中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共5条,第1-5条 帮助

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Pharmacological characterization of TQ05310, a potent inhibitor of isocitrate dehydrogenase 2 R140Q and R172K mutants 期刊论文  OAI收割
CANCER SCIENCE, 2019, 页码: 9
作者:  
Gao, Mingzhao;  Zhu, Hongmei;  Fu, Li;  Li, Yun;  Bao, Xubin
  |  收藏  |  浏览/下载:29/0  |  提交时间:2020/07/01
AG-221  IDH2  leukemia  R140Q  R172K  
Discovery of DC_H31 as potential mutant IDH1 inhibitor through NADPH-based high throughput screening 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2019, 卷号: 27, 期号: 15, 页码: 3229-3236
作者:  
Duan, Zhe;  Liu, Jingqiu;  Niu, Liping;  Wang, Jun;  Feng, Mingqian
  |  收藏  |  浏览/下载:24/0  |  提交时间:2020/07/01
Synthesis and biological evaluation of 3-aryl-4-indolyl-maleimides as potent mutant isocitrate dehydrogenase-1 inhibitors 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2019, 卷号: 27, 期号: 4, 页码: 589-603
作者:  
Liu, Xiaoqi;  Hu, Yuanyuan;  Gao, Anhui;  Xu, Meng;  Gao, Lixin
  |  收藏  |  浏览/下载:22/0  |  提交时间:2020/07/01
3-(7-Azaindolyl)-4-indolylmaleimides as a novel class of mutant isocitrate dehydrogenase-1 inhibitors: Design, synthesis, and biological evaluation 期刊论文  OAI收割
ARCHIV DER PHARMAZIE, 2018, 卷号: 351, 期号: 10
作者:  
Hu, Yuanyuan;  Gao, Anhui;  Liao, Honghui;  Zhang, Mengmeng;  Xu, Gaoya
  |  收藏  |  浏览/下载:32/0  |  提交时间:2019/01/08
A New Breviane Spiroditerpenoid from the Marine-Derived Fungus Penicillium sp TJ403-1 期刊论文  OAI收割
MARINE DRUGS, 2018, 卷号: 16, 期号: 4, 页码: 110
作者:  
Yang, Beiye;  Sun, Weiguang;  Wang, Jianping;  Lin, Shuang;  Li, Xiao-Nian
  |  收藏  |  浏览/下载:35/0  |  提交时间:2018/07/02