中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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  • 2016 [125]
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Design, Synthesis, and Pharmacological Evaluation of 2-(2,5-Dimethyl-5,6,7,8-tetrahydroquinolin-8-yl)-N-aryl Propanamides as Novel Smoothened (Smo) Antagonists 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 24, 页码: 11050-11068
作者:  
Liu, Gang;  Xue, Ding;  Yang, Jun;  Wan, Juan;  Liu, Xiaohua
  |  收藏  |  浏览/下载:54/0  |  提交时间:2019/01/08
Identification and characterization of naturally occurring inhibitors against human carboxylesterase 2 in White Mulberry Root-bark 期刊论文  OAI收割
FITOTERAPIA, 2016, 卷号: 115, 页码: 57-63
作者:  
Liang, Xin-Miao;  Liu, Ya-Jing;  Li, Shi-Yang;  Hou, Jie;  Liu, Yan-Fang
收藏  |  浏览/下载:25/0  |  提交时间:2017/10/29
Crystal structure of FabZ-ACP complex reveals a dynamic seesaw-like catalytic mechanism of dehydratase in fatty acid biosynthesis 期刊论文  OAI收割
CELL RESEARCH, 2016, 卷号: 26, 期号: 12, 页码: 1330-1344
作者:  
Zhang, Lin;  Xiao, Jianfeng;  Xu, Jianrong;  Fu, Tianran;  Cao, Zhiwei
  |  收藏  |  浏览/下载:15/0  |  提交时间:2019/01/08
Targeting Hsp90 with FS-108 circumvents gefitinib resistance in EGFR mutant non-small cell lung cancer cells 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2016, 卷号: 37, 期号: 12, 页码: 1587-1596
作者:  
Wang, Yue-qin;  Shen, Ai-jun;  Sun, Jing-ya;  Wang, Xin
  |  收藏  |  浏览/下载:31/0  |  提交时间:2019/01/08
Design, synthesis and biological evaluation of novel non-covalent piperidine-containing peptidyl proteasome inhibitors 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 23, 页码: 6206-6214
作者:  
Zhang, Jiankang;  Gao, Lixin;  Xi, Jianjun;  Sheng, Li;  Zhao, Yanmei
  |  收藏  |  浏览/下载:51/0  |  提交时间:2019/01/08
DESIGN, SYNTHESIS, IN VITRO ANTIPROLIFERATIVE ACTIVITY EVALUATION OF 2-ALICANOYLAMIDOTHIOPHENE-3-CARBOXAMIDE DERIVATIVES 期刊论文  OAI收割
HETEROCYCLES, 2016, 卷号: 92, 期号: 12, 页码: 2145-2165
作者:  
Zhang, Jiefeng;  Guan, Fengjie;  Qiu, Jiakun;  Fang, Yanfen;  Yu, Lifang
  |  收藏  |  浏览/下载:28/0  |  提交时间:2019/01/08
Identification and biochemical characterization of DC07090 as a novel potent small molecule inhibitor against human enterovirus 71 3C protease by structure-based virtual screening 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 124, 页码: 981-991
作者:  
Ma, Guang-Hui;  Ye, Yan;  Zhang, Dan;  Xu, Xin;  Si, Pei
  |  收藏  |  浏览/下载:29/0  |  提交时间:2019/01/08
Potent Antitumor Activities and Structure Basis of the Chiral beta-Lactam Bridged Analogue of Combretastatin A-4 Binding to Tubulin 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 22, 页码: 10329-10334
作者:  
Zhou, Pengfei;  Liu, Yan;  Zhou, Lu;  Zhu, Kongkai;  Feng, Kechang
  |  收藏  |  浏览/下载:21/0  |  提交时间:2019/01/08
16-nor Limonoids from Harrisonia perforata as promising selective 11 beta-HSD1 inhibitors 期刊论文  OAI收割
SCIENTIFIC REPORTS, 2016, 卷号: 6
作者:  
Xiao-HuiYan;  Yi, Ping;  Cao, Pei;  Yang, Shi-Ying;  Fang, Xin
  |  收藏  |  浏览/下载:14/0  |  提交时间:2019/01/08
An Update on Poly(ADP-ribose)polymerase-1 (PARP-1) Inhibitors: Opportunities and Challenges in Cancer Therapy 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 21, 页码: 9575-9598
作者:  
Wang, Ying-Qing;  Wang, Ping-Yuan;  Wang, Yu-Ting;  Yang, Guang-Fu;  Zhang, Ao
  |  收藏  |  浏览/下载:15/0  |  提交时间:2019/01/08