机构

• 上海药物研究所 [6]
• 上海生物化学与细胞生... [5]
• 昆明动物研究所 [2]

采集方式

• OAI收割 [13]

内容类型

• 期刊论文 [13]

发表日期

• 2025 [1]
• 2024 [2]
• 2021 [1]
• 2019 [1]
• 2018 [3]
• 2015 [3]
• 更多

学科主题

• Biochemist... [1]
• Cell Biolo... [1]
• Developmen... [1]

筛选

浏览/检索结果: 共13条，第1-10条 帮助 条数/页： 5101520253035404550556065707580859095100 排序方式： 请选择题名升序题名降序发表日期升序发表日期降序提交时间升序提交时间降序作者升序作者降序 In vitro and In vivo Drug Metabolism Analysis of BPI-460372-A Covalent TEAD1/3/4 Inhibitor 期刊论文  OAI收割 CURRENT DRUG METABOLISM, 2025, 页码: 15 作者:  Liu, Xiaoyun;  Zhong, Dafang;  Tang, Chongzhuang;  Xu, Xiaofeng;  Lan, Hong   |  收藏  |  浏览/下载：0/0  |  提交时间：2025/04/24 Hippo signaling pathway  TEAD inhibitor  covalent inhibitor  BPI-460372  UHPLC-Orbitrap-HRMS  cysteine  S-conjugate beta-lyase.   Design, Synthesis, and Bioevaluation of Transcriptional Enhanced Assocciated Domain (TEAD) PROTAC Degraders 期刊论文  OAI收割 ACS MEDICINAL CHEMISTRY LETTERS, 2024, 卷号: 15, 期号: 5, 页码: 631-639 作者:  Li, Huajie;  Ge, Zhiming;  Lin, Kexin;  He, Wei;  Chu, Qinyu   |  收藏  |  浏览/下载：41/0  |  提交时间：2024/06/27 Hippo pathway  TEAD  PROTAC  Selectivity   Regulation of hippo signaling mediated apoptosis by Rauvolfia tetraphylla in triple-negative breast cancer 期刊论文  OAI收割 MEDICAL ONCOLOGY, 2024, 卷号: 41, 期号: 5, 页码: 14 作者:  Balavaishnavi, B.;  Kamaraj, M.;  Nithya, T. G.;  Santhosh, P.;  Gokilalakshmi, S.   |  收藏  |  浏览/下载：19/0  |  提交时间：2024/05/07 Anti-proliferative effect  Hippo pathway  MDA-MB-231 cells  Apoptosis  Rauvolfia tetraphylla   Discovery of a subtype-selective, covalent inhibitor against palmitoylation pocket of TEAD3 期刊论文  OAI收割 ACTA PHARMACEUTICA SINICA B, 2021, 卷号: 11, 期号: 10, 页码: 3206-3219 作者:  Lu, Tian;  Li, Yong;  Lu, Wenchao;  Spitters, Twgm;  Fang, Xueyu   |  收藏  |  浏览/下载：54/0  |  提交时间：2021/12/01 Hippo pathway  TEAD3  Covalent inhibitor  Palmitoylation inhibitor   Discovery and biological evaluation of vinylsulfonamide derivatives as highly potent, covalent TEAD autopalmitoylation inhibitors 期刊论文  OAI收割 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 184, 页码: 15 作者:  Lu, Wenchao;  Wang, Jun;  Li, Yong;  Tao, Hongru;  Xiong, Huan   |  收藏  |  浏览/下载：102/0  |  提交时间：2020/07/01 Hippo pathway  TEAD transcription factor  Covalent inhibitor  Palmitoylation inhibitor   Cyclopeptide RA-V Inhibits Organ Enlargement and Tumorigenesis Induced by YAP Activation 期刊论文  OAI收割 CANCERS, 2018, 卷号: 10, 期号: 11 作者:  Ji, Xinyan   |  收藏  |  浏览/下载：103/0  |  提交时间：2019/01/08 hippo pathway  YAP  TAZ  RA-V  cancer  organ size  protein synthesis   Targeting IRF3 as a YAP agonist therapy against gastric cancer 期刊论文  OAI收割 JOURNAL OF EXPERIMENTAL MEDICINE, 2018, 卷号: 215, 期号: 2, 页码: 699-718 作者:  Jiao, Shi;  Guan, Jingmin;  Chen, Min;  Wang, Wenjia   |  收藏  |  浏览/下载：82/0  |  提交时间：2019/04/28 Hippo Signaling Pathway  Organ Size Control  Interferon Regulatory Factor-3  Minor Aphthous Ulceration  Cell Contact Inhibition  Tumor-suppressor  Innate Immunity  Growth-control  Intestinal Regeneration  Colorectal-cancer   PRDM4 mediates YAP-induced cell invasion by activating leukocyte-specific integrin beta 2 expression 期刊论文  OAI收割 EMBO REPORTS, 2018, 卷号: 19, 期号: 6, 页码: - 作者:  Liu, Huan;  Dai, Xiaoming   |  收藏  |  浏览/下载：60/0  |  提交时间：2019/04/28 Yes-associated Protein  Histone Methyltransferase Complex  Hippo Signaling Pathway  Organ Size Control  Transcription Factor  Prostate-cancer  Tissue Homeostasis  Gene-expression  Growth-control  Myeloid Cells   Structural dissection of Hippo signaling 期刊论文  OAI收割 ACTA BIOCHIMICA ET BIOPHYSICA SINICA, 2015, 卷号: 47, 期号: 1, 页码: 29-38 作者:  Shi, ZB;  Jiao, S;  Zhou, ZC 收藏  |  浏览/下载：35/0  |  提交时间：2015/07/22 Hippo pathway  three-dimensional structure  protein-protein  DNA interaction  regulatory mechanism   The interplay between TEAD4 and KLF5 promotes breast cancer partially through inhibiting the transcription of p27(Kip1) 期刊论文  OAI收割 ONCOTARGET, 2015, 卷号: 6, 期号: 19, 页码: 17685-17697 作者:  Wang CY;  Nie Z;  Zhou ZM;  Zhang HL;  Liu R 收藏  |  浏览/下载：22/0  |  提交时间：2015/09/01 TEAD4  KLF5  p27  hippo pathway  TNBC