中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [233]
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OAI收割 [233]
内容类型
期刊论文 [230]
会议论文 [3]
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2024 [4]
2023 [14]
2022 [24]
2021 [20]
2020 [28]
2019 [16]
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浏览/检索结果:
共233条,第1-10条
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专题:上海药物研究所
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Formyl phloroglucinol meroterpenoids from the leaves of
Eucalyptus
globulus
subsp.
maidenii
and their ATP-citrate lyase inhibitory activities
期刊论文
OAI收割
FITOTERAPIA, 2024, 卷号: 173, 页码: 6
作者:
Hu, Zhu
;
Liu, Yi-Nan
;
Yu, Mei-Hua
;
Hou, Ai -Jun
;
Li, Jing-Ya
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2024/03/13
Eucalyptus globulus subsp. maidenii
Meroterpenoids
ATP-citrate lyase
7-Dehydrocholesterol dictates ferroptosis sensitivity
期刊论文
OAI收割
NATURE, 2024, 卷号: 626, 期号: 7998, 页码: 29
作者:
Li, Yaxu
;
Ran, Qiao
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2024/04/09
Discovery of a potent and selective covalent threonine tyrosine kinase (TTK) inhibitor
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2024, 卷号: 143, 页码: 16
作者:
Sun, Yaoliang
;
Chen, Zhiwen
;
Liu, Guobin
;
Chen, Xiaoai
;
Shi, Zihan
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2024/03/25
Inhibitor
Cancer
Threonine tyrosine kinase (TTK)
Covalent
Safety, pharmacokinetics, and food effect of sudapyridine (WX-081), a novel anti-tuberculosis candidate in healthy Chinese subjects
期刊论文
OAI收割
CTS-CLINICAL AND TRANSLATIONAL SCIENCE, 2024, 卷号: 17, 期号: 2, 页码: 10
作者:
Yu, Chengyin
;
Qian, Hongjie
;
Wu, Qingqing
;
Zou, Yang
;
Ding, Qicheng
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2024/03/06
Development of a potent benzonitrile-based inhibitor of glutaminyl-peptide cyclotransferase-like protein (QPCTL) with antitumor efficacy
期刊论文
OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2023, 卷号: 8, 期号: 1, 页码: 3
作者:
Yu, Lei
;
Zhao, Pengcheng
;
Sun, Yaoliang
;
Zheng, Zening
;
Du, Wenhao
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2024/01/26
A first-in-human phase 1 study of simnotrelvir, a 3CL-like protease inhibitor for treatment of COVID-19, in healthy adult subjects
期刊论文
OAI收割
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2023, 卷号: 191, 页码: 9
作者:
Yang, Xin-Mei
;
Yang, Yang
;
Yao, Bu-Fan
;
Ye, Pan-Pan
;
Xu, Yan
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/12/11
COVID-19
Simnotrelvir
Safety
Pharmacokinetics
Healthy subjects
Natural product P57 induces hypothermia through targeting pyridoxal kinase
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 15
作者:
Wang, Ruina
;
Xiao, Lei
;
Pan, Jianbo
;
Bao, Guangsen
;
Zhu, Yunmei
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2024/02/19
Addition of a-synuclein aggregates to the intestinal environment recapitulates Parkinsonian symptoms in model systems
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2023, 页码: 16
作者:
Yang, Ze-xian
;
Zhang, Yu
;
Wang, Qing
;
Zhang, Lei
;
Liu, Yi-fei
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2023/12/08
Parkinson's disease
gut-brain axis
a-Synuclein
inflammation
microbiota
intestinal mouse coloclysis model
Ligand recognition and G protein coupling of the human itch receptor MRGPRX1
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 12
作者:
Guo, Lulu
;
Zhang, Yumu
;
Fang, Guoxing
;
Tie, Lu
;
Zhuang, Yuming
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2024/01/16
Repurposed Fenoprofen Targeting SaeR Attenuates Staphylococcus aureus Virulence in Implant-Associated Infections
期刊论文
OAI收割
ACS CENTRAL SCIENCE, 2023, 页码: 20
作者:
Jiang, Feng
;
Chen, Yingjia
;
Yu, Jinlong
;
Zhang, Feiyang
;
Liu, Qian
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2023/10/17