中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [84]
广州能源研究所 [8]
植物研究所 [6]
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大连化学物理研究所 [3]
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期刊论文 [124]
学位论文 [1]
发表日期
2016 [125]
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Plant Scie... [4]
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共125条,第1-10条
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发表日期:2016
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Design, Synthesis, and Pharmacological Evaluation of 2-(2,5-Dimethyl-5,6,7,8-tetrahydroquinolin-8-yl)-N-aryl Propanamides as Novel Smoothened (Smo) Antagonists
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 24, 页码: 11050-11068
作者:
Liu, Gang
;
Xue, Ding
;
Yang, Jun
;
Wan, Juan
;
Liu, Xiaohua
  |  
收藏
  |  
浏览/下载:54/0
  |  
提交时间:2019/01/08
Identification and characterization of naturally occurring inhibitors against human carboxylesterase 2 in White Mulberry Root-bark
期刊论文
OAI收割
FITOTERAPIA, 2016, 卷号: 115, 页码: 57-63
作者:
Liang, Xin-Miao
;
Liu, Ya-Jing
;
Li, Shi-Yang
;
Hou, Jie
;
Liu, Yan-Fang
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2017/10/29
White Mulberry Root-bark
Human carboxylesterase 2 (hCE2)
Inhibitory effects
Sanggenone D
Kuwanon G
Sanggenone C
Crystal structure of FabZ-ACP complex reveals a dynamic seesaw-like catalytic mechanism of dehydratase in fatty acid biosynthesis
期刊论文
OAI收割
CELL RESEARCH, 2016, 卷号: 26, 期号: 12, 页码: 1330-1344
作者:
Zhang, Lin
;
Xiao, Jianfeng
;
Xu, Jianrong
;
Fu, Tianran
;
Cao, Zhiwei
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2019/01/08
fatty acid biosynthesis
dehydratase
ACP
complex structure
Targeting Hsp90 with FS-108 circumvents gefitinib resistance in EGFR mutant non-small cell lung cancer cells
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2016, 卷号: 37, 期号: 12, 页码: 1587-1596
作者:
Wang, Yue-qin
;
Shen, Ai-jun
;
Sun, Jing-ya
;
Wang, Xin
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2019/01/08
non-small cell lung cancer
gefitinib resistance
Hsp90
Design, synthesis and biological evaluation of novel non-covalent piperidine-containing peptidyl proteasome inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 23, 页码: 6206-6214
作者:
Zhang, Jiankang
;
Gao, Lixin
;
Xi, Jianjun
;
Sheng, Li
;
Zhao, Yanmei
  |  
收藏
  |  
浏览/下载:51/0
  |  
提交时间:2019/01/08
Proteasome inhibitors
Piperidine
Non-covalent
Anti-cancer
SARs
DESIGN, SYNTHESIS, IN VITRO ANTIPROLIFERATIVE ACTIVITY EVALUATION OF 2-ALICANOYLAMIDOTHIOPHENE-3-CARBOXAMIDE DERIVATIVES
期刊论文
OAI收割
HETEROCYCLES, 2016, 卷号: 92, 期号: 12, 页码: 2145-2165
作者:
Zhang, Jiefeng
;
Guan, Fengjie
;
Qiu, Jiakun
;
Fang, Yanfen
;
Yu, Lifang
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收藏
  |  
浏览/下载:28/0
  |  
提交时间:2019/01/08
Identification and biochemical characterization of DC07090 as a novel potent small molecule inhibitor against human enterovirus 71 3C protease by structure-based virtual screening
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 124, 页码: 981-991
作者:
Ma, Guang-Hui
;
Ye, Yan
;
Zhang, Dan
;
Xu, Xin
;
Si, Pei
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2019/01/08
HFMD
EV71 3C(Pro)
Non-peptidyl inhibitor
Virtual screening
Potent Antitumor Activities and Structure Basis of the Chiral beta-Lactam Bridged Analogue of Combretastatin A-4 Binding to Tubulin
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 22, 页码: 10329-10334
作者:
Zhou, Pengfei
;
Liu, Yan
;
Zhou, Lu
;
Zhu, Kongkai
;
Feng, Kechang
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收藏
  |  
浏览/下载:21/0
  |  
提交时间:2019/01/08
16-nor Limonoids from Harrisonia perforata as promising selective 11 beta-HSD1 inhibitors
期刊论文
OAI收割
SCIENTIFIC REPORTS, 2016, 卷号: 6
作者:
Xiao-HuiYan
;
Yi, Ping
;
Cao, Pei
;
Yang, Shi-Ying
;
Fang, Xin
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2019/01/08
An Update on Poly(ADP-ribose)polymerase-1 (PARP-1) Inhibitors: Opportunities and Challenges in Cancer Therapy
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 21, 页码: 9575-9598
作者:
Wang, Ying-Qing
;
Wang, Ping-Yuan
;
Wang, Yu-Ting
;
Yang, Guang-Fu
;
Zhang, Ao
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2019/01/08