机构

• 上海药物研究所 [8]

采集方式

• OAI收割 [8]

内容类型

• 期刊论文 [8]

发表日期

• 2023 [1]
• 2022 [1]
• 2021 [1]
• 2018 [1]
• 2017 [1]
• 2016 [1]
• 更多

学科主题

筛选

浏览/检索结果: 共8条，第1-8条 帮助 限定条件 专题：上海药物研究所    第一署名单位    第一作者单位    通讯作者单位     条数/页： 5101520253035404550556065707580859095100 排序方式： 请选择提交时间升序提交时间降序发表日期升序发表日期降序题名升序题名降序作者升序作者降序 Exploration of novel four-membered-heterocycle constructed peptidyl proteasome inhibitors with improved metabolic stability for cancer treatment 期刊论文  OAI收割 BIOORGANIC CHEMISTRY, 2023, 卷号: 138, 页码: 22 作者:  Wang, Hanlin;  Wu, Zhaoxiao;  Cao, Yu;  Gao, Lixin;  Shao, Jiaan   |  收藏  |  浏览/下载：13/0  |  提交时间：2023/10/17 Metabolic stability  Four-membered heterocycles  Proteasome inhibitors  Multiple myeloma   Metabolism guided optimization of peptidomimetics as non-covalent proteasome inhibitors for cancer treatment 期刊论文  OAI收割 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 233, 页码: 18 作者:  Cao, Yu;  Tu, Yutong;  Fu, Liping;  Yu, Qian;  Gao, Lixin   |  收藏  |  浏览/下载：27/0  |  提交时间：2022/06/15 Metabolism  Design  Proteasome inhibitors  Non-covalent  Multiple myeloma   Optimization of piperidine constructed peptidyl derivatives as proteasome inhibitors 期刊论文  OAI收割 BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 29, 页码: 14 作者:  Zhao, Yanmei;  Xu, Lei;  Zhang, Jiankang;  Zhang, Mengmeng;  Lu, Jingyi   |  收藏  |  浏览/下载：20/0  |  提交时间：2021/05/24 Proteasome inhibitor  Piperidine  Peptidyl  Anti-cancer  SAR   Development of Macrocyclic Peptides Containing Epoxyketone with Oral Availability as Proteasome Inhibitors 期刊论文  OAI收割 JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 20, 页码: 9177-9204 作者:  Li, Daqiang;  Zhang, Xiaotuan;  Ma, Xiaodong;  Xu, Lei;  Yu, Jianjun   |  收藏  |  浏览/下载：30/0  |  提交时间：2019/01/08 Exploration of novel piperazine or piperidine constructed non-covalent peptidyl derivatives as proteasome inhibitors 期刊论文  OAI收割 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 126, 页码: 1056-1070 作者:  Zhuang, Rangxiao;  Gao, Lixin;  Lv, Xiaoqing;  Xi, Jianjun;  Sheng, Li   |  收藏  |  浏览/下载：21/0  |  提交时间：2019/01/08 Proteasome inhibitors  Piperazine or piperidine  Non-covalent  Peptidyl derivatives  Anti-cancer   Design, synthesis and biological evaluation of novel non-covalent piperidine-containing peptidyl proteasome inhibitors 期刊论文  OAI收割 BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 23, 页码: 6206-6214 作者:  Zhang, Jiankang;  Gao, Lixin;  Xi, Jianjun;  Sheng, Li;  Zhao, Yanmei   |  收藏  |  浏览/下载：51/0  |  提交时间：2019/01/08 Proteasome inhibitors  Piperidine  Non-covalent  Anti-cancer  SARs   Design, Synthesis and Biological Evaluation of Peptidyl Epoxyketone Proteasome Inhibitors Composed of beta-amino Acids 期刊论文  OAI收割 CHEMICAL BIOLOGY & DRUG DESIGN, 2014, 卷号: 84, 期号: 5, 页码: 497-504 作者:  Zhang, Jiankang;  Han, Mengmeng;  Ma, Xiaodong;  Xu, Lei;  Cao, Jiayi   |  收藏  |  浏览/下载：15/0  |  提交时间：2019/01/08 anti-cancer  di- and tripeptides  epoxyketone  proteasome inhibitors  -amino acid   Design, synthesis and biological evaluation of novel tripeptidyl epoxyketone derivatives constructed from beta-amino acid as proteasome inhibitors 期刊论文  OAI收割 BIOORGANIC & MEDICINAL CHEMISTRY, 2014, 卷号: 22, 期号: 11, 页码: 2955-2965 作者:  Zhang, Jiankang;  Cao, Jiayi;  Xu, Lei;  Zhou, Yubo;  Liu, Tao   |  收藏  |  浏览/下载：11/0  |  提交时间：2019/01/08 Proteasome inhibitors  beta-Amino acid  Epoxyketone  Anti-cancer  Drug design  SARs