRATEGY
CYCLOADDITION
2-PYRIDONE
ANNULATION
QUINOLINES
EFFICIENT
Efficient one-pot synthesis of highly substituted pyridin-2(1H)-ones via the Vilsmeier-Haack reaction of 1-acetyl,1-carbamoyl cyclopropanes
期刊论文
OAI收割
organic letters, 2007, 卷号: 9, 期号: 12, 页码: 2421-2423
Pan W
;
Dong DW
;
Wang KW
;
Zhang J
;
Wu R
;
Xiang DX
;
Liu Q
收藏
  |  
浏览/下载:178/37
  |  
提交时间:2010/07/13
PYRIDINE RINGS
CYCLOADDITION
DERIVATIVES
2-PYRIDONE
STRATEGY
INHIBITORS
PYRIDONES