中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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  • 上海药物研究所 [68]
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Epigenetic-based combination therapy and liposomal codelivery overcomes osimertinib-resistant NSCLC via repolarizing tumor-associated macrophages 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2023, 页码: 12
作者:  
Lin, Ting-ting;  Xiong, Wei;  Chen, Gui-hua;  He, Yang;  Long, Li
  |  收藏  |  浏览/下载:6/0  |  提交时间:2024/01/26
A first-in-human phase 1 study of simnotrelvir, a 3CL-like protease inhibitor for treatment of COVID-19, in healthy adult subjects 期刊论文  OAI收割
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2023, 卷号: 191, 页码: 9
作者:  
Yang, Xin-Mei;  Yang, Yang;  Yao, Bu-Fan;  Ye, Pan-Pan;  Xu, Yan
  |  收藏  |  浏览/下载:11/0  |  提交时间:2023/12/11
Versatile Biocatalytic C(sp(3))-H Oxyfunctionalization for the Site- Selective and Stereodivergent Synthesis of & alpha;- and & beta;-Hydroxy Acids 期刊论文  OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2023, 页码: 9
作者:  
Mao, Yingle;  Zhang, Weijie;  Fu, Zunyun;  Liu, Yanqiong;  Chen, Lin
  |  收藏  |  浏览/下载:18/0  |  提交时间:2023/10/17
Prime editing-based gene correction alleviates the hyperexcitable phenotype and seizures of a genetic epilepsy mouse model 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2023, 页码: 4
作者:  
Cao, Bi-rong;  Huang, Yi-ming;  Tian, Fu-yun;  Li, Jin-hui;  Xu, Chun-long
  |  收藏  |  浏览/下载:26/0  |  提交时间:2023/10/17
The PIWI-specific insertion module helps load longer piRNAs for translational activation essential for male fertility 期刊论文  OAI收割
SCIENCE CHINA-LIFE SCIENCES, 2023, 页码: 23
作者:  
Wang, Xin;  Lin, Di-Hang;  Yan, Yue;  Wang, An-Hui;  Liao, Jiaoyang
  |  收藏  |  浏览/下载:21/0  |  提交时间:2023/10/17
ETCM v2.0: An update with comprehensive resource and rich annotations for traditional Chinese medicine 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13, 期号: 6, 页码: 2559-2571
作者:  
Zhang, Yanqiong;  Li, Xin;  Shi, Yulong;  Chen, Tong;  Xu, Zhijian
  |  收藏  |  浏览/下载:21/0  |  提交时间:2023/10/17
A heterobifunctional molecule recruits cereblon to an RNA scaffold and activates its PROTAC function 期刊论文  OAI收割
CELL REPORTS PHYSICAL SCIENCE, 2022, 卷号: 3, 期号: 10, 页码: 12
作者:  
Xu, Yan;  Fu, Dingqiang;  Yuan, Yi;  Peng, Yan;  Dong, Juan
  |  收藏  |  浏览/下载:15/0  |  提交时间:2023/04/10

A novel aromatic amide derivative SY-65 co-targeted tubulin and histone deacetylase 1 with potent anticancer activity in vitro and in vivo

期刊论文  OAI收割

BIOCHEMICAL PHARMACOLOGY, 2022, 卷号: 201, 页码: 12
作者:  
Li, Yin-Ru;  Liu, Fang-Fang;  Liu, Wen-Bo;  Zhang, Yi-Fan;  Tian, Xin-Yi
  |  收藏  |  浏览/下载:24/0  |  提交时间:2022/08/16
A novel aromatic amide derivative SY-65 co-targeted tubulin and histone deacetylase 1 with potent anticancer activity in vitro and in vivo 期刊论文  OAI收割
BIOCHEMICAL PHARMACOLOGY, 2022, 卷号: 201, 页码: 115070
作者:  
Li, Yin-Ru;  Liu, Fang-Fang;  Liu, Wen-Bo;  Zhang, Yi-Fan;  Tian, Xin-Yi
  |  收藏  |  浏览/下载:10/0  |  提交时间:2024/03/21
Discovery of PHGDH inhibitors by virtual screening and preliminary structure-activity relationship study 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2022, 卷号: 121, 页码: 13
作者:  
  |  收藏  |  浏览/下载:22/0  |  提交时间:2022/06/15