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  • 上海药物研究所 [3]
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Discovery, synthesis and mechanism study of 2,3,5-substituted [1,2,4]-thiadiazoles as covalent inhibitors targeting 3C-Like protease of SARS-CoV-2 期刊论文  OAI收割
European journal of medicinal chemistry, 2023, 卷号: 249, 页码: 115129
作者:  
Ren, Pengxuan;  Yu, Changyue;  Zhang, Ruxue;  Nie, Tianqing;  Hu, Qiaoyu
  |  收藏  |  浏览/下载:9/0  |  提交时间:2024/03/26
Rhodium(III)-Catalyzed C-H Alkenylation/Directing Group Migration for the Regio- and Stereoselective Synthesis of Tetrasubstituted Alkenes 期刊论文  OAI收割
ORGANIC LETTERS, 2020, 卷号: 22, 期号: 23, 页码: 9163-9168
作者:  
Wu, Xiaowei;  Lu, Yangbin;  Qiao, Jin;  Dai, Wenhao;  Jia, Xiuwen
  |  收藏  |  浏览/下载:13/0  |  提交时间:2021/05/24
Optimization of P2Y(12) Antagonist Ethyl 6-(4-((Benzylsulfonyl)carbarnoyl)piperidin-1-yl)-5-cyano-2-methylnicotinate (AZD1283) Led to the Discovery of an Oral Antiplatelet Agent with Improved Druglike Properties 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 6, 页码: 3088-3106
作者:  
Kong, Deyu;  Xue, Tao;  Guo, Bin;  Cheng, Jianjun;  Liu, Shunyin
  |  收藏  |  浏览/下载:11/0  |  提交时间:2020/07/01